An inhibitor of RORγ for chronic pulmonary obstructive disease treatment von Desai, Harshada, Marathe, Megha, Potdar, Varada, Tiwari, Prabhakar, Joshi, Ashwini, Kadam, Sheetal R., Joshi, Arti Rajesh, Kulkarni, Abhay, Bhosale, Vikram, Hadambar, Avinash, Lodhiya, Bhavik, Udupa, Venkatesha, Behera, Dayanidhi, Chaudhari, Sachin S., Das, Sanjib, Bajpai, Malini, Gowda, Nagaraj, Iyer, Pravin S.

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Oxidative DMSO Cyclization Cascade to Bicyclic Hydroxyketonitriles von Kornfeind, John, Iyer, Pravin S, Keller, Taylor M, Fleming, Fraser F

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1,4-azaindole, a potential drug candidate for treatment of tuberculosis von Chatterji, Monalisa, Shandil, Radha, Manjunatha, M R, Solapure, Suresh, Ramachandran, Vasanthi, Kumar, Naveen, Saralaya, Ramanatha, Panduga, Vijender, Reddy, Jitendar, Prabhakar, K R, Sharma, Sreevalli, Sadler, Claire, Cooper, Christopher B, Mdluli, Khisi, Iyer, Pravin S, Narayanan, Shridhar, Shirude, Pravin S

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Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo von Shirude, Pravin S, Shandil, Radha, Sadler, Claire, Naik, Maruti, Hosagrahara, Vinayak, Hameed, Shahul, Shinde, Vikas, Bathula, Chandramohan, Humnabadkar, Vaishali, Kumar, Naveen, Reddy, Jitendar, Panduga, Vijender, Sharma, Sreevalli, Ambady, Anisha, Hegde, Naina, Whiteaker, James, McLaughlin, Robert E, Gardner, Humphrey, Madhavapeddi, Prashanti, Ramachandran, Vasanthi, Kaur, Parvinder, Narayan, Ashwini, Guptha, Supreeth, Awasthy, Disha, Narayan, Chandan, Mahadevaswamy, Jyothi, Vishwas, KG, Ahuja, Vijaykamal, Srivastava, Abhishek, Prabhakar, KR, Bharath, Sowmya, Kale, Ramesh, Ramaiah, Manjunatha, Choudhury, Nilanjana Roy, Sambandamurthy, Vasan K, Solapure, Suresh, Iyer, Pravin S, Narayanan, Shridhar, Chatterji, Monalisa

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Synthesis and in vitro evaluation of novel 8-aminoquinoline–pyrazolopyrimidine hybrids as potent antimalarial agents von Kannan, Murugan, Raichurkar, Anandkumar V., Khan, Fazlur Rahman Nawaz, Iyer, Pravin S.

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Development of potent and selective Cathepsin C inhibitors free of aortic binding liability by application of a conformational restriction strategy von Banerjee, Abhisek, Velagaleti, Ranganadh, Patil, Sandip, Pawar, Mahesh, Yadav, Pravin, Kadam, Pradip, Qadri, Mohammad Mohsin, Chakraborti, Samitabh, Saini, Jagmohan S., Behera, Dayanidhi B., Karanjai, Keya, Iyer, Pravin S., Gharat, Laxmikant A., Das, Sanjib

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Lead Optimization of 1,4-Azaindoles as Antimycobacterial Agents von Shirude, Pravin S, Shandil, Radha K, Manjunatha, M. R, Sadler, Claire, Panda, Manoranjan, Panduga, Vijender, Reddy, Jitendar, Saralaya, Ramanatha, Nanduri, Robert, Ambady, Anisha, Ravishankar, Sudha, Sambandamurthy, Vasan K, Humnabadkar, Vaishali, Jena, Lalit K, Suresh, Rudrapatna S, Srivastava, Abhishek, Prabhakar, K. R, Whiteaker, James, McLaughlin, Robert E, Sharma, Sreevalli, Cooper, Christopher B, Mdluli, Khisi, Butler, Scott, Iyer, Pravin S, Narayanan, Shridhar, Chatterji, Monalisa

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Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity von R, Manjunatha M, Shandil, Radha, Panda, Manoranjan, Sadler, Claire, Ambady, Anisha, Panduga, Vijender, Kumar, Naveen, Mahadevaswamy, Jyothi, Sreenivasaiah, M, Narayan, Ashwini, Guptha, Supreeth, Sharma, Sreevalli, Sambandamurthy, Vasan K, Ramachandran, Vasanthi, Mallya, Meenakshi, Cooper, Christopher, Mdluli, Khisi, Butler, Scott, Tommasi, Ruben, Iyer, Pravin S, Narayanan, Shridhar, Chatterji, Monalisa, Shirude, Pravin S

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4‑Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity von Naik, Maruti, Humnabadkar, Vaishali, Tantry, Subramanyam J, Panda, Manoranjan, Narayan, Ashwini, Guptha, Supreeth, Panduga, Vijender, Manjrekar, Praveena, Jena, Lalit kumar, Koushik, Krishna, Shanbhag, Gajanan, Jatheendranath, Sandesh, Manjunatha, M. R, Gorai, Gopinath, Bathula, Chandramohan, Rudrapatna, Suresh, Achar, Vijayashree, Sharma, Sreevalli, Ambady, Anisha, Hegde, Naina, Mahadevaswamy, Jyothi, Kaur, Parvinder, Sambandamurthy, Vasan K, Awasthy, Disha, Narayan, Chandan, Ravishankar, Sudha, Madhavapeddi, Prashanti, Reddy, Jitendar, Prabhakar, KR, Saralaya, Ramanatha, Chatterji, Monalisa, Whiteaker, James, McLaughlin, Bob, Chiarelli, Laurent R, Riccardi, Giovanna, Pasca, Maria Rosalia, Binda, Claudia, Neres, João, Dhar, Neeraj, Signorino-Gelo, François, McKinney, John D, Ramachandran, Vasanthi, Shandil, Radha, Tommasi, Ruben, Iyer, Pravin S, Narayanan, Shridhar, Hosagrahara, Vinayak, Kavanagh, Stefan, Dinesh, Neela, Ghorpade, Sandeep R

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Synthesis of benzofused 1,4-azaborinols via [4 + 2] annulation strategy and its application in indole synthesis von Chinnapattu, Murugan, Sathiyanarayanan, Kulathu Iyer, Iyer, Pravin S.

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Synthesis and biological evaluation of adamantane-based aminophenols as a novel class of antiplasmodial agents von Chinnapattu, Murugan, Sathiyanarayanan, Kulathu Iyer, Iyer, Pravin S.

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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate von Hameed P., Shahul, Solapure, Suresh, Patil, Vikas, Henrich, Philipp P., Magistrado, Pamela A., Bharath, Sowmya, Murugan, Kannan, Viswanath, Pavithra, Puttur, Jayashree, Srivastava, Abhishek, Bellale, Eknath, Panduga, Vijender, Shanbag, Gajanan, Awasthy, Disha, Landge, Sudhir, Morayya, Sapna, Koushik, Krishna, Saralaya, Ramanatha, Raichurkar, Anandkumar, Rautela, Nikhil, Roy Choudhury, Nilanjana, Ambady, Anisha, Nandishaiah, Radha, Reddy, Jitendar, Prabhakar, K. R., Menasinakai, Sreenivasaiah, Rudrapatna, Suresh, Chatterji, Monalisa, Jiménez-Díaz, María Belén, Martínez, María Santos, Sanz, Laura María, Coburn-Flynn, Olivia, Fidock, David A., Lukens, Amanda K., Wirth, Dyann F., Bandodkar, Balachandra, Mukherjee, Kakoli, McLaughlin, Robert E., Waterson, David, Rosenbrier-Ribeiro, Lyn, Hickling, Kevin, Balasubramanian, V., Warner, Peter, Hosagrahara, Vinayak, Dudley, Adam, Iyer, Pravin S., Narayanan, Shridhar, Kavanagh, Stefan, Sambandamurthy, Vasan K.

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Discovery of Novel PI3-Kinase δ Specific Inhibitors for the Treatment of Rheumatoid Arthritis: Taming CYP3A4 Time-Dependent Inhibition von Safina, Brian S, Baker, Stewart, Baumgardner, Matt, Blaney, Paul M, Chan, Bryan K, Chen, Yung-Hsiang, Cartwright, Matthew W, Castanedo, Georgette, Chabot, Christine, Cheguillaume, Arnaud J, Goldsmith, Paul, Goldstein, David M, Goyal, Bindu, Hancox, Timothy, Handa, Raj K, Iyer, Pravin S, Kaur, Jasmit, Kondru, Rama, Kenny, Jane R, Krintel, Sussie L, Li, Jun, Lesnick, John, Lucas, Matthew C, Lewis, Cristina, Mukadam, Sophie, Murray, Jeremy, Nadin, Alan J, Nonomiya, Jim, Padilla, Fernando, Palmer, Wylie S, Pang, Jodie, Pegg, Neil, Price, Steve, Reif, Karin, Salphati, Laurent, Savy, Pascal A, Seward, Eileen M, Shuttleworth, Stephen, Sohal, Sukhjit, Sweeney, Zachary K, Tay, Suzanne, Tivitmahaisoon, Parcharee, Waszkowycz, Bohdan, Wei, Binqing, Yue, Qin, Zhang, Chenghong, Sutherlin, Daniel P

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N‑Aryl-2-aminobenzimidazoles: Novel, Efficacious, Antimalarial Lead Compounds von Ramachandran, Sreekanth, Hameed P, Shahul, Srivastava, Abhishek, Shanbhag, Gajanan, Morayya, Sapna, Rautela, Nikhil, Awasthy, Disha, Kavanagh, Stefan, Bharath, Sowmya, Reddy, Jitendar, Panduga, Vijender, Prabhakar, K. R, Saralaya, Ramanatha, Nanduri, Robert, Raichurkar, Anandkumar, Menasinakai, Sreenivasaiah, Achar, Vijayashree, Jiménez-Díaz, María Belén, Martínez, María Santos, Angulo-Barturen, Iñigo, Ferrer, Santiago, Sanz, Laura María, Gamo, Francisco Javier, Duffy, Sandra, Avery, Vicky M, Waterson, David, Lee, Marcus C. S, Coburn-Flynn, Olivia, Fidock, David A, Iyer, Pravin S, Narayanan, Shridhar, Hosagrahara, Vinayak, Sambandamurthy, Vasan K

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Aminoazabenzimidazoles, a Novel Class of Orally Active Antimalarial Agents von Hameed P, Shahul, Chinnapattu, Murugan, Shanbag, Gajanan, Manjrekar, Praveena, Koushik, Krishna, Raichurkar, Anandkumar, Patil, Vikas, Jatheendranath, Sandesh, Rudrapatna, Suresh S, Barde, Shubhada P, Rautela, Nikhil, Awasthy, Disha, Morayya, Sapna, Narayan, Chandan, Kavanagh, Stefan, Saralaya, Ramanatha, Bharath, Sowmya, Viswanath, Pavithra, Mukherjee, Kakoli, Bandodkar, Balachandra, Srivastava, Abhishek, Panduga, Vijender, Reddy, Jitender, Prabhakar, K. R, Sinha, Achyut, Jiménez-Díaz, María Belén, Martínez, María Santos, Angulo-Barturen, Iñigo, Ferrer, Santiago, Sanz, Laura María, Gamo, Francisco Javier, Duffy, Sandra, Avery, Vicky M, Magistrado, Pamela A, Lukens, Amanda K, Wirth, Dyann F, Waterson, David, Balasubramanian, V, Iyer, Pravin S, Narayanan, Shridhar, Hosagrahara, Vinayak, Sambandamurthy, Vasan K, Ramachandran, Sreekanth

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Synthesis of novel benzoxaborinin-4-ones and its application in indolin-2-ones synthesis using a Suzuki–Miyaura reaction protocol von Murugan, Kannan, Chinnapattu, Murugan, Nawaz Khan, Fazlur-Rahman, Iyer, Pravin S.

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2‑Phenylindole and Arylsulphonamide: Novel Scaffolds Bactericidal against Mycobacterium tuberculosis von Naik, Maruti, Ghorpade, Sandeep, Jena, Lalit Kumar, Gorai, Gopinath, Narayan, Ashwini, Guptha, Supreeth, Sharma, Sreevalli, Dinesh, Neela, Kaur, Parvinder, Nandishaiah, Radha, Bhat, Jyothi, Balakrishnan, Gayathri, Humnabadkar, Vaishali, Ramachandran, Vasanthi, Naviri, Lava Kumar, Khadtare, Pallavi, Panda, Manoranjan, Iyer, Pravin S, Chatterji, Monalisa

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Reagent-Based DOS: Developing a Diastereoselective Methodology to Access Spirocyclic- and Fused Heterocyclic Ring Systems von Damerla, V. Surendra Babu, Tulluri, Chiranjeevi, Gundla, Rambabu, Naviri, Lava, Adepally, Uma, Iyer, Pravin S., Murthy, Y. L. N., Prabhakar, Nampally, Sen, Subhabrata

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2-Substituted N-aryl piperazines as novel triple reuptake inhibitors for the treatment of depression von Carter, David S., Cai, Hai-Ying, Lee, Eun Kyung, Iyer, Pravin S., Lucas, Matthew C., Roetz, Ralf, Schoenfeld, Ryan C., Weikert, Robert J.

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Synthesis of Privileged Scaffolds by Using Diversity-Oriented Synthesis von Surakanti, Ramu, Sanivarapu, Sumalatha, Thulluri, Chiranjeevi, Iyer, Pravin S., Tangirala, Raghuram S., Gundla, Rambabu, Addepally, Uma, Murthy, Y. L. N., Velide, Lakshmi, Sen, Subhabrata

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