bioPROTACs as versatile modulators of intracellular therapeutic targets including proliferating cell nuclear antigen (PCNA) von Lim, Shuhui, Khoo, Regina, Peh, Khong Ming, Teo, Jinkai, Chang, Shih Chieh, Ng, Simon, Beilhartz, Greg L., Melnyk, Roman A., Johannes, Charles W., Brown, Christopher J., Lane, David P., Henry, Brian, Partridge, Anthony W.

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Design-rules for stapled peptides with in vivo activity and their application to Mdm2/X antagonists von Chandramohan, Arun, Josien, Hubert, Yuen, Tsz Ying, Duggal, Ruchia, Spiegelberg, Diana, Yan, Lin, Juang, Yu-Chi Angela, Ge, Lan, Aronica, Pietro G., Kaan, Hung Yi Kristal, Lim, Yee Hwee, Peier, Andrea, Sherborne, Brad, Hochman, Jerome, Lin, Songnian, Biswas, Kaustav, Nestor, Marika, Verma, Chandra S., Lane, David P., Sawyer, Tomi K., Garbaccio, Robert, Henry, Brian, Kannan, Srinivasaraghavan, Brown, Christopher J., Johannes, Charles W., Partridge, Anthony W.

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Natural product-like synthetic libraries von Thomas, Gemma L, Johannes, Charles W

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De Novo Sequencing of Synthetic Bis-cysteine Peptide Macrocycles Enabled by “Chemical Linearization” of Compound Mixtures von Chen, Zhi’ang, Lim, Yi Wee, Neo, Jin Yong, Ting Chan, Rachel Shu, Koh, Li Quan, Yuen, Tsz Ying, Lim, Yee Hwee, Johannes, Charles W., Gates, Zachary P.

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Synthesis of Chiral Alkenyl Cyclopropane Amino Acids for Incorporation into Stapled Peptides von Yuen, Tsz Ying, Brown, Christopher J, Tan, Yaw Sing, Johannes, Charles W

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Probabilistic Modelling of Geologically Complex Veins of the Barberton Greenstone Complex at Fairview Mine, South Africa von Mutobvu, Tyson, Pretorius, Hendrik, Muller, Charles Johannes, Mabala, Mahlomola Isaac

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Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles von Yuen, Tsz Ying, Brown, Christopher J, Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J, Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W, Verma, Chandra S, Lane, David P, Johannes, Charles W

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NanoClick: A High Throughput, Target-Agnostic Peptide Cell Permeability Assay von Peier, Andrea, Ge, Lan, Boyer, Nicolas, Frost, John, Duggal, Ruchia, Biswas, Kaustav, Edmondson, Scott, Hermes, Jeffrey D, Yan, Lin, Zimprich, Chad, Sadruddin, Ahmad, Kristal Kaan, Hung Yi, Chandramohan, Arun, Brown, Christopher J, Thean, Dawn, Lee, Xue Er, Yuen, Tsz Ying, Ferrer-Gago, Fernando J, Johannes, Charles W, Lane, David P, Sherborne, Brad, Corona, Cesear, Robers, Matthew B, Sawyer, Tomi K, Partridge, Anthony W

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A New Route to Bicyclo[1.1.1]pentan-1-amine from 1‑Azido-3-iodobicyclo[1.1.1]pentane von Goh, Yi Ling, Tam, Eric K.W, Bernardo, Paul H, Cheong, Choon Boon, Johannes, Charles W, William, Anthony D, Adsool, Vikrant A

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Macrocyclization of an all-d linear alpha-helical peptide imparts cellular permeability von Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Lian, Dawn Thean Gek, Frosi, Yuri, Chee, Sharon, Jiang, Shimin, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Renia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.

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Tandem oxidative amidation of benzyl alcohols with amine hydrochloride salts catalysed by iron nitrate von Ghosh, Subhash Chandra, Ngiam, Joyce S.Y., Seayad, Abdul M., Tuan, Dang Thanh, Johannes, Charles W., Chen, Anqi

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De-risking Drug Discovery of Intracellular Targeting Peptides: Screening Strategies to Eliminate False-Positive Hits von Ng, Simon, Juang, Yu-Chi, Chandramohan, Arun, Kaan, Hung Yi Kristal, Sadruddin, Ahmad, Yuen, Tsz Ying, Ferrer-Gago, Fernando J, Lee, Xue’Er Cheryl, Liew, Xi, Johannes, Charles W, Brown, Christopher J, Kannan, Srinivasaraghavan, Aronica, Pietro G, Berglund, Nils A, Verma, Chandra S, Liu, Lijuan, Stoeck, Alexander, Sawyer, Tomi K, Partridge, Anthony W, Lane, David P

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A Versatile and Efficient Palladium-meta-Terarylphosphine Catalyst for the Copper-Free Sonogashira Coupling of (Hetero-)Aryl Chlorides and Alkynes von Yang, Yong, Chew, Xinying, Johannes, Charles W., Robins, Edward G., Jong, Howard, Lim, Yee Hwee

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Direct Conversion of Indoles to 3,3-Difluoro-2-oxindoles via Electrophilic Fluorination von Lim, Yee Hwee, Ong, Qunxiang, Duong, Hung A, Nguyen, Tuan Minh, Johannes, Charles W

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An intramolecular tryptophan-condensation approach for peptide stapling von Hui, Eunice Y-L, Rout, Bhimsen, Tan, Yaw Sing, Verma, Chandra S, Chan, Kok-Ping, Johannes, Charles W

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Palladium-meta-Terarylphosphine Catalyst for the Mizoroki–Heck Reaction of (Hetero)Aryl Bromides and Functional Olefins von Tay, Daniel Weiliang, Jong, Howard, Lim, Yee Hwee, Wu, Wenqin, Chew, Xinying, Robins, Edward G, Johannes, Charles W

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Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties von Partridge, Anthony W, Kaan, Hung Yi Kristal, Juang, Yu-Chi, Sadruddin, Ahmad, Lim, Shuhui, Brown, Christopher J, Ng, Simon, Thean, Dawn, Ferrer, Fernando, Johannes, Charles, Yuen, Tsz Ying, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Pradhan, Mohan R, Verma, Chandra S, Hochman, Jerome, Chen, Shiying, Wan, Hui, Ha, Sookhee, Sherborne, Brad, Lane, David P, Sawyer, Tomi K

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Discovery of cell active macrocyclic peptides with on-target inhibition of KRAS signaling von Lim, Shuhui, Boyer, Nicolas, Boo, Nicole, Huang, Chunhui, Venkatachalam, Gireedhar, Angela Juang, Yu-Chi, Garrigou, Michael, Kaan, Hung Yi Kristal, Duggal, Ruchia, Peh, Khong Ming, Sadruddin, Ahmad, Gopal, Pooja, Yuen, Tsz Ying, Ng, Simon, Kannan, Srinivasaraghavan, Brown, Christopher J, Verma, Chandra S, Orth, Peter, Peier, Andrea, Ge, Lan, Yu, Xiang, Bhatt, Bhavana, Chen, Feifei, Wang, Erjia, Li, Nianyu Jason, Gonzales, Raymond J, Stoeck, Alexander, Henry, Brian, Sawyer, Tomi K, Lane, David P, Johannes, Charles W, Biswas, Kaustav, Partridge, Anthony W

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Mechanistic Insights and Implications of Dearomative Rearrangement in Copper-Free Sonogashira Cross-Coupling Catalyzed by Pd-CyPhine von Mak, Adrian M, Lim, Yee Hwee, Jong, Howard, Yang, Yong, Johannes, Charles W, Robins, Edward G, Sullivan, Michael B

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Stitched peptides as potential cell permeable inhibitors of oncogenic DAXX protein von Jelinska, Clare, Kannan, Srinivasaraghavan, Frosi, Yuri, Ramlan, Siti Radhiah, Winnerdy, Fernaldo, Lakshminarayanan, Rajamani, Johannes, Charles W, Brown, Christopher J, Phan, Anh-Tuan, Rhodes, Daniela, Verma, Chandra S

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