Small molecule antagonists for chemokine CCR3 receptors von Willems, Lianne I., IJzerman, Ad P.

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Differential Expression of Adenosine A3 Receptors Controls Adenosine A2A Receptor-Mediated Inhibition of TLR Responses in Microglia von van der Putten, Celine, Zuiderwijk-Sick, Ella A, van Straalen, Linda, de Geus, Eveline D, Boven, Leonie A, Kondova, Ivanela, IJzerman, Ad P, Bajramovic, Jeffrey J

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Inverse agonism at G protein‐coupled receptors: (patho)physiological relevance and implications for drug discovery von De Ligt, Rianne A F, Kourounakis, Angeliki P, IJzerman, Ad P

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Allosteric modulation of adenosine receptors von Göblyös, Anikó, IJzerman, Ad P.

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The Molecule Evoluator. An Interactive Evolutionary Algorithm for the Design of Drug-Like Molecules von Lameijer, Eric-Wubbo, Kok, Joost N, Bäck, Thomas, IJzerman, Ad P

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How to Catch a Membrane Protein in Action: A Review of Functional Membrane Protein Immobilization Strategies and Their Applications von Früh, Virginie, IJzerman, Ad P, Siegal, Gregg

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Recent developments in constitutive receptor activity and inverse agonism, and their potential for GPCR drug discovery von Bond, Richard A., IJzerman, Ad P.

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The adhesion G protein-coupled receptor G2 (ADGRG2/GPR64) constitutively activates SRE and NFκB and is involved in cell adhesion and migration von Peeters, Miriam C., Fokkelman, Michiel, Boogaard, Bob, Egerod, Kristoffer L., van de Water, Bob, IJzerman, Ad P., Schwartz, Thue W.

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Synthesis and evaluation of homo-bivalent GnRHR ligands von Bonger, Kimberly M., van den Berg, Richard J.B.H.N., Heitman, Laura H., IJzerman, Ad P., Oosterom, Julia, Timmers, Cornelis M., Overkleeft, Herman S., van der Marel, Gijsbert A.

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LUF7244 plus Dofetilide Rescues Aberrant Kv11.1 Trafficking and Produces Functional IKv11.1 von Qile, Muge, Ji, Yuan, Golden, Tyona D., Houtman, Marien J.C., Romunde, Fee, Fransen, Doreth, van Ham, Willem B., IJzerman, Ad P., January, Craig T., Heitman, Laura H., Stary-Weinzinger, Anna, Delisle, Brian P., van der Heyden, Marcel A.G.

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Scintillation proximity assay (SPA) as a new approach to determine a ligand’s kinetic profile. A case in point for the adenosine A1 receptor von Xia, Lizi, de Vries, Henk, IJzerman, Ad P., Heitman, Laura H.

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TreeSOM: Cluster analysis in the self-organizing map von Samsonova, Elena V., Kok, Joost N., IJzerman, Ad P.

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LUF7244 plus Dofetilide Rescues Aberrant K-v 11.1 Trafficking and Produces Functional I-Kv11.1 von Qile, Muge, Ji, Yuan, Golden, Tyona D., Houtman, Marien J. C., Romunde, Fee, Fransen, Doreth, van Ham, Willem B., IJzerman, Ad P., January, Craig T., Heitman, Laura H., Stary-Weinzinger, Anna, Delisle, Brian P., van der Heyden, Marcel A. G.

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Functional selectivity of adenosine receptor ligands von Verzijl, Dennis, IJzerman, Ad P.

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LUF7244, an allosteric modulator/activator of Kv11.1 channels, counteracts dofetilide‐induced torsades de pointes arrhythmia in the chronic atrioventricular block dog model von Qile, Muge, Beekman, Henriette D.M., Sprenkeler, David J., Houtman, Marien J.C., Ham, Willem B., Stary‐Weinzinger, Anna, Beyl, Stanislav, Hering, Steffen, Berg, Dirk‐Jan, Lange, Elizabeth C.M., Heitman, Laura H., IJzerman, Ad P., Vos, Marc A., Heyden, Marcel A.G.

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TLR-Induced IL-12 and CCL2 Production by Myeloid Cells Is Dependent on Adenosine A3 Receptor–Mediated Signaling von van der Putten, Céline, Veth, Jennifer, Sukurova, Lejla, Zuiderwijk-Sick, Ella A., Simonetti, Elles, Koenen, Hans J. P .M., Burm, Saskia M., van Noort, Johannes M., IJzerman, Ad P., van Hijum, Sacha A. F. T., Diavatopoulos, Dimitri, Bajramovic, Jeffrey J.

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A covalent antagonist for the human adenosine A2A receptor von Yang, Xue, Dong, Guo, Michiels, Thomas J.M., Lenselink, Eelke B., Heitman, Laura, Louvel, Julien, IJzerman, Ad P.

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LUF7244, an allosteric modulator/activator of K v 11.1 channels, counteracts dofetilide-induced torsades de pointes arrhythmia in the chronic atrioventricular block dog model von Qile, Muge, Beekman, Henriette D M, Sprenkeler, David J, Houtman, Marien J C, van Ham, Willem B, Stary-Weinzinger, Anna, Beyl, Stanislav, Hering, Steffen, van den Berg, Dirk-Jan, de Lange, Elizabeth C M, Heitman, Laura H, IJzerman, Ad P, Vos, Marc A, van der Heyden, Marcel A G

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The endocannabinoid 2-arachidonylglycerol is a negative allosteric modulator of the human A3 adenosine receptor von Lane, J. Robert, Beukers, Margot W., Mulder-Krieger, Thea, IJzerman, Ad P.

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Allosteric modulation of G protein-coupled receptors: perspectives and recent developments von Soudijn, Willem, van Wijngaarden, Ineke, IJzerman, Ad P.

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