Small molecule absorption by PDMS in the context of drug response bioassays von van Meer, B.J., de Vries, H., Firth, K.S.A., van Weerd, J., Tertoolen, L.G.J., Karperien, H.B.J., Jonkheijm, P., Denning, C., IJzerman, A.P., Mummery, C.L.

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Importance of the extracellular loops in G protein-coupled receptors for ligand recognition and receptor activation von Peeters, M.C, van Westen, G.J.P, Li, Q, IJzerman, A.P

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The role of the second and third extracellular loops of the adenosine A1 receptor in activation and allosteric modulation von Peeters, M.C., Wisse, L.E., Dinaj, A., Vroling, B., Vriend, G., IJzerman, A.P.

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Role of ceramide 1 in the molecular organization of the stratum corneum lipids von Bouwstra, J A, Gooris, G S, Dubbelaar, F E, Weerheim, A M, Ijzerman, A P, Ponec, M

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Structure–activity relationships of trans-substituted-propenoic acid derivatives on the nicotinic acid receptor HCA2 (GPR109A) von van Veldhoven, J.P.D., Blad, C.C., Artsen, C.M., Klopman, C., Wolfram, D.R., Abdelkadir, M.J., Lane, J.R., Brussee, J., IJzerman, A.P.

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Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism von den Hollander, L.S., Béquignon, O.J.M., Wang, X., van Wezel, K., Broekhuis, J., Gorostiola González, M., de Visser, K.E., IJzerman, A.P., van Westen, G.J.P., Heitman, L.H.

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Kinetic binding and activation profiles of endogenous tachykinins targeting the NK1 receptor von Nederpelt, I., Bleeker, D., Tuijt, B., IJzerman, A.P., Heitman, L.H.

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Corrigendum to “Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism” [Biochem. Pharmacol. 208 (2023) 115399] von den Hollander, L.S., Béquignon, O.J.M., Wang, X., van Wezel, K., Broekhuis, J., Gorostiola González, M., de Visser, K.E., IJzerman, A.P., van Westen, G.J.P., Heitman, L.H.

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Persistent GnRH receptor activation in pituitary αT3-1 cells analyzed with a label-free technology von Nederpelt, I., Vergroesen, R.D., IJzerman, A.P., Heitman, L.H.

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Pharmacological and biochemical analysis of FPL 67156, a novel, selective inhibitor of ecto‐ATPase von Crack, B.E., Pollard, C.E., Beukers, M.W., Roberts, S.M., Hunt, S.F., Ingall, A.H., McKechnie, K.C.W., IJzerman, A.P., Leff, P.

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Getting personal: Endogenous adenosine receptor signaling in lymphoblastoid cell lines von Hillger, J.M., Diehl, C., van Spronsen, E., Boomsma, D.I., Slagboom, P.E., Heitman, L.H., IJzerman, A.P.

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Pharmacological analysis of ecto‐ATPase inhibition: evidence for combined enzyme inhibition and receptor antagonism in P2X‐purinoceptor ligands von Crack, B.E., Beukers, M.W., McKechnie, K.C.W., IJzerman, A.P., Leff, P.

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Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives von Vilums, M., Zweemer, A.J.M., Dekkers, S., Askar, Y., de Vries, H., Saunders, J., Stamos, D., Brussee, J., Heitman, L.H., IJzerman, A.P.

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Pharmacological characterization of allosteric modulators: a case for chemokine receptors von Hollander, L.S. den, IJzerman, A.P., Heitman, L.H.

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Gonadotrophin-releasing hormone receptors in GtoPdb v.2023.1 von Heitman, L.H., IJzerman, A.P., McArdle, C.A., Pawson, A.J.

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Luteolin, a compound with adenosine A1 receptor-binding activity, and chromone and dihydronaphthalenone constituents from Senna siamea von Ingkaninan, K, IJzerman, A.P, Verpoorte, R

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Computational characterization of membrane proteins as anticancer targets: current challenges and opportunities von Gorostiola González, M.: Rakers, P.R.J., Jespers, W., IJzerman, A.P., Heitman, L.H., Westen, G.J.P. van

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International Union of Basic and Clinical Pharmacology. CXII: adenosine receptors: a further update von IJzerman, A.P., Jacobson, K.A., Müller, C.E., Cronstein, B.N., Cunha, R.A.

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Targeting solute carriers to modulate receptor-ligand interactions von Sijben, H.J., Superti-Furga, G., IJzerman, A.P., Heitman, L.H.

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MPP+-induced changes in cellular impedance as a measure for organic cation transporter (SLC22A1-3) activity and inhibition von Mocking, T.A.M., Sijben, H.J., Vermeulen, Y., IJzerman, A.P., Heitman, L.H.

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