High-throughput screening assays for the identification of chemical probes von Inglese, James, Johnson, Ronald L, Simeonov, Anton, Xia, Menghang, Zheng, Wei, Austin, Christopher P, Auld, Douglas S

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Comprehensive characterization of cytochrome P450 isozyme selectivity across chemical libraries von Veith, Henrike, Lloyd, David G, Inglese, James, Southall, Noel, James, Tim, Fayne, Darren, Auld, Douglas S, Huang, Ruili, Artemenko, Natalia, Shen, Min, Austin, Christopher P

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High-Throughput Screening to Identify Inhibitors of the Type I Interferon–Major Histocompatibility Complex Class I Pathway in Skeletal Muscle von Kinder, Travis B, Dranchak, Patricia K, Inglese, James

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Mechanism of PTC124 activity in cell-based luciferase assays of nonsense codon suppression von Auld, Douglas S, Thorne, Natasha, Maguire, William F, Inglese, James

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Identification of oxadiazoles as new drug leads for the control of schistosomiasis von Austin, Christopher P, Williams, David L, Sayed, Ahmed A, Simeonov, Anton, Thomas, Craig J, Inglese, James

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In vivo quantitative high-throughput screening for drug discovery and comparative toxicology von Dranchak, Patricia K, Oliphant, Erin, Queme, Bryan, Lamy, Laurence, Wang, Yuhong, Huang, Ruili, Xia, Menghang, Tao, Dingyin, Inglese, James

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Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors von Miller, Thomas W, Amason, Joshua D, Garcin, Elsa D, Lamy, Laurence, Dranchak, Patricia K, Macarthur, Ryan, Braisted, John, Rubin, Jeffrey S, Burgess, Teresa L, Farrell, Catherine L, Roberts, David D, Inglese, James

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Macrocycle peptides delineate locked-open inhibition mechanism for microorganism phosphoglycerate mutases von Yu, Hao, Dranchak, Patricia, Li, Zhiru, MacArthur, Ryan, Munson, Matthew S., Mehzabeen, Nurjahan, Baird, Nathan J., Battalie, Kevin P., Ross, David, Lovell, Scott, Carlow, Clotilde K. S., Suga, Hiroaki, Inglese, James

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Molecular basis for the high-affinity binding and stabilization of firefly luciferase by PTC124 von Auld, Douglas S, Lovell, Scott, Thorne, Natasha, Lea, Wendy A, Maloney, David J, Shen, Min, Rai, Ganesha, Battaile, Kevin P, Thomas, Craig J, Simeonov, Anton, Hanzlik, Robert P, Inglese, James

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ICE1 promotes the link between splicing and nonsense-mediated mRNA decay von Baird, Thomas D, Cheng, Ken Chih-Chien, Chen, Yu-Chi, Buehler, Eugen, Martin, Scott E, Inglese, James, Hogg, J Robert

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Characterization of Chemical Libraries for Luciferase Inhibitory Activity von Auld, Douglas S, Southall, Noel T, Jadhav, Ajit, Johnson, Ronald L, Diller, David J, Simeonov, Anton, Austin, Christopher P, Inglese, James

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Structure–activity relationship of ipglycermide binding to phosphoglycerate mutases von Wiedmann, Mareike, Dranchak, Patricia K., Aitha, Mahesh, Queme, Bryan, Collmus, Christopher D., Kashipathy, Maithri M., Kanter, Liza, Lamy, Laurence, Rogers, Joseph M., Tao, Dingyin, Battaile, Kevin P., Rai, Ganesha, Lovell, Scott, Suga, Hiroaki, Inglese, James

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Reporting data from high-throughput screening of small-molecule libraries von Shamu, Caroline E, Guy, R Kiplin, Inglese, James

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Small-molecule agonists for the thyrotropin receptor stimulate thyroid function in human thyrocytes and mice von Neumann, Susanne, Huang, Wenwei, Titus, Steve, Krause, Gerd, Kleinau, Gunnar, Alberobello, Anna Teresa, Zheng, Wei, Southall, Noel T, Inglese, James, Austin, Christopher P, Celi, Francesco S, Gavrilova, Oksana, Thomas, Craig J, Raaka, Bruce M, Gershengorn, Marvin C

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A robotic platform for quantitative high-throughput screening von Michael, Sam, Auld, Douglas, Klumpp, Carleen, Jadhav, Ajit, Zheng, Wei, Thorne, Natasha, Austin, Christopher P, Inglese, James, Simeonov, Anton

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A Basis for Reduced Chemical Library Inhibition of Firefly Luciferase Obtained from Directed Evolution von Auld, Douglas S, Zhang, Ya-Qin, Southall, Noel T, Rai, Ganesha, Landsman, Marc, MacLure, Jennifer, Langevin, Daniel, Thomas, Craig J, Austin, Christopher P, Inglese, James

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A bioluminescent cytotoxicity assay for assessment of membrane integrity using a proteolytic biomarker von Cho, Ming-Hsuang, Niles, Andrew, Huang, Ruili, Inglese, James, Austin, Christopher P., Riss, Terry, Xia, Menghang

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Structure Mechanism Insights and the Role of Nitric Oxide Donation Guide the Development of Oxadiazole-2-Oxides as Therapeutic Agents against Schistosomiasis von Rai, Ganesha, Sayed, Ahmed A, Lea, Wendy A, Luecke, Hans F, Chakrapani, Harinath, Prast-Nielsen, Stefanie, Jadhav, Ajit, Leister, William, Shen, Min, Inglese, James, Austin, Christopher P, Keefer, Larry, Arnér, Elias S. J, Simeonov, Anton, Maloney, David J, Williams, David L, Thomas, Craig J

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Differentiating Alzheimer disease-associated aggregates with small molecules von Honson, Nicolette S, Johnson, Ronald L, Huang, Wenwei, Inglese, James, Austin, Christopher P, Kuret, Jeff

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Identification of compounds that potentiate CREB signaling as possible enhancers of long-term memory von Xia, Menghang, Huang, Ruili, Guo, Vicky, Southall, Noel, Cho, Ming-Hsuang, Inglese, James, Austin, Christopher P, Nirenberg, Marshall

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