Trivalent PROTACs enhance protein degradation via combined avidity and cooperativity von Imaide, Satomi, Riching, Kristin M., Makukhin, Nikolai, Vetma, Vesna, Whitworth, Claire, Hughes, Scott J., Trainor, Nicole, Mahan, Sarah D., Murphy, Nancy, Cowan, Angus D., Chan, Kwok-Ho, Craigon, Conner, Testa, Andrea, Maniaci, Chiara, Urh, Marjeta, Daniels, Danette L., Ciulli, Alessio

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The Combination of Binding Avidity of Ovomucoid-Specific IgE Antibody and Specific IgG4 Antibody Can Predict Positive Outcomes of Oral Food Challenges during Stepwise Slow Oral Imm... von Taniuchi, Shoichiro, Sakai, Rika, Nishida, Takahiro, Goma, Meguru, Mitomori, Masatoshi, Imaide, Aya, Enomoto, Masahiro, Nishino, Masamitsu, Okizuka, Yo, Kido, Hiroshi

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Acetic Anhydride Mediated Retro-Ene Reaction via a [4.4.3]Propel­lane Skeleton Intermediate Containing a Quaternary Ammonium Linkage von Kutsumura, Noriki, Okada, Takahiro, Imaide, Satomi, Fujii, Hideaki, Nagase, Hiroshi

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The application of a specific morphinan template to the synthesis of galanthamine von Yamamoto, Naoshi, Okada, Takahiro, Harada, Yukimasa, Kutsumura, Noriki, Imaide, Satomi, Saitoh, Tsuyoshi, Fujii, Hideaki, Nagase, Hiroshi

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Evaluation of liquefaction probability of earth-fill dam over next 50 years using geostatistical method based on CPT von Imaide, Kazunari, Nishimura, Shin-ichi, Shibata, Toshifumi, Shuku, Takayuki, Murakami, Akira, Fujisawa, Kazunori

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Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain von Cipriano, Alessandra, Milite, Ciro, Feoli, Alessandra, Viviano, Monica, Pepe, Giacomo, Campiglia, Pietro, Sarno, Giuliana, Picaud, Sarah, Imaide, Satomi, Makukhin, Nikolai, Filippakopoulos, Panagis, Ciulli, Alessio, Castellano, Sabrina, Sbardella, Gianluca

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Transformation of naltrexone into mesembrane and investigation of the binding properties of its intermediate derivatives to opioid receptors von Konoura, Kazuya, Fujii, Hideaki, Imaide, Satomi, Gouda, Hiroaki, Hirayama, Shigeto, Hirono, Shuichi, Nagase, Hiroshi

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Front Cover: Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain (ChemMedChem 20/2022... von Cipriano, Alessandra, Milite, Ciro, Feoli, Alessandra, Viviano, Monica, Pepe, Giacomo, Campiglia, Pietro, Sarno, Giuliana, Picaud, Sarah, Imaide, Satomi, Makukhin, Nikolai, Filippakopoulos, Panagis, Ciulli, Alessio, Castellano, Sabrina, Sbardella, Gianluca

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Discovery of Benzoimidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain von Cipriano, Alessandra, Milite, Ciro, Feoli, Alessandra, Viviano, Monica, Pepe, Giacomo, Campiglia, Pietro, Sarno, Giuliana, Picaud, Sarah, Imaide, Satomi, Makukhin, Nikolai, Filippakopoulos, Panagis, Ciulli, Alessio, Castellano, Sabrina, Sbardella, Gianluca

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Essential structure of opioid κ receptor agonist nalfurafine for binding to the κ receptor 2: Synthesis of decahydro(iminoethano)phenanthrene derivatives and their pharmacologies von Nagase, Hiroshi, Imaide, Satomi, Hirayama, Shigeto, Nemoto, Toru, Fujii, Hideaki

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Essential Structure of Opioid κ Receptor Agonist Nalfurafine for Binding to κ Receptor 1: Synthesis of Decahydroisoquinoline Derivatives and Their Pharmacologies von Nagase, Hiroshi, Imaide, Satomi, Yamada, Takaaki, Hirayama, Shigeto, Nemoto, Toru, Yamaotsu, Noriyuki, Hirono, Shuichi, Fujii, Hideaki

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Discovery and SAR Studies of Orally Active Somatostatin Receptor Subtype‑2 (SSTR2) Agonists for the Treatment of Acromegaly von Ishida, Akiharu, Tajima, Yohei, Okabe, Yasuyuki, Matsushita, Takeshi, Sekiguchi, Tetsuya, Imaide, Satomi, Nomura, Yoshinori, Tanaka, Motoyuki, Nojima, Shoji, Yoshida, Atsushi, Iyoda, Yoko, Aoki, Shohei, Nishio, Takuya, Komagata, Tatsuya, Iwaki, Masanori, Shono, Tomoyuki, Naganawa, Atsushi, Imagawa, Akira

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Synthesis of (−)-Homogalanthamine from Naltrexone von Yamamoto, Naoshi, Fujii, Hideaki, Imaide, Satomi, Hirayama, Shigeto, Nemoto, Toru, Inokoshi, Junji, Tomoda, Hiroshi, Nagase, Hiroshi

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Novel cleavage reaction of the C16–N17 bond in naltrexone derivatives von Fujii, Hideaki, Imaide, Satomi, Watanabe, Akio, Nemoto, Toru, Nagase, Hiroshi

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Evaluation of strength distribution at cut slope of decomposed granite with the use of sounding method and geophysical exploration method von Ueta, Tatsuya, Nishimura, Shin-Ichi, Imaide, Kazunari, Shibata, Toshifumi, Shuku, Takayuki

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Essential structure of opioid κ receptor agonist nalfurafine for binding to the κ receptor 3: Synthesis of decahydro(iminoethano)phenanthrene derivatives with an oxygen functionali... von Fujii, Hideaki, Imaide, Satomi, Hirayama, Shigeto, Nemoto, Toru, Gouda, Hiroaki, Hirono, Shuichi, Nagase, Hiroshi

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A Double Decarboxylation Reaction of an Oxazolidinone and Carboxylic Acid: Its Application to the Synthesis of a New Opioid Lead Compound von Fujii, Hideaki, Imaide, Satomi, Watanabe, Akio, Yoza, Kenji, Nakajima, Mayumi, Nakao, Kaoru, Mochizuki, Hidenori, Sato, Noriko, Nemoto, Toru, Nagase, Hiroshi

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EVALUATION OF THE SPATIAL VARIABILITY OF CONE PENETRATION RESISTANCE INSIDE AN EARTH-FILL DAM COMPOSED OF MATERIALS WITH DIFFERENT PARTICLE SIZE DISTRIBUTION von IMAIDE, Kazunari, NISHIMURA, Shin-ichi, SHIBATA, Toshifumi, SHUKU, Takayuki

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Essential structure of opioid [kappa] receptor agonist nalfurafine for binding to the [kappa] receptor 3: Synthesis of decahydro(iminoethano)phenanthrene derivatives with an oxygen... von Fujii, Hideaki, Imaide, Satomi, Hirayama, Shigeto, Nemoto, Toru, Gouda, Hiroaki, Hirono, Shuichi, Nagase, Hiroshi

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Essential Structure of Opioid [kappa] Receptor Agonist Nalfurafine for Binding to [kappa] Receptor 1 von Nagase, Hiroshi, Imaide, Satomi, Yamada, Takaaki, Hirayama, Shigeto, Nemoto, Toru, Yamaotsu, Noriyuki, Hirono, Shuichi, Fujii, Hideaki

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