Development and Prospects of Furin Inhibitors for Therapeutic Applications von Ivachtchenko, Alexandre V, Khvat, Alexander V, Shkil, Dmitrii O

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Aprotinin-Drug against Respiratory Diseases von Ivachtchenko, Alexandre V, Ivashchenko, Andrey A, Shkil, Dmitrii O, Ivashchenko, Ilya A

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Resistance profiles for the investigational neuraminidase inhibitor AV5080 in influenza A and B viruses von Ivashchenko, Andrei A, Jones, Jeremy C, Shkil, Dmitry O, Ivanenkov, Yan A, Pascua, Philippe Noriel Q, Penaflor, Melissa K, Karapetian, Ruben N, Govorkova, Elena A, Ivachtchenko, Alexandre V

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The Efficacy of Aprotinin Combinations with Selected Antiviral Drugs in Mouse Models of Influenza Pneumonia and Coronavirus Infection Caused by SARS-CoV-2 von Ivashchenko, Andrey A, Zagribelnyy, Bogdan A, Ivanenkov, Yan A, Ivashchenko, Ilya A, Karapetian, Ruben N, Kravchenko, Dmitry V, Savchuk, Nikolay P, Yakubova, Elena V, Ivachtchenko, Alexandre V

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Effect of Aprotinin and Avifavir(R) Combination Therapy for Moderate COVID-19 Patients von Ivashchenko, Andrey A., Azarova, Valeria N., Egorova, Alina N., Karapetian, Ruben N., Kravchenko, Dmitry, Krivonos, Natalia, Loginov, Vladimir G., Poyarkov, Stanislav, Merkulova, Elena A., Rosinkova, Olga S., Savchuk, Nikolay P., Topr, Mikhail A., Simakina, Elena N., Yakubova, Elena, Ivachtchenko, Alexandre

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Methylation of Methyl 4-Hydroxy-2-thioxo-1,2-dihydroquinoline-3-carboxylate: Synthetic, Crystallographic, and Molecular Docking Studies von Kovalenko, Sergiy M., Drushlyak, Oleksandr G., Shishkina, Svitlana, Konovalova, Irina S., Mariutsa, Illia O., Bunyatyan, Natalya D., Kravchenko, Dmitry, Ivanov, Vladimir V., Ivachtchenko, Alexandre, Langer, Thierry

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Safety and efficacy of aviandr in patients with generalized anxiety disorder: A multicenter, randomized, double-blind, placebo-controlled, dose-finding, pilot study von Ivashchenko, Andrey A., Morozova, Margarita A., Vostokova, Natalia V., Beniashvily, Allan G., Bukhanovskaya, Olga A., Burminskiy, Denis S., Egorova, Alina N., Gluskina, Lubov Y., Gorchakov, Dmitriy S., Karapetian, Ruben N., Kasimova, Lala N., Kravchenko, Dmitry V., Lepilkina, Taissia A., Merkulova, Elena A., Mitkin, Oleg D., Penchul, Nataliya A., Potanin, Sergey S., Rupchev, George E., Ivachtchenko, Alexandre V.

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AVIFAVIR for Treatment of Patients With Moderate Coronavirus Disease 2019 (COVID-19): Interim Results of a Phase II/III Multicenter Randomized Clinical Trial von Ivashchenko, Andrey A., Dmitriev, Kirill A., Vostokova, Natalia V., Azarova, Valeria N., Blinow, Andrew A., Egorova, Alina N., Gordeev, Ivan G., Ilin, Alexey P., Karapetian, Ruben N., Kravchenko, Dmitry, Lomakin, Nikita, Merkulova, Elena A., Papazova, Natalia A., Pavlikova, Elena P., Savchuk, Nikolay P., Simakina, Elena N., Sitdekov, Tagir A., Smolyarchuk, Elena A., Tikhomolova, Elena G., Yakubova, Elena, Ivachtchenko, Alexandre

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Influenza C virus susceptibility to antivirals with different mechanisms of action von Chesnokov, Anton, Ivashchenko, Andrei A, Matsuzaki, Yoko, Takashita, Emi, Mishin, Vasiliy P, Ivachtchenko, Alexandre V, Gubareva, Larisa V

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Synthesis, X-ray crystal structure, Hirshfeld surface analysis, and molecular docking study of novel inhibitor of hepatitis B: methyl 4-fluoro-3-(morpholinosulfonyl)benzo[b]thiophe... von Ivachtchenko, Alexandre V., Mitkin, Oleg D., Kravchenko, Dmitry V., Kovalenko, Sergiy M., Shishkina, Svitlana V., Bunyatyan, Natalya D., Konovalova, Irina S., Dmitrieva, Irina G., Ivanov, Vladimir V., Langer, Thierry

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Novel One-Pot Synthesis of Methyl 4-Hydroxy-2-thioxo-1,2-dihydroquinoline-3-carboxylate: Synthetic and Crystallographic Studies von Kovalenko, Sergiy M., Drushlyak, Oleksandr G., Konovalova, Irina S., Mariutsa, Illia O., Kravchenko, Dmitry V., Ivachtchenko, Alexandre V., Mitkin, Oleg D.

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AVN-211, Novel and Highly Selective 5‑HT6 Receptor Small Molecule Antagonist, for the Treatment of Alzheimer’s Disease von Ivachtchenko, Alexandre V, Lavrovsky, Yan, Ivanenkov, Yan A

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Antiviral susceptibility of clade 2.3.4.4b highly pathogenic avian influenza A(H5N1) viruses isolated from birds and mammals in the United States, 2022 von Nguyen, Ha T., Chesnokov, Anton, De La Cruz, Juan, Pascua, Philippe Noriel Q., Mishin, Vasiliy P., Jang, Yunho, Jones, Joyce, Di, Han, Ivashchenko, Andrei A., Killian, Mary Lea, Torchetti, Mia K., Lantz, Kristina, Wentworth, David E., Davis, Charles T., Ivachtchenko, Alexandre V., Gubareva, Larisa V.

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Synthesis, inhibitory activity and oral dosing formulation of AV5124, the structural analogue of influenza virus endonuclease inhibitor baloxavir von Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Karapetian, Ruben N, Kravchenko, Dmitry V, Mochalov, Stephan V, Ryakhovskiy, Alexey A, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V

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Non-rigid Diarylmethyl Analogs of Baloxavir as Cap-Dependent Endonuclease Inhibitors of Influenza Viruses von Ivashchenko, Andrei A, Mitkin, Oleg D, Jones, Jeremy C, Nikitin, Alexander V, Koryakova, Angela G, Ryakhovskiy, Alexey, Karapetian, Ruben N, Kravchenko, Dmitry V, Aladinskiy, Vladimir, Leneva, Irina A, Falynskova, Irina N, Glubokova, Ekaterina A, Govorkova, Elena A, Ivachtchenko, Alexandre V

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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) A... von Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M

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New Four-Component Ugi-Type Reaction. Synthesis of Heterocyclic Structures Containing a Pyrrolo[1,2-a][1,4]diazepine Fragment von Ilyn, Alexey P, Trifilenkov, Andrey S, Kuzovkova, Julia A, Kutepov, Sergey A, Nikitin, Alexandre V, Ivachtchenko, Alexandre V

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Complexity-Enhancing Acid-Promoted Rearrangement of Tricyclic Products of Tandem Ugi 4CC/Intramolecular Diels−Alder Reaction von Ilyin, Alexei, Kysil, Volodymyr, Krasavin, Mikhail, Kurashvili, Irina, Ivachtchenko, Alexandre V

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Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists von Ivachtchenko, Alexandre V., Ivanenkov, Yan A., Mitkin, Oleg D., Vorobiev, Anton A., Kuznetsova, Irina V., Shevkun, Natalia A., Koryakova, Angela G., Karapetian, Ruben N., Trifelenkov, Andrey S., Kravchenko, Dmitry V., Veselov, Mark S., Chufarova, Nina V.

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(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor von Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Okun, Ilya M, Tkachenko, Sergey E, Vorobiev, Anton A

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