Orexin-1 and orexin-2 receptor antagonists reduce ethanol self-administration in high-drinking rodent models von Anderson, Rachel I, Becker, Howard C, Adams, Benjamin L, Jesudason, Cynthia D, Rorick-Kehn, Linda M

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Selective Phosphodiesterase 1 Inhibitor BTTQ Reduces Blood Pressure in Spontaneously Hypertensive and Dahl Salt Sensitive Rats: Role of Peripheral Vasodilation von Dey, Asim B., Khedr, Sherif, Bean, James, Porras, Leah L., Meredith, Tamika D., Willard, Francis S., Hass, Joseph V., Zhou, Xin, Terashvili, Maia, Jesudason, Cynthia D., Ruley, Kevin M., Wiley, Michael R., Kowala, Mark, Atkinson, Simon J., Staruschenko, Alexander, Rekhter, Mark D.

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SHIP1 therapeutic target enablement: Identification and evaluation of inhibitors for the treatment of late‐onset Alzheimer's disease von Jesudason, Cynthia D., Mason, Emily R., Chu, Shaoyou, Oblak, Adrian L., Javens‐Wolfe, June, Moussaif, Mustapha, Durst, Greg, Hipskind, Philip, Beck, Daniel E., Dong, Jiajun, Amarasinghe, Ovini, Zhang, Zhong‐Yin, Hamdani, Adam K., Singhal, Kratika, Mesecar, Andrew D., Souza, Sarah, Jacobson, Marlene, Salvo, Jerry Di, Soni, Disha M., Kandasamy, Murugesh, Masters, Andrea R., Quinney, Sara K, Doolen, Suzanne, Huhe, Hasi, Rizzo, Stacey J. Sukoff, Lamb, Bruce T., Palkowitz, Alan D., Richardson, Timothy I.

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LSN2424100: a novel, potent orexin-2 receptor antagonist with selectivity over orexin-1 receptors and activity in an animal model predictive of antidepressant-like efficacy von Fitch, Thomas E, Benvenga, Mark J, Jesudason, Cynthia D, Zink, Charity, Vandergriff, Amy B, Menezes, Michelle M, Schober, Douglas A, Rorick-Kehn, Linda M

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The First Synthesis of a Daphnane Diterpene:  The Enantiocontrolled Total Synthesis of (+)-Resiniferatoxin von Wender, Paul A, Jesudason, Cynthia D, Nakahira, Hiroyuki, Tamura, Norikazu, Tebbe, Anne Louise, Ueno, Yoshihide

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Synthesis and SAR of novel histamine H3 receptor antagonists von Jesudason, Cynthia D., Beavers, Lisa S., Cramer, Jeffrey W., Dill, Joelle, Finley, Don R., Lindsley, Craig W., Stevens, F. Craig, Gadski, Robert A., Oldham, Samuel W., Pickard, R. Todd, Siedem, Christopher S., Sindelar, Dana K., Singh, Ajay, Watson, Brian M., Hipskind, Philip A.

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Combination of a Beta Adrenoceptor Modulator and a Norepinephrine-Serotonin Uptake Inhibitor for the Treatment of Obesity von Jesudason, Cynthia D., Baker, James E., Bryant, Robert D., Fisher, Jack W., O’Farrell, Libbey S., Gaich, Gregory A., He, Minxia M., Kahl, Steven D., Kriauciunas, Aidas V., Heiman, Mark L., Peters, Mary A., Rito, Christopher J., Satterwhite, Julie H., Tinsley, Frank C., Trankle, William G., Shuker, Anthony J.

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Potent oxindole based human β3 adrenergic receptor agonists von STEVENS, F. Craig, BLOOMQUIST, William E, BOREL, Anthony G, COHEN, Marlene L, DROSTE, Christine A, HEIMAN, Mark L, KRIAUCIUNAS, Aidas, SALL, Daniel J, TINSLEY, Frank C, JESUDASON, Cynthia D

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SHIP1 phosphatase as a Late‐Onset Alzheimer’s Disease therapeutic target von Singhal, Kratika, Hamdani, Adam K, Jesudason, Cynthia D, Beck, Daniel E, Clayton, Brent, Richardson, Timothy I., Mesecar, Andrew D.

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Optimization of SHIP1 Inhibitors for the treatment of Alzheimer’s disease von Jesudason, Cynthia D, Lin, Peter Bor‐Chian, Soni, Disha, Perkins, Bridget M, Lee‐Gosselin, Audrey, Ingraham, Cynthia M, Hamilton, Will, Mason, Emily R, Jordi, Omar El, Souza, Sarah, Jacobson, Marlene, Salvo, Jerry Di, Clayton, Brent, Chu, Shaoyou, Dage, Jeffrey L., Oblak, Adrian L, Richardson, Timothy I.

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Potent benzimidazolone based human beta(3)-adrenergic receptor agonists von Finley, Don R, Bell, Michael G, Borel, Anthony G, Bloomquist, William E, Cohen, Marlene L, Heiman, Mark L, Kriauciunas, Aidas, Matthews, Donald P, Miles, Tania, Neel, David A, Rito, Christopher J, Sall, Daniel J, Shuker, Anthony J, Stephens, Thomas W, Tinsley, Frank C, Winter, Mark A, Jesudason, Cynthia D

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Potent benzimidazolone based human β3-adrenergic receptor agonists von FINLEY, Don R, BELL, Michael G, RITO, Christopher J, SAIL, Daniel J, SHUKER, Anthony J, STEPHENS, Thomas W, TINSLEY, Frank C, WINTER, Mark A, JESUDASON, Cynthia D, BOREL, Anthony G, BLOOMQUIST, William E, COHEN, Marlene L, HEIMAN, Mark. L, KRIAUCIUNAS, Aidas, MATTHEWS, Donald P, MILES, Tania, NEEL, David A

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A Target Enablement Package for the Inhibition of SHIP1 as a Therapeutic Strategy for the Treatment of Alzheimer’s Disease von Richardson, Timothy I, Jesudason, Cynthia D, Lobb, Karen L, Durst, Gregory L, Clayton, Brent, Massey, Steven M, Beck, Daniel E, Zhang, Zhong‐Yin, Dong, Jiajun, Lin, Jianping, Miao, Jinmin, Putt, Karson S, Mesecar, Andrew D, Hamdani, Adam K, Lendy, Emma K, Souza, Sarah, Jacobson, Marlene, Salvo, Jerry Di, Chu, Shaoyou, Mason, Emily R, Oblak, Adrian L, Soni, Disha, Quinney, Sara K, Silva, Larissa L, Kandasamy, Murugesh, Masters, Andrea R, Rizzo, Stacey J Sukoff, Doolen, Suzanne, Huang, Kun, Zhang, Jie, Lamb, Bruce T, Palkowitz, Alan D

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The use of high-throughput synthesis and purification in the preparation of a directed library of adrenergic agents von Siegel, M G, Shuker, A J, Droste, C A, Hahn, P J, Jesudason, C D, McDonald, 3rd, J H, Matthews, D P, Rito, C J, Thorpe, A J

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Potent oxindole based human beta sub(3) adrenergic receptor agonists von Stevens, FCraig, Bloomquist, William E, Borel, Anthony G, Cohen, Marlene L, Droste, Christine A, Heiman, Mark L, Kriauciunas, Aidas, Sall, Daniel J, Tinsley, Frank C, Jesudason, Cynthia D

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Potent oxindole based human beta3 adrenergic receptor agonists von Stevens, F Craig, Bloomquist, William E, Borel, Anthony G, Cohen, Marlene L, Droste, Christine A, Heiman, Mark L, Kriauciunas, Aidas, Sall, Daniel J, Tinsley, Frank C, Jesudason, Cynthia D

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Potent oxindole based human β 3 adrenergic receptor agonists von Stevens, F. Craig, Bloomquist, William E., Borel, Anthony G., Cohen, Marlene L., Droste, Christine A., Heiman, Mark L., Kriauciunas, Aidas, Sall, Daniel J., Tinsley, Frank C., Jesudason, Cynthia D.

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Synthesis and SAR of novel histamine H sub(3) receptor antagonists von Jesudason, Cynthia D, Beavers, Lisa S, Cramer, Jeffrey W, Dill, Joelle, Finley, Don R, Lindsley, Craig W, Stevens, FCraig, Gadski, Robert A, Oldham, Samuel W, Pickard, RTodd, Siedem, Christopher S, Sindelar, Dana K, Singh, Ajay, Watson, Brian M, Hipskind, Philip A

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Potent benzimidazolone based human beta sub(3)-adrenergic receptor agonists von Finley, Don R, Bell, Michael G, Borel, Anthony G, Bloomquist, William E, Cohen, Marlene L, Heiman, MarkL, Kriauciunas, Aidas, Matthews, Donald P, Miles, Tania, Neel, David A, Rito, Christopher J, Sall, Daniel J, Shuker, Anthony J, Stephens, Thomas W, Tinsley, Frank C, Winter, Mark A, Jesudason, Cynthia D

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Potent benzimidazolone based human β 3-adrenergic receptor agonists von Finley, Don R., Bell, Michael G., Borel, Anthony G., Bloomquist, William E., Cohen, Marlene L., Heiman, Mark. L., Kriauciunas, Aidas, Matthews, Donald P., Miles, Tania, Neel, David A., Rito, Christopher J., Sall, Daniel J., Shuker, Anthony J., Stephens, Thomas W., Tinsley, Frank C., Winter, Mark A., Jesudason, Cynthia D.

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