A Divergent and Stereoselective Approach for the Syntheses of Some Polyhydroxylated Indolizidine and Pyrrolizidine Iminosugars von Rajender, Anugula, Rao, Jalagam Prasada, Rao, Batchu Venkateswara

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Identification of benzothiazole derived monosaccharides as potent, selective, and orally bioavailable inhibitors of human and mouse galectin-3; a rare example of using a S···O bind... von Liu, Chunjian, Wang, Wei, Feng, Jianxin, Beno, Brett, Raja, Thiruvenkadam, Swidorski, Jacob, Manepalli, Raju K.V.L.P., Vetrichelvan, Muthalagu, Rao Jalagam, Prasada, Nair, Satheesh K., Gupta, Anuradha, Panda, Manoranjan, Ghosh, Kaushik, Kaushikkumar Shukla, Jinal, Sale, Harinath, Shah, Devang, Singh Gautam, Shashyendra, Patel, Dipal, Mathur, Arvind, Ellsworth, Bruce A., Cheng, Dong, Regueiro-Ren, Alicia

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Atropisomerism Observed in Galactose-Based Monosaccharide Inhibitors of Galectin-3 Comprising 2-Methyl-4-phenyl-2,4-dihydro-3 H -1,2,4-triazole-3-thione von Yoon, David S, Liu, Chunjian, Jalagam, Prasada Rao, Feng, Jianxin, Wang, Wei, Swidorski, Jacob J, Xu, Li, Hartz, Richard A, Nair, Satheesh K, Beno, Brett R, Panda, Manoranjan, Ghosh, Kaushik, Kumar, Amit, Sale, Harinath, Shah, Devang, Mathur, Arvind, Ellsworth, Bruce A, Cheng, Dong, Regueiro-Ren, Alicia

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Atropisomerism Observed in Galactose-Based Monosaccharide Inhibitors of Galectin‑3 Comprising 2‑Methyl-4-phenyl-2,4-dihydro‑3H‑1,2,4-triazole-3-thione von Yoon, David S., Liu, Chunjian, Jalagam, Prasada Rao, Feng, Jianxin, Wang, Wei, Swidorski, Jacob J., Xu, Li, Hartz, Richard A., Nair, Satheesh K., Beno, Brett R., Panda, Manoranjan, Ghosh, Kaushik, Kumar, Amit, Sale, Harinath, Shah, Devang, Mathur, Arvind, Ellsworth, Bruce A., Cheng, Dong, Regueiro-Ren, Alicia

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Identification of Monosaccharide Derivatives as Potent, Selective, and Orally Bioavailable Inhibitors of Human and Mouse Galectin‑3 von Liu, Chunjian, Jalagam, Prasada Rao, Feng, Jianxin, Wang, Wei, Raja, Thiruvenkadam, Sura, Mallikarjuna Reddy, Manepalli, Raju K. V. L. P., Aliphedi, Bheema Reddy, Medavarapu, Santosh, Nair, Satheesh K., Muthalagu, Vetrichelvan, Natesan, Ramesh, Gupta, Anuradha, Beno, Brett, Panda, Manoranjan, Ghosh, Kaushik, Shukla, Jinal Kaushikkumar, Sale, Harinath, Haldar, Priyanka, Kalidindi, Narasimharaju, Shah, Devang, Patel, Dipal, Mathur, Arvind, Ellsworth, Bruce A., Cheng, Dong, Regueiro-Ren, Alicia

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A new stereoselective approach to aminocyclohexitols using RCM von Rajender, Anugula, Rao, Jalagam Prasada, Rao, Batchu Venkateswara

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Optimization of physicochemical properties of pyrrolidine GPR40 AgoPAMs results in a differentiated profile with improved pharmacokinetics and reduced off-target activities von Jurica, Elizabeth A., Wu, Ximao, Williams, Kristin N., Haque, Lauren E., Rampulla, Richard A., Mathur, Arvind, Zhou, Min, Cao, Gary, Cai, Hong, Wang, Tao, Liu, Heng, Xu, Carrie, Kunselman, Lori K., Antrilli, Thomas M., Hicks, Michael B., Sun, Qin, Dierks, Elizabeth A., Apedo, Atsu, Moore, Douglas B., Foster, Kimberly A., Cvijic, Mary Ellen, Panemangalore, Reshma, Khandelwal, Purnima, Wilkes, Jason J., Zinker, Bradley A., Robertson, Donald G., Janovitz, Evan B., Galella, Michael, Li, Yi-Xin, Li, Julia, Ramar, Thangeswaran, Jalagam, Prasada Rao, Jayaram, Ramya, Whaley, Jean M., Barrish, Joel C., Robl, Jeffrey A., Ewing, William R., Ellsworth, Bruce A.

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Formal Synthesis of (−)-Cyclaradine Using Ring Closing Metathesis von Raju, Gurrapu, Rao, Jalagam Prasada, Rao, Batchu Venkateswara

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von Jalagam, Prasada Rao, Panda, Manoranjan, Natesan, Murugesan, Devasthale, Pratik, Nara, Susheel Jethanand

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von Nair, Satheesh Kesavan, Jalagam, Prasada Rao, Panda, Manoranjan, Regueiro-Ren, Alicia, Devasthale, Pratik, Nara, Susheel Jethanand

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Tetrahydropyran-based thiodisaccharide mimics as Galectin-3 inhibitors von Nair, Satheesh Kesavan, Jalagam, Prasada Rao, Panda, Manoranjan, Regueiro-Ren, Alicia, Xu, Li, Hartz, Richard A, Yoon, David S

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SUBSTITUTED HETEROARYL COMPOUNDS USEFUL AS T CELL ACTIVATORS von Jalagam, Prasada Rao, Velaparthi, Upender, Olson, Richard E, Warrier, Jayakumar Sankara, Darne, Chetan Padmakar

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von NATESAN, Murugesan, DEVASTHALE, Pratik, PANDA, Manoranjan, JALAGAM, Prasada Rao, NARA, Susheel Jethanand

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von DEVASTHALE, Pratik, PANDA, Manoranjan, JALAGAM, Prasada Rao, NAIR, Satheesh Kesavan, NARA, Susheel Jethanand, REGUEIRO-REN, Alicia

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SUBSTITUTED HETEROARYL COMPOUNDS USEFUL AS T CELL ACTIVATORS von VELAPARTHI, Upender, DARNE, Chetan Padmakar, WARRIER, Jayakumar Sankara, OLSON, Richard E, JALAGAM, Prasada Rao

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Substituted heteroaryl compounds useful as T cell activators von VELAPARTHI, Upender, DARNE, Chetan Padmakar, WARRIER, Jayakumar Sankara, OLSON, Richard E, JALAGAM, Prasada Rao

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Substituted heteroaryl compounds useful as t cell activators von WARRIER Jayakumar Sankara, VELAPARTHI Upender, DARNE Chetan Padmakar, OLSON Richard E, JALAGAM Prasada Rao

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Substituted bicyclic compounds useful as T cell activators von Ding, Min, Jalagam, Prasada Rao, Chupak, Louis S, Velaparthi, Upender, Martin, Scott W, Olson, Richard E, Roy, Saumya, Warrier, Jayakumar Sankara, Gentles, Robert G, Grunenfelder, Denise Christine

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SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS von VELAPARTHI, Upender, DARNE, Chetan Padmakar, WARRIER, Jayakumar Sankara, ROY, Saumya, OLSON, Richard E, JALAGAM, Prasada Rao, GRUNENFELDER, Denise C, RAHAMAN, Hasibur, DASGUPTA, Bireshwar

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SMALL MOLECULE INHIBITORS OF GALECTIN-3 von NATESAN, Murugesan, DEVASTHALE, Pratik, PANDA, Manoranjan, JALAGAM, Prasada Rao, NARA, Susheel Jethanand

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