Pyrazole-Based Thrombin Inhibitors with a Serine-Trapping Mechanism of Action: Synthesis and Biological Activity von Dunker, Calvin, Imberg, Lukas, Siutkina, Alena I, Erbacher, Catharina, Daniliuc, Constantin G, Karst, Uwe, Kalinin, Dmitrii V

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N‐Pyrazolyl‐ and N‐Triazolylamines and ‐Ureas as Antileishmanial and Antitrypanosomal Drugs von Winge, Tobias, Imberg, Lukas, Perry, Ben, Matheeussen, An, Caljon, Guy, Kalinin, Dmitrii, Wünsch, Bernhard

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Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors von Platte, Simon, Korff, Marvin, Imberg, Lukas, Balicioglu, Ilker, Erbacher, Catharina, Will, Jonas M., Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.

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Acylated 1 H -1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action von Korff, Marvin, Imberg, Lukas, Will, Jonas M, Bückreiß, Nico, Kalinina, Svetlana A, Wenzel, Benjamin M, Kastner, Gregor A, Daniliuc, Constantin G, Barth, Maximilian, Ovsepyan, Ruzanna A, Butov, Kirill R, Humpf, Hans-Ulrich, Lehr, Matthias, Panteleev, Mikhail A, Poso, Antti, Karst, Uwe, Steinmetzer, Torsten, Bendas, Gerd, Kalinin, Dmitrii V

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Acylated 1H‑1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action von Korff, Marvin, Imberg, Lukas, Will, Jonas M, Bückreiß, Nico, Kalinina, Svetlana A, Wenzel, Benjamin M, Kastner, Gregor A, Daniliuc, Constantin G, Barth, Maximilian, Ovsepyan, Ruzanna A, Butov, Kirill R, Humpf, Hans-Ulrich, Lehr, Matthias, Panteleev, Mikhail A, Poso, Antti, Karst, Uwe, Steinmetzer, Torsten, Bendas, Gerd, Kalinin, Dmitrii V

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An automated analysis method enabling the screening of covalent thrombin and factor XIIa inhibitors via liquid chromatography‐mass spectrometry von Erbacher, Catharina, Athmer, Mathis, Kröger, Erik, Dahrendorf, Laureen, Imberg, Lukas, Kalinin, Dmitrii V., Karst, Uwe

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Cover Feature: Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors (ChemMedChem 24/2021) von Platte, Simon, Korff, Marvin, Imberg, Lukas, Balicioglu, Ilker, Erbacher, Catharina, Will, Jonas M., Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.

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Amide-functionalized 1,2,4-Triazol-5-amines as Covalent Inhibitors of Blood Coagulation Factor XIIa and Thrombin von Imberg, Lukas, Platte, Simon, Erbacher, Catharina, Daniliuc, Constantin G., Kalinina, Svetlana A., Dörner, Wolfgang, Poso, Antti, Karst, Uwe, Kalinin, Dmitrii V.

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