Isothiourea-Catalyzed Enantioselective Carboxy Group Transfer von Joannesse, Caroline, Johnston, Craig P, Concellón, Carmen, Simal, Carmen, Philp, Douglas, Smith, Andrew D

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Discovery of N‑(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro‑4H‑thieno[2,3‑c]pyran-2-yl)‑lH‑pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mutant Cy... von Van der Plas, Steven E, Kelgtermans, Hans, De Munck, Tom, Martina, Sébastien L. X, Dropsit, Sébastien, Quinton, Evelyne, De Blieck, Ann, Joannesse, Caroline, Tomaskovic, Linda, Jans, Mia, Christophe, Thierry, van der Aar, Ellen, Borgonovi, Monica, Nelles, Luc, Gees, Maarten, Stouten, Pieter, Van Der Schueren, Jan, Mammoliti, Oscar, Conrath, Katja, Andrews, Martin

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Structure-enantioselectivity effects in 3,4-dihydropyrimido[2,1-b]benzothiazole-based isothioureas as enantioselective acylation catalysts von Belmessieri, Dorine, Joannesse, Caroline, Woods, Philip A, MacGregor, Callum, Jones, Caroline, Campbell, Craig D, Johnston, Craig P, Duguet, Nicolas, Concellón, Carmen, Bragg, Ryan A, Smith, Andrew D

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Regiodivergent Lewis base-promoted O- to C-carboxyl transfer of furanyl carbonates von Campbell, Craig D, Joannesse, Caroline, Morrill, Louis C, Philp, Douglas, Smith, Andrew D

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Isothiourea-Mediated Asymmetric O- to C-Carboxyl Transfer of Oxazolyl Carbonates: Structure-Selectivity Profiles and Mechanistic Studies von Joannesse, Caroline, Johnston, Craig P., Morrill, Louis C., Woods, Philip A., Kieffer, Madeleine, Nigst, Tobias A., Mayr, Herbert, Lebl, Tomas, Philp, Douglas, Bragg, Ryan A., Smith, Andrew D.

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Design of a potent and selective dual JAK1/TYK2 inhibitor von Mammoliti, Oscar, Menet, Christel, Cottereaux, Céline, Blanc, Javier, De Blieck, Ann, Coti, Ghjuvanni, Geney, Raphaël, Oste, Line, Ostyn, Koen, Palisse, Adeline, Quinton, Evelyne, Schmitt, Benoit, Borgonovi, Monica, Parent, Isabelle, Jagerschmidt, Catherine, De Vos, Steve, Vayssiere, Béatrice, López-Ramos, Miriam, Shoji, Kenji, Brys, Reginald, Amantini, David, Galien, René, Joannesse, Caroline

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Discovery of the S1P2 Antagonist GLPG2938 (1-[2-Ethoxy-6-(trifluoromethyl)-4-pyridyl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea), a Precli... von Mammoliti, Oscar, Palisse, Adeline, Joannesse, Caroline, El Bkassiny, Sandy, Allart, Brigitte, Jaunet, Alex, Menet, Christel, Coornaert, Beatrice, Sonck, Kathleen, Duys, Inge, Clément-Lacroix, Philippe, Oste, Line, Borgonovi, Monica, Wakselman, Emanuelle, Christophe, Thierry, Houvenaghel, Nicolas, Jans, Mia, Heckmann, Bertrand, Sanière, Laurent, Brys, Reginald

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Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis von Van der Plas, Steven E, Kelgtermans, Hans, Mammoliti, Oscar, Menet, Christel, Tricarico, Giovanni, De Blieck, Ann, Joannesse, Caroline, De Munck, Tom, Lambin, Dominique, Cowart, Marlon, Dropsit, Sebastien, Martina, Sebastien L X, Gees, Maarten, Wesse, Anne-Sophie, Conrath, Katja, Andrews, Martin

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Correction to “Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis” von Van der Plas, Steven E, Kelgtermans, Hans, Mammoliti, Oscar, Menet, Christel, Tricarico, Giovanni, De Blieck, Ann, Joannesse, Caroline, De Munck, Tom, Lambin, Dominique, Cowart, Marlon, Dropsit, Sebastien, Martina, Sebastien L. X, Gees, Maarten, Wesse, Anne-Sophie, Conrath, Katja, Andrews, Martin

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Nucleophilicities and Lewis Basicities of Isothiourea Derivatives von Maji, Biplab, Joannesse, Caroline, Nigst, Tobias A, Smith, Andrew D, Mayr, Herbert

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Regiodivergent Lewis base-promoted O- to C-carboxyl transfer of furanyl carbonatesElectronic supplementary information (ESI) available: Full experimental procedures and characteris... von Campbell, Craig D, Joannesse, Caroline, Morrill, Louis C, Philp, Douglas, Smith, Andrew D

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Discovery of N -(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro-4 H -thieno[2,3- c ]pyran-2-yl)-l H -pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mu... von Van der Plas, Steven E., Kelgtermans, Hans, De Munck, Tom, Martina, Sébastien L. X., Dropsit, Sébastien, Quinton, Evelyne, De Blieck, Ann, Joannesse, Caroline, Tomaskovic, Linda, Jans, Mia, Christophe, Thierry, van der Aar, Ellen, Borgonovi, Monica, Nelles, Luc, Gees, Maarten, Stouten, Pieter, Van Der Schueren, Jan, Mammoliti, Oscar, Conrath, Katja, Andrews, Martin

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Amidine catalysed O- to C-carboxyl transfer of heterocyclic carbonate derivatives von Joannesse, Caroline, Simal, Carmen, Concellón, Carmen, Thomson, Jennifer E, Campbell, Craig D, Slawin, Alexandra M Z, Smith, Andrew D

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Structure-enantioselectivity effects in 3,4-dihydropyrimido[2,1-b]benzothiazole-based isothioureas as enantioselective acylation catalystsElectronic supplementary information (ESI)... von Belmessieri, Dorine, Joannesse, Caroline, Woods, Philip A, MacGregor, Callum, Jones, Caroline, Campbell, Craig D, Johnston, Craig P, Duguet, Nicolas, Concellón, Carmen, Bragg, Ryan A, Smith, Andrew D

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Isothiourea-Catalyzed Enantioselective Carboxy Group Transfer von Joannesse, Caroline, Johnston, Craig P., Concellón, Carmen, Simal, Carmen, Philp, Douglas, Smith, Andrew D.

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2-OXO-5H-CHROMENO[4,3-B]PYRIDINES FOR USE IN THE TREATMENT OF HEPATITIS B von JOANNESSE, Caroline, Martine, Andrée, Marie, JAUNET, Alexis, Patrick, Claude, CATANA, Cornel, DUTHION, Béranger, LARUELLE, Chris, Ronan, DE BLIECK, Ann, MAMMOLITI, Oscar, VAN DER PLAS, Steven, Emiel, DE MUNCK, Tom, Roger, Lisette, PALISSE, Adeline, Marie, Elise

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NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS von EL BKASSINY, Sandy, ALLART, Brigitte, MAMMOLITI, Oscar, JANSEN, Koen, Karel, PALISSE, Adeline, Marie, Elise, MENET, Christel, Jeanne, Marie, JOANNESSE, Caroline, Martine, Andrée-Marie

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NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS von EL BKASSINY, Sandy, ALLART, Brigitte, MENET, Christel Jeanne Marie, MAMMOLITI, Oscar, JANSEN, Koen Karel, JOANNESSE, Caroline Martine Andrée Marie, PALISSE, Adeline Marie Elise

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2-OXO-5H-CHROMENO[4,3-B]PYRIDINES FOR USE IN THE TREATMENT OF HEPATITIS B von JOANNESSE, Caroline, Martine, Andrée, Marie, JAUNET, Alexis, Patrick, Claude, CATANA, Cornel, DUTHION, Béranger, LARUELLE, Chris, Ronan, DE BLIECK, Ann, MAMMOLITI, Oscar, VAN DER PLAS, Steven, Emiel, DE MUNCK, Tom, Roger, Lisette, PALISSE, Adeline, Marie, Elise

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NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS von JANSEN, Koen, PALISSE, Adeline, EL BKASSINY, Sandy, JOANNESSE, Caroline, ALLART, Brigitte, MAMMOLITI, Oscar, MENET, Christel

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