Small molecule absorption by PDMS in the context of drug response bioassays von van Meer, B.J., de Vries, H., Firth, K.S.A., van Weerd, J., Tertoolen, L.G.J., Karperien, H.B.J., Jonkheijm, P., Denning, C., IJzerman, A.P., Mummery, C.L.

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Papyrus: a large-scale curated dataset aimed at bioactivity predictions von Béquignon, O. J. M., Bongers, B. J., Jespers, W., IJzerman, A. P., van der Water, B., van Westen, G. J. P.

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Importance of the extracellular loops in G protein-coupled receptors for ligand recognition and receptor activation von Peeters, M.C, van Westen, G.J.P, Li, Q, IJzerman, A.P

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Pan-cancer functional analysis of somatic mutations in G protein-coupled receptors von Bongers, B. J., Gorostiola González, M., Wang, X., van Vlijmen, H. W. T., Jespers, W., Gutiérrez-de-Terán, H., Ye, K., IJzerman, A. P., Heitman, L. H., van Westen, G. J. P.

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Kv11.1 (hERG)‐induced cardiotoxicity: a molecular insight from a binding kinetics study of prototypical Kv11.1 (hERG) inhibitors von Yu, Z, IJzerman, A P, Heitman, L H

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Impact of cancer-associated mutations in CC chemokine receptor 2 on receptor function and antagonism von den Hollander, L.S., Béquignon, O.J.M., Wang, X., van Wezel, K., Broekhuis, J., Gorostiola González, M., de Visser, K.E., IJzerman, A.P., van Westen, G.J.P., Heitman, L.H.

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Kinetic binding and activation profiles of endogenous tachykinins targeting the NK1 receptor von Nederpelt, I., Bleeker, D., Tuijt, B., IJzerman, A.P., Heitman, L.H.

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Persistent GnRH receptor activation in pituitary αT3-1 cells analyzed with a label-free technology von Nederpelt, I., Vergroesen, R.D., IJzerman, A.P., Heitman, L.H.

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The role of the second and third extracellular loops of the adenosine A1 receptor in activation and allosteric modulation von Peeters, M.C., Wisse, L.E., Dinaj, A., Vroling, B., Vriend, G., IJzerman, A.P.

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Correlation between human ether‐a‐go‐go‐related gene channel inhibition and action potential prolongation von Saxena, P, Hortigon‐Vinagre, M P, Beyl, S, Baburin, I, Andranovits, S, Iqbal, S M, Costa, A, IJzerman, A P, Kügler, P, Timin, E, Smith, G L, Hering, S

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Getting personal: Endogenous adenosine receptor signaling in lymphoblastoid cell lines von Hillger, J.M., Diehl, C., van Spronsen, E., Boomsma, D.I., Slagboom, P.E., Heitman, L.H., IJzerman, A.P.

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Inverse agonism at G protein‐coupled receptors: (patho)physiological relevance and implications for drug discovery von De Ligt, Rianne A F, Kourounakis, Angeliki P, IJzerman, Ad P

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Role of ceramide 1 in the molecular organization of the stratum corneum lipids von Bouwstra, J A, Gooris, G S, Dubbelaar, F E, Weerheim, A M, Ijzerman, A P, Ponec, M

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Reduced hepatitis B and D viral entry using novel clinically-applied inhibitors of the sodium taurocholate co-transporting polypeptide von Donkers, J, Zehnder, B, van Westen, G, IJzerman, A, Kwakkenbos, M, Urban, S, Elferink, R.O, van de Graaf, S

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Interleukin-6 Upregulates Neuronal Adenosine A1 Receptors: Implications for Neuromodulation and Neuroprotection von Biber, Knut, Pinto-Duarte, A, Wittendorp, M C, Dolga, A M, Fernandes, C C, Von Frijtag Drabbe Künzel, J, Keijser, J N, de Vries, R, Ijzerman, A P, Ribeiro, J A, Eisel, U, Sebastião, A M, Boddeke, H W G M

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Structure‐activity relationships of pentamidine‐affected ion channel trafficking and dofetilide mediated rescue von Varkevisser, R, Houtman, M J C, Linder, T, Git, K C G, Beekman, H D M, Tidwell, R R, IJzerman, A P, Stary‐Weinzinger, A, Vos, M A, Heyden, M A G

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Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors von Massink, A., Holzheimer, M., Hölscher, A., Louvel, J., Guo, D., Spijksma, G., Hankemeier, T., IJzerman, A. P.

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Pyrazole Derivatives as Partial Agonists for the Nicotinic Acid Receptor von van Herk, T, Brussee, J, van den Nieuwendijk, A. M. C. H, van der Klein, P. A. M, IJzerman, A. P, Stannek, C, Burmeister, A, Lorenzen, A

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Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives von Vilums, M., Zweemer, A.J.M., Dekkers, S., Askar, Y., de Vries, H., Saunders, J., Stamos, D., Brussee, J., Heitman, L.H., IJzerman, A.P.

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Thiazole and Thiadiazole Analogues as a Novel Class of Adenosine Receptor Antagonists von van Muijlwijk-Koezen, Jacqueline E, Timmerman, Hendrik, Vollinga, Roeland C, Frijtag von Drabbe Künzel, Jacobien, de Groote, Miriam, Visser, Sven, IJzerman, Adriaan P

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