Chrysin, baicalein and galangin are indirect activators of the human constitutive androstane receptor (CAR) von Carazo Fernández, Alejandro, Smutny, Tomas, Hyrsová, Lucie, Berka, Karel, Pavek, Petr

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Transcriptional and post-transcriptional regulation of the pregnane X receptor: a rationale for interindividual variability in drug metabolism von Smutny, Tomas, Hyrsova, Lucie, Braeuning, Albert, Ingelman-Sundberg, Magnus, Pavek, Petr

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The pregnane X receptor down‐regulates organic cation transporter 1 (SLC22A1) in human hepatocytes by competing for (“squelching”) SRC‐1 coactivator von Hyrsova, Lucie, Smutny, Tomas, Carazo, Alejandro, Moravcik, Stefan, Mandikova, Jana, Trejtnar, Frantisek, Gerbal‐Chaloin, Sabine, Pavek, Petr

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Acetylated deoxycholic (DCA) and cholic (CA) acids are potent ligands of pregnane X (PXR) receptor von Carazo, Alejandro, Hyrsova, Lucie, Dusek, Jan, Chodounska, Hana, Horvatova, Alzbeta, Berka, Karel, Bazgier, Vaclav, Gan-Schreier, Hongying, Chamulitrat, Waleé, Kudova, Eva, Pavek, Petr

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The 3ʹ-untranslated region contributes to the pregnane X receptor (PXR) expression down-regulation by PXR ligands and up-regulation by glucocorticoids von Smutny, Tomas, Dusek, Jan, Hyrsova, Lucie, Nekvindova, Jana, Horvatova, Alzbeta, Micuda, Stanislav, Gerbal-Chaloin, Sabine, Pavek, Petr

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Teriflunomide Is an Indirect Human Constitutive Androstane Receptor (CAR) Activator Interacting With Epidermal Growth Factor (EGF) Signaling von Carazo, Alejandro, Dusek, Jan, Holas, Ondrej, Skoda, Josef, Hyrsova, Lucie, Smutny, Tomas, Soukup, Tomas, Dosedel, Martin, Pávek, Petr

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Resveratrol modifies biliary secretion of cholephilic compounds in sham-operated and cholestatic rats von Dolezelova, Eva, Prasnicka, Alena, Cermanova, Jolana, Carazo, Alejandro, Hyrsova, Lucie, Hroch, Milos, Mokry, Jaroslav, Adamcova, Michaela, Mrkvicova, Alena, Pavek, Petr, Micuda, Stanislav

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Trans-resveratrol, but not other natural stilbenes occurring in food, carries the risk of drug-food interaction via inhibition of cytochrome P450 enzymes or interaction with xenose... von Hyrsova, Lucie, Vanduchova, Alena, Dusek, Jan, Smutny, Tomas, Carazo, Alejandro, Maresova, Veronika, Trejtnar, Frantisek, Barta, Pavel, Anzenbacher, Pavel, Dvorak, Zdenek, Pavek, Petr

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Steviol, an aglycone of steviol glycoside sweeteners, interacts with the pregnane X (PXR) and aryl hydrocarbon (AHR) receptors in detoxification regulation von Dusek, Jan, Carazo, Alejandro, Trejtnar, Frantisek, Hyrsova, Lucie, Holas, Ondřej, Smutny, Tomas, Micuda, Stanislav, Pavek, Petr

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2‑(3-Methoxyphenyl)quinazoline Derivatives: A New Class of Direct Constitutive Androstane Receptor (CAR) Agonists von Smutny, Tomas, Nova, Alice, Drechslerová, Marcela, Carazo, Alejandro, Hyrsova, Lucie, Hrušková, Zuzana Rania, Kuneš, Jiří, Pour, Milan, Špulák, Marcel, Pavek, Petr

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Correction to 2‑(3-Methoxyphenyl)quinazoline Derivatives: A New Class of Direct Constitutive Androstane Receptor (CAR) Agonists von Smutny, Tomas, Nova, Alice, Drechslerová, Marcela, Carazo, Alejandro, Hyrsova, Lucie, Hrušková, Zuzana Rania, Kuneš, Jiří, Pour, Milan, Špulák, Marcel, Pavek, Petr

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Entecavir Interacts with Influx Transporters hOAT1, hCNT2, hCNT3, but Not with hOCT2: The Potential for Renal Transporter-Mediated Cytotoxicity and Drug-Drug Interactions von Mandíková, Jana, Volková, Marie, Pávek, Petr, Navrátilová, Lucie, Hyršová, Lucie, Janeba, Zlatko, Pavlík, Jan, Bárta, Pavel, Trejtnar, František

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