Induced protein degradation of anaplastic lymphoma kinase (ALK) by proteolysis targeting chimera (PROTAC) von Kang, Chung Hyo, Lee, Dong Ho, Lee, Chong Ock, Du Ha, Jae, Park, Chi Hoon, Hwang, Jong Yeon

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Design and characterization of cereblon-mediated androgen receptor proteolysis-targeting chimeras von Takwale, Akshay D., Jo, Seung-Hyun, Jeon, Yeong Uk, Kim, Hyung Soo, Shin, Choong Hoon, Lee, Heung Kyoung, Ahn, Sunjoo, Lee, Chong Ock, Du Ha, Jae, Kim, Jeong-Hoon, Hwang, Jong Yeon

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Combination Treatment with GSK126 and Pomalidomide Induces B-Cell Differentiation in EZH2 Gain-of-Function Mutant Diffuse Large B-Cell Lymphoma von Park, Sungryul, Jo, Seung-Hyun, Kim, Jong-Hwan, Kim, Seon-Young, Ha, Jae Du, Hwang, Jong Yeon, Lee, Myeong Youl, Kang, Jong Soon, Han, Tae-Su, Park, Sung Goo, Kim, Sunhong, Park, Byoung Chul, Kim, Jeong-Hoon

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Synthesis and biological evaluation of rhodanine derivatives as PRL-3 inhibitors von Ahn, Jin Hee, Kim, Seung Jun, Park, Woul Seong, Cho, Sung Yun, Ha, Jae Du, Kim, Sung Soo, Kang, Seung Kyu, Jeong, Dae Gwin, Jung, Suk-Kyeong, Lee, Sang-Hyeup, Kim, Hwan Mook, Park, Song Kyu, Lee, Ki Ho, Lee, Chang Woo, Ryu, Seong Eon, Choi, Joong-Kwon

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Augmentation of the antitumor effects of PARP inhibitors in triple-negative breast cancer via degradation by hydrophobic tagging modulation von Go, Ahra, Jang, Jeong Woon, Lee, Woori, Ha, Jae Du, Kim, Hyun Jin, Nam, Hye Jin

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Cereblon contributes to cardiac dysfunction by degrading Cav1.2α von Park, Nammi, Marquez, Jubert, Pham, Trong Kha, Ko, Tae Hee, Youm, Jae Boum, Kim, Min, Choi, Seung Hak, Moon, Jiyoung, Flores, Jessa, Ko, Kyung Soo, Rhee, Byoung Doo, Shimizu, Ippei, Minamino, Tohru, Ha, Jae Du, Hwang, Jong Yeon, Yang, Seung Joo, Park, Chul-Seung, Kim, Hyoung Kyu, Han, Jin

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A Novel Series of Highly Potent Small Molecule Inhibitors of Rhinovirus Replication von Kim, Jinwoo, Jung, Yu Kyoung, Kim, Chonsaeng, Shin, Jin Soo, Scheers, Els, Lee, Joo-Youn, Han, Soo Bong, Lee, Chong-Kyo, Neyts, Johan, Ha, Jae-Du, Jung, Young-Sik

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Synthesis and structure–activity relationship of aminopyridines with substituted benzoxazoles as c-Met kinase inhibitors von Lee, Jongkook, Han, Sun-Young, Jung, Heejung, Yang, Jeon, Choi, Jie-Won, Chae, Chong Hack, Park, Chi Hoon, Choi, Sang Un, Lee, Kwangho, Ha, Jae Du, Lee, Chong Ock, Ryu, Jae Wook, Kim, Hyoung Rae, Koh, Jong Sung, Cho, Sung Yun

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Disordered region of cereblon is required for efficient degradation by proteolysis-targeting chimera von Kim, Kidae, Lee, Dong Ho, Park, Sungryul, Jo, Seung-Hyun, Ku, Bonsu, Park, Sung Goo, Park, Byoung Chul, Jeon, Yeong Uk, Ahn, Sunjoo, Kang, Chung Hyo, Hwang, Daehee, Chae, Sehyun, Ha, Jae Du, Kim, Sunhong, Hwang, Jong Yeon, Kim, Jeong-Hoon

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Discovery of aminopyridines substituted with benzoxazole as orally active c-Met kinase inhibitors von Cho, Sung Yun, Han, Sun-Young, Ha, Jae Du, Ryu, Jae Wook, Lee, Chong Ock, Jung, Heejung, Kang, Nam Sook, Kim, Hyoung Rae, Koh, Jong Sung, Lee, Jongkook

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Synthesis and biological evaluation of N9-cis-cyclobutylpurine derivatives for use as cyclin-dependent kinase (CDK) inhibitors von Park, Sun Jun, Kim, Eunjin, Yoo, Miyoun, Lee, Joo-Youn, Park, Chi Hoon, Hwang, Jong Yeon, Ha, Jae Du

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Design and synthesis of triazolopyridazines substituted with methylisoquinolinone as selective c-Met kinase inhibitors von Ryu, Jae Wook, Han, Sun-Young, Yun, Jeong In, Choi, Sang-Un, Jung, Heejung, Ha, Jae Du, Cho, Sung Yun, Lee, Chong Ock, Kang, Nam Sook, Koh, Jong Sung, Kim, Hyoung Rae, Lee, Jongkook

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Replacing the terminal piperidine in ceritinib with aliphatic amines confers activities against crizotinib-resistant mutants including G1202R von Mathi, Gangadhar Rao, Kang, Chung Hyo, Lee, Heung Kyoung, Achary, Raghavendra, Lee, Ha-Yeon, Lee, Joo-Youn, Ha, Jae Du, Ahn, Sunjoo, Park, Chi Hoon, Lee, Chong Ock, Hwang, Jong Yeon, Yun, Chang-Soo, Jung, Hee Jung, Cho, Sung Yun, Kim, Hyoung Rae, Kim, Pilho

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Synthesis and evaluation of novel 2,4-diaminopyrimidines bearing bicyclic aminobenzazepines for anaplastic lymphoma kinase (ALK) inhibitor von Kang, Ga Ae, Lee, Minji, Song, Dawn, Lee, Heung Kyoung, Ahn, Sunjoo, Park, Chi Hoon, Lee, Chong Ock, Yun, Chang Soo, Jung, Heejung, Kim, Pilho, Ha, Jae Du, Cho, Sung Yun, Kim, Hyoung Rae, Hwang, Jong Yeon

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cIAPs promote the proteasomal degradation of mutant SOD1 linked to familial amyotrophic lateral sclerosis von Choi, Jin Sun, Kim, Kidae, Lee, Do Hee, Cho, Sayeon, Ha, Jae Du, Park, Byoung Chul, Kim, Sunhong, Park, Sung Goo, Kim, Jeong-Hoon

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4-Substituted quinazoline derivatives as novel EphA2 receptor tyrosine kinase inhibitors von Lim, Chae Jo, Oh, Kwang-Seok, Ha, Jae Du, Lee, Jeong Hyun, Seo, Ho Won, Chae, Chong Hack, Kim, Dae-Ghon, Lee, Mi-Jin, Lee, Byung Ho

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Therapeutic Efficacy of ABN401, a Highly Potent and Selective MET Inhibitor, Based on Diagnostic Biomarker Test in MET-Addicted Cancer von Kim, Jooseok, Park, Kyung Eui, Jeong, Yoo-Seong, Kim, YeongMun, Park, Hayeon, Nam, Ji-Hye, Jung, Kyungsoo, Son, Woo Sung, Jung, Hun Soon, Lee, Jong-Hwa, Jeong, Seong Hoon, Kim, Nam Ah, Ha, Jae Du, Cho, Sung Yun, Choi, Yoon-La, Chung, Suk-Jae, Choi, Jun Young, Hong, Sungyoul, Shin, Young Kee

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Design and synthesis of novel 3-(benzo[d]oxazol-2-yl)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine derivatives as selective G-protein-coupled receptor kinase-2 and -5 inhi... von Cho, Sung Yun, Lee, Byung Ho, Jung, Heejung, Yun, Chang Soo, Ha, Jae Du, Kim, Hyoung Rae, Chae, Chong Hak, Lee, Jeong Hyun, Seo, Ho Won, Oh, Kwang-Seok

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New Pyrimidine Derivatives possessing ALK Inhibitory Activities von Yang, Eun Hye, Yun, Jeong In, Latif, Muhammad, Lee, Hyeon Ji, Yun, Chang-Soo, Lee, Kwangho, Park, Chi Hoon, Cho, Sung Yun, Jung, Hee Jung, Kim, Pilho, Ha, Jae Du, Kim, Hyoung Rae

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Novel bis-ortho-alkoxy-para-piperazinesubstituted-2,4-dianilinopyrimidines (KRCA-0008) as potent and selective ALK inhibitors for anticancer treatment von Park, Chi Hoon, Choe, Hyeonjeong, Jang, In-Young, Kwon, So Yeong, Latif, Muhammad, Lee, Heung Kyoung, Lee, Hyeon Ji, Yang, Eun Hye, Yun, Jeong In, Chae, Chong Hak, Cho, Sung Yun, Choi, Sang Un, Ha, Jae Du, Jung, Heejung, Kim, Hyoung Rae, Kim, Pilho, Lee, Chong Ock, Yun, Chang-Soo, Lee, Kwangho

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