alpha.-Diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases von Angelastro, Michael R, Mehdi, Shujaath, Burkhart, Joseph P, Peet, Norton P, Bey, Philippe

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Synthesis of peptidyl fluoromethyl ketones and peptidyl α-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsi... von PEET, N. P, BURKHART, J. P, ANGELASTRO, M. R, GIROUX, E. L, SHUJAATH MEHDI, BEY, P, KOLB, M, NEISES, B, SCHIRLIN, D

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Preparation of α-keto ester enol acetates as potential prodrugs of human neutrophil elastase inhibitors von Burkhart, Joseph P., Mehdi, Shujaath, Koehl, Jack R., Angelastro, Michael R., Bey, Philippe, Peet, Norton P.

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Substrate-induced inactivation of aromatase by allenic and acetylenic steroids von Metcalf, B. W, Wright, C. L, Burkhart, J. P, Johnston, J. O

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The inhibition of human neutrophil elastase and cathepsin G by peptidyl 1,2-dicarbonyl derivatives von Mehdi, Shujaath, Angelastro, Michael P., Burkhart, Joseph P., Koehl, Jack R., Peet, Norton P., Bey, Philippe

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Novel time-dependent inhibitors of human placental aromatase von Burkhart, Joseph P, Peet, Norton P, Wright, C. Lee, Johnston, J. O'Neal

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Biological characterization of A-ring steroids von O'Neal Johnston, J., Lee Wright, C., Burkhart, Joseph P., Peet, Norton P.

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A-ring bridged steroids as potent inhibitors of aromatase von Peet, Norton P., Johnston, J.O'Neal, Burkhart, Joseph P., Wright, C.Lee

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Novel silylated steroids as aromatase inhibitors von Burkhart, Joseph P., Weintraub, Philip M., Wright, C.Lee, Johnston, J.O'Neal

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Inhibition of Human Neutrophil Elastase. 3. An Orally Active Enol Acetate Prodrug von Burkhart, Joseph P, Koehl, Jack R, Mehdi, Shujaath, Durham, Sherrie L, Janusz, Michael J, Huber, Edward W, Angelastro, Michael R, Sunder, Shyam, Metz, William A

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Efficient preparation of peptidyl pentafluoroethyl ketones von ANGELASTRO, M. R, BURKHART, J. P, BEY, P, PEET, N. P

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Oxidation of α-hydroxy esters to α-keto esters using the dess-martin periodinane reagent von Burkhart, Joseph P, Peet, Norton P, Bey, Philippe

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Time-dependent inhibition of human placental aromatase with a 2,19-methyleneoxy-bridged androstenedione von Peet, Norton P, Burkhart, Joseph P, Wright, C. Lee, Johnston, J. O'Neal

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A novel method for the preparation of peptidyl α-keto esters von Burkhart, Joseph P., Peet, Norton P., Bey, Philippe

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Synthesis of 2,19-bridged androstenediones von Burkhart, Joseph P, Huber, Edward W, Laskovics, F. Mark, Peet, Norton P

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The synthesis of α,α-difluoroaldehydes and ketones via claisen rearrangements von Metcalf, Brian W., Jarvi, Esa T., Burkhart, Joseph P.

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Molecular Design and Characterization of an α-Thrombin Inhibitor Containing a Novel P1 Moiety von Malikayil, J. A, Burkhart, Joseph P, Schreuder, Herman A, Broersma, Robert J, Tardif, Chantal, Kutcher, Louis W, Mehdi, Shujaath, Schatzman, Gerald L, Neises, Bernhard, Peet, Norton P

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Inhibition of Human Neutrophil Elastase with Peptidyl Electrophilic Ketones. 2. Orally Active PG-Val-Pro-Val Pentafluoroethyl Ketones von Angelastro, Michael R, Baugh, Larry E, Bey, Philippe, Burkhart, Joseph P, Chen, Teng-Man, Durham, Sherrie L, Hare, C. Michelle, Huber, Edward W, Janusz, Michael J

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Synthesis of polycyclic ketones via carbonylative cyclization of organopalladium compounds derived from norbornene and norbornadiene von Larock, Richard C., Takagi, Kentaro, Burkhart, Joseph P., Hershberger, Susan S.

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Organopalladium approaches to prostaglandins. 2. Synthesis of prostaglandin endoperoxide analogs via π-allylpalladium additions to bicyclic olefins von Larock, R.C., Burkhart, J.P., Oertle, K.

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