Discovery of Novel Urea-Based Hepatitis C Protease Inhibitors with High Potency against Protease-Inhibitor-Resistant Mutants von Kazmierski, Wieslaw M, Hamatake, Robert, Duan, Maosheng, Wright, Lois L, Smith, Gary K, Jarvest, Richard L, Ji, Jing-Jing, Cooper, Joel P, Tallant, Matthew D, Crosby, Renae M, Creech, Katrina, Wang, Amy, Li, Xianfeng, Zhang, Suoming, Zhang, Yong-Kang, Liu, Yang, Ding, Charles Z, Zhou, Yasheen, Plattner, Jacob J, Baker, Stephen J, Bu, Wei, Liu, Liang

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Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties von Li, Xianfeng, Zhang, Suoming, Zhang, Yong-Kang, Liu, Yang, Ding, Charles Z., Zhou, Yasheen, Plattner, Jacob J., Baker, Stephen J., Bu, Wei, Liu, Liang, Kazmierski, Wieslaw M., Duan, Maosheng, Grimes, Richard M., Wright, Lois L., Smith, Gary K., Jarvest, Richard L., Ji, Jing-Jing, Cooper, Joel P., Tallant, Matthew D., Crosby, Renae M., Creech, Katrina, Ni, Zhi-Jie, Zou, Wuxin, Wright, Jon

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A Peroxisome Proliferator-Activated Receptor γ Ligand Inhibits Adipocyte Differentiation von Oberfield, Jennifer L., Collins, Jon L., Holmes, Christopher P., Goreham, Donna M., Cooper, Joel P., Cobb, Jeffery E., Lenhard, James M., Hull-Ryde, Emily A., Mohr, Christopher P., Blanchard, Steven G., Parks, Derek J., Moore, Linda B., Lehmann, Jürgen M., Plunket, Kelli, Miller, Ann B., Milburn, Michael V., Kliewer, Steven A., Willson, Timothy M.

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Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease von Li, Xianfeng, Zhang, Yong-Kang, Liu, Yang, Zhang, Suoming, Ding, Charles Z., Zhou, Yasheen, Plattner, Jacob J., Baker, Stephen J., Liu, Liang, Bu, Wei, Kazmierski, Wieslaw M., Wright, Lois L., Smith, Gary K., Jarvest, Richard L., Duan, Maosheng, Ji, Jing-Jing, Cooper, Joel P., Tallant, Matthew D., Crosby, Renae M., Creech, Katrina, Ni, Zhi-Jie, Zou, Wuxin, Wright, Jon

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Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groups von Li, Xianfeng, Liu, Yang, Zhang, Yong-Kang, Plattner, Jacob J., Baker, Stephen J., Bu, Wei, Liu, Liang, Zhou, Yasheen, Ding, Charles Z., Zhang, Suoming, Kazmierski, Wieslaw M., Hamatake, Robert, Duan, Maosheng, Wright, Lois L., Smith, Gary K., Jarvest, Richard L., Ji, Jing-Jing, Cooper, Joel P., Tallant, Matthew D., Crosby, Renae M., Creech, Katrina, Wang, Amy

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Anthranilimide based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes. Part 3: X-ray crystallographic characterization, core and urea optimization and in vivo... von Thomson, Stephen A., Banker, Pierette, Bickett, D. Mark, Boucheron, Joyce A., Carter, H. Luke, Clancy, Daphne C., Cooper, Joel P., Dickerson, Scott H., Garrido, Dulce M., Nolte, Robert T., Peat, Andrew J., Sheckler, Lauren R., Sparks, Steven M., Tavares, Francis X., Wang, Liping, Wang, Tony Y., Weiel, James E.

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The discovery and optimization of pyrimidinone-containing MCH R1 antagonists von Hertzog, Donald L., Al-Barazanji, Kamal A., Bigham, Eric C., Bishop, Michael J., Britt, Christy S., Carlton, David L., Cooper, Joel P., Daniels, Alex J., Garrido, Dulce M., Goetz, Aaron S., Grizzle, Mary K., Guo, Yu C., Handlon, Anthony L., Ignar, Diane M., Morgan, Ronda O., Peat, Andrew J., Tavares, Francis X., Zhou, Huiqiang

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Novel benzimidazole-based MCH R1 antagonists von Carpenter, Andrew J., Al-Barazanji, Kamal A., Barvian, Kevin K., Bishop, Michael J., Britt, Christy S., Cooper, Joel P., Goetz, Aaron S., Grizzle, Mary K., Hertzog, Donald L., Ignar, Diane M., Morgan, Ronda O., Peckham, Gregory E., Speake, Jason D., Swain, Will R.

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N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 3. Structure−Activity Relationship and Optimization of the N-Aryl Substituent von Cobb, Jeff E, Blanchard, Steven G, Boswell, Evan G, Brown, Kathleen K, Charifson, Paul S, Cooper, Joel P, Collins, Jon L, Dezube, Milana, Henke, Brad R, Hull-Ryde, Emily A, Lake, Debra H, Lenhard, James M, Oliver, William, Oplinger, Jeffery, Pentti, Mila, Parks, Derek J, Plunket, Kelli D, Tong, Wei-Qin

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6-(4-Chlorophenyl)-3-substituted-thieno[3,2-d]pyrimidin-4(3H)-one-Based Melanin-Concentrating Hormone Receptor 1 Antagonist von Tavares, Francis X, Al-Barazanji, Kamal A, Bishop, Michael J, Britt, Christy S, Carlton, David L, Cooper, Joel P, Feldman, Paul L, Garrido, Dulce M, Goetz, Aaron S, Grizzle, Mary K, Hertzog, Donald L, Ignar, Diane M, Lang, Daniel G, McIntyre, Maggie S, Ott, Ronda J, Peat, Andrew J, Zhou, Hui-Qiang

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Peptide and Peptide Mimetic Inhibitors of Antigen Presentation by HLA-DR Class II MHC Molecules. Design, Structure−Activity Relationships, and X-ray Crystal Structures von Bolin, David R, Swain, Amy L, Sarabu, Ramakanth, Berthel, Steven J, Gillespie, Paul, Huby, Nicholas J. S, Makofske, Raymond, Orzechowski, Lucja, Perrotta, Agostino, Toth, Katherine, Cooper, Joel P, Jiang, Nan, Falcioni, Fiorenza, Campbell, Robert, Cox, Donald, Gaizband, Diana, Belunis, Charles J, Vidovic, Damir, Ito, Kouichi, Crowther, Robert, Kammlott, Ursula, Zhang, Xiaolei, Palermo, Robert, Weber, David, Guenot, Jeanmarie, Nagy, Zoltan, Olson, Gary L

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Highly selective heterogeneous palladium-catalyzed hydrogenations using triethoxysilane and water von Tour, James M, Cooper, Joel P, Pendalwar, Shekhar L

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Homogeneous deposition of palladium(0) into sol-gel-derived materials von Tour, James M, Pendalwar, Shekhar L, Cooper, Joel P

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Oxazole- and imidazole-based Ser-Leu dipeptide mimetics in potent inhibitors of antigen presentation by MHC class II DR molecules von SARABU, Ramakanth, BOLIN, David R, CAMPBELL, Robert, COOPER, Joel P, COX, Donald, GAIZBAND, Diana, MAKOFSKE, Raymond, NAGY, Zoltan, OLSON, Gary L

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Dispersion of Rh/Cu in a sol-gel matrix. Highly chemo- and stereoselective catalyst for the reduction of alkynes to Z-alkenes von Tour, James M, Pendalwar, Shekhar L, Kafka, Cynthia M, Cooper, Joel P

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Oxazole- and Imidazole-Based Ser-Leu Dipeptide Mimetics in Potent Inhibitors of Antigen Presentation by MHC Class II DR Molecules von Sarabu, Ramakanth, Bolin, David R., Campbell, Robert, Cooper, Joel P., Cox, Donald, Gaizband, Diana, Makofske, Raymond, Nagy, Zoltan, Olson, Gary L.

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COMPOUNDS von GRIMES, RICHARD MARTIN, DUAN, MAOSHENG, KAZMIERSKI, WIESLAW MIECZYSLAW, COOPER, JOEL P, TALLANT, MATTHEW D

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COMPOUNDS von GRIMES, RICHARD MARTIN, DUAN, MAOSHENG, KAZMIERSKI, WIESLAW MIECZYSLAW, COOPER, JOEL P, TALLANT, MATTHEW D

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COMPOUNDS von GRIMES, RICHARD MARTIN, DUAN, MAOSHENG, KAZMIERSKI, WIESLAW MIECZYSLAW, COOPER, JOEL P, TALLANT, MATTHEW D

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CHEMICAL COMPOUNDS von BASKARAN, SUBRAMANIAN, MCFADYEN, ROBERT BLOUNT, BOTYANSZKI, JANOS, REDMAN, ANIKO, DUAN, MAOSHENG, KAZMIERSKI, WIESLAW MIECZYSLAW, COOPER, JOEL P

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