Intestinal serine protease inhibition increases FGF21 and improves metabolism in obese mice von Albarazanji, Kamal, Jennis, Matthew, Cavanaugh, Cassandre R, Lang, Wensheng, Singh, Bhanu, Lanter, James C, Lenhard, James M, Hornby, Pamela J

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Discovery of quinuclidine modulators of cellular progranulin von Lanter, James C., Chen, Angela Y.-P., Williamson, Toni, Koenig, Gerhard, Blain, Jean-François, Burnett, Duane A.

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Discovery of oxazoline enhancers of cellular progranulin release von Peng, Xiaowen, Lanter, James C., Y.-P. Chen, Angela, Brand, Morgan A., Wozniak, Mary K., Hoekman, Steven, Longin, Ondřej, Regeling, Hendrik, Zonneveld, Wim, P. L. Bell, Roel, Koenig, Gerhard, Hurst, Raymond S., Blain, Jean-François, Burnett, Duane A.

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Discovery and characterization of novel TRPML1 agonists von Peng, Xiaowen, Holler, Christopher J., Alves, Anna-Maria F., Oliviera, Michelle G., Speake, Michael, Pugliese, Angelo, Oskouei, Mina R., de Freitas, Ivan D., Chen, Angela Y.-P., Gallegos, Richard, McTighe, Stephanie M., Koenig, Gerhard, Hurst, Raymond S., Blain, Jean-François, Lanter, James C., Burnett, Duane A.

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Direct dehydrative cross-coupling of tautomerizable heterocycles with alkynes via Pd/Cu-catalyzed phosphonium coupling von Kang, Fu-An, Lanter, James C, Cai, Chaozhong, Sui, Zhihua, Murray, William V

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Conjugation of a peptide to an antibody engineered with free cysteines dramatically improves half-life and activity von Camacho, Raul C., You, Seohee, D’Aquino, Katharine E., Li, Wenyu, Wang, Yuanping, Gunnet, Joseph, Littrell, James, Qi, Jian Shen, Kang, Lijuan, Jian, Wenying, MacDonald, Mary, Tat, Timothy, Steiner, Derek, Zhang, Yue-Mei, Lanter, James, Patch, Raymond, Zhang, Rui, Li, Jiali, Edavettal, Suzanne, Edwards, Wilson, Dinh, Thai, Wang, Li Ying, Connor, Judy, Hunter, Michael, Chi, Ellen, Swanson, Ronald V., Leonard, James N., Case, Martin A.

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Discovery of a GPR40 Superagonist: The Impact of Aryl Propionic Acid α‑Fluorination von Huang, Hui, Meegalla, Sanath K, Lanter, James C, Winters, Michael P, Zhao, Shuyuan, Littrell, James, Qi, Jenson, Rady, Brian, Lee, Paul S, Liu, Jianying, Martin, Tonya, Lam, Wing W, Xu, Fran, Lim, Heng Keang, Wilde, Thomas, Silva, Jose, Otieno, Monicah, Pocai, Alessandro, Player, Mark R

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Asymmetric Aza-Mannich Reactions of Sulfinimines:  Scope and Application to the Total Synthesis of a Bromopyrrole Alkaloid von Lanter, James C, Chen, Hongfeng, Zhang, Xuqing, Sui, Zhihua

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Recent advances in the development of selective androgen receptor modulators von Zhang, Xuqing, Lanter, James C, Sui, Zhihua

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Lab-Scale Preparation of a Novel Cyclopenta[b]furan Chemokine Receptor Antagonist von Teleha, Christopher A, Branum, Shawn, Zhang, Yongzheng, Reuman, Michael E, Van Der Steen, Luc, Verbeek, Marc, Fawzy, Nagy, Leo, Gregory C, Winters, Michael P, Kang, Fu-An, Kolpak, Michael, Beauchamp, Derek A, Lanter, James C, Russell, Ronald K, Sui, Zhihua, Vanbaelen, Hilde

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Silicon-Directed Oxa-Pictet−Spengler Cyclization and an Unusual Dimerization of 2-Trimethylsilanyl Tryptophols von Zhang, Xuqing, Li, Xiaojie, Lanter, James C, Sui, Zhihua

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Overcoming hERG activity in the discovery of a series of 4-azetidinyl-1-aryl-cyclohexanes as CCR2 antagonists von Zhang, Xuqing, Hufnagel, Heather, Markotan, Thomas, Lanter, James, Cai, Chaozhong, Hou, Cuifen, Singer, Monica, Opas, Evan, McKenney, Sandra, Crysler, Carl, Johnson, Dana, Sui, Zhihua

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The discovery of a potent orally efficacious indole androgen receptor antagonist through in vivo screening von Lanter, James C., Fiordeliso, James J., Jiang, Weiqin, Allan, George F., Lai, Muh-Tsann, Linton, Olivia, Hahn, Do Won, Lundeen, Scott G., Sui, Zhihua

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The discovery of novel cyclohexylamide CCR2 antagonists von Lanter, James C., Markotan, Thomas P., Zhang, Xuqing, Subasinghe, Nalin, Kang, Fu-An, Hou, Cuifen, Singer, Monica, Opas, Evan, McKenney, Sandra, Crysler, Carl, Johnson, Dana, Molloy, Christopher J., Sui, Zhihua

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Synthesis of potent and tissue-selective androgen receptor modulators (SARMs): 2-(2,2,2)-Trifluoroethyl-benzimidazole scaffold von Ng, Raymond A., Lanter, James C., Alford, Vernon C., Allan, George F., Sbriscia, Tifanie, Lundeen, Scott G., Sui, Zhihua

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Targeting Enteropeptidase with Reversible Covalent Inhibitors To Achieve Metabolic Benefits von Sun, Weimei, Zhang, Xuqing, Cummings, Maxwell D., Albarazanji, Kamal, Wu, Jiejun, Wang, Mina, Alexander, Richard, Zhu, Bin, Zhang, YueMei, Leonard, James, Lanter, James, Lenhard, James

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A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands von Lanter, James C., Fiordeliso, James J., Allan, George F., Musto, Amy, Hahn, Do Won, Sui, Zhihua

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Synthesis and SAR of potent and selective androgen receptor antagonists: 5,6-Dichloro-benzimidazole derivatives von Ng, Raymond A., Guan, Jihua, Alford, Vernon C., Lanter, James C., Allan, George F., Sbriscia, Tifanie, Linton, Olivia, Lundeen, Scott G., Sui, Zhihua

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Discovery of a novel series of guanidinebenzoates as gut-restricted enteropeptidase and trypsin dual inhibitors for the treatment of metabolic syndrome von Zhang, Xuqing, Zhu, Bin, Sun, Weimei, Wang, Mina, Albarazanji, Kamal, Ghosh, Brahma, Cummings, Maxwell, Lenhard, James, Leonard, James, Macielag, Mark, Lanter, James

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2-(2,2,2-Trifluoroethyl)-5,6-dichlorobenzimidazole derivatives as potent androgen receptor antagonists von Ng, Raymond A., Guan, Jihua, Alford, Vernon C., Lanter, James C., Allan, George F., Sbriscia, Tifanie, Lundeen, Scott G., Sui, Zhihua

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