Molecular engineering of safe and efficacious oral basal insulin von Hubálek, Frantisek, Refsgaard, Hanne H. F., Gram-Nielsen, Sanne, Madsen, Peter, Nishimura, Erica, Münzel, Martin, Brand, Christian Lehn, Stidsen, Carsten Enggaard, Claussen, Christian Hove, Wulff, Erik Max, Pridal, Lone, Ribel, Ulla, Kildegaard, Jonas, Porsgaard, Trine, Johansson, Eva, Steensgaard, Dorte Bjerre, Hovgaard, Lars, Glendorf, Tine, Hansen, Bo Falck, Jensen, Maja Kirkegaard, Nielsen, Peter Kresten, Ludvigsen, Svend, Rugh, Susanne, Garibay, Patrick W., Moore, Mary Courtney, Cherrington, Alan D., Kjeldsen, Thomas

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An ingestible self-orienting system for oral delivery of macromolecules von Abramson, Alex, Caffarel-Salvador, Ester, Khang, Minsoo, Dellal, David, Silverstein, David, Gao, Yuan, Frederiksen, Morten Revsgaard, Vegge, Andreas, Hubálek, František, Water, Jorrit J, Friderichsen, Anders V, Fels, Johannes, Kirk, Rikke Kaae, Cleveland, Cody, Collins, Joy, Tamang, Siddartha, Hayward, Alison, Landh, Tomas, Buckley, Stephen T, Roxhed, Niclas, Rahbek, Ulrik, Langer, Robert, Traverso, Giovanni

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Insights into the Mode of Inhibition of Human Mitochondrial Monoamine Oxidase B from High-Resolution Crystal Structures von Binda, Claudia, Li, Min, Hubálek, Frantisek, Restelli, Nadia, Edmondson, Dale E., Mattevi, Andrea

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Demonstration of Isoleucine 199 as a Structural Determinant for the Selective Inhibition of Human Monoamine Oxidase B by Specific Reversible Inhibitors von Hubálek, Frantisek, Binda, Claudia, Khalil, Ashraf, Li, Min, Mattevi, Andrea, Castagnoli, Neal, Edmondson, Dale E.

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Author Correction: Molecular engineering of safe and efficacious oral basal insulin von Hubálek, Frantisek, Refsgaard, Hanne H. F., Gram-Nielsen, Sanne, Madsen, Peter, Nishimura, Erica, Münzel, Martin, Brand, Christian Lehn, Stidsen, Carsten Enggaard, Claussen, Christian Hove, Wulff, Erik Max, Pridal, Lone, Ribel, Ulla, Kildegaard, Jonas, Porsgaard, Trine, Johansson, Eva, Steensgaard, Dorte Bjerre, Hovgaard, Lars, Glendorf, Tine, Hansen, Bo Falck, Jensen, Maja Kirkegaard, Nielsen, Peter Kresten, Ludvigsen, Svend, Rugh, Susanne, Garibay, Patrick W., Moore, Mary Courtney, Cherrington, Alan D., Kjeldsen, Thomas

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Structure of human monoamine oxidase B, a drug target for the treatment of neurological disorders von Edmondson, Dale E, Mattevi, Andrea, Binda, Claudia, Newton-Vinson, Paige, Hubálek, Frantisek

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Oral delivery of systemic monoclonal antibodies, peptides and small molecules using gastric auto-injectors von Abramson, Alex, Frederiksen, Morten Revsgaard, Vegge, Andreas, Jensen, Brian, Poulsen, Mette, Mouridsen, Brian, Jespersen, Mikkel Oliver, Kirk, Rikke Kaae, Windum, Jesper, Hubálek, František, Water, Jorrit J., Fels, Johannes, Gunnarsson, Stefán B., Bohr, Adam, Straarup, Ellen Marie, Ley, Mikkel Wennemoes Hvitfeld, Lu, Xiaoya, Wainer, Jacob, Collins, Joy, Tamang, Siddartha, Ishida, Keiko, Hayward, Alison, Herskind, Peter, Buckley, Stephen T., Roxhed, Niclas, Langer, Robert, Rahbek, Ulrik, Traverso, Giovanni

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Molecular Engineering of Insulin Icodec, the First Acylated Insulin Analog for Once-Weekly Administration in Humans von Kjeldsen, Thomas B, Hubálek, František, Hjørringgaard, Claudia U, Tagmose, Tina M, Nishimura, Erica, Stidsen, Carsten E, Porsgaard, Trine, Fledelius, Christian, Refsgaard, Hanne H. F, Gram-Nielsen, Sanne, Naver, Helle, Pridal, Lone, Hoeg-Jensen, Thomas, Jeppesen, Claus Bekker, Manfè, Valentina, Ludvigsen, Svend, Lautrup-Larsen, Inger, Madsen, Peter

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Chemo- and Regioselective Ethynylation of Tryptophan-Containing Peptides and Proteins von Hansen, Morten Borre, Hubálek, František, Skrydstrup, Troels, Hoeg-Jensen, Thomas

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Investigation of the Physico-Chemical Properties that Enable Co-Formulation of Basal Insulin Degludec with Fast-Acting Insulin Aspart von Havelund, Svend, Ribel, Ulla, Hubálek, František, Hoeg-Jensen, Thomas, Wahlund, Per-Olof, Jonassen, Ib

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Purification and Identification of High Molecular Weight Products Formed During Storage of Neutral Formulation of Human Insulin von Hjorth, Christian Fogt, Hubálek, František, Andersson, Jonatan, Poulsen, Christian, Otzen, Daniel, Naver, Helle

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Expression, Receptor Binding, and Biophysical Characterization of Guinea Pig Insulin desB30: A Monomeric Insulin Variant von Engholm, Ebbe, Hansen, Thomas H., Johansson, Eva, Strauss, Holger M., Vinther, Tine N., Jensen, Knud J., Hubálek, Frantisek, Kjeldsen, Thomas B.

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Molecular and pharmacological characterization of insulin icodec: a new basal insulin analog designed for once-weekly dosing von Nishimura, Erica, Pridal, Lone, Glendorf, Tine, Hansen, Bo Falk, Hubálek, František, Kjeldsen, Thomas, Kristensen, Niels Rode, Lützen, Anne, Lyby, Karsten, Madsen, Peter, Pedersen, Thomas Åskov, Ribel-Madsen, Rasmus, Stidsen, Carsten Enggaard, Haahr, Hanne

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Insulin analog with additional disulfide bond has increased stability and preserved activity von Vinther, Tine N., Norrman, Mathias, Ribel, Ulla, Huus, Kasper, Schlein, Morten, Steensgaard, Dorte B., Pedersen, Thomas Å., Pettersson, Ingrid, Ludvigsen, Svend, Kjeldsen, Thomas, Jensen, Knud J., Hubálek, František

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Enhanced disulphide bond stability contributes to the once-weekly profile of insulin icodec von Hubálek, František, Cramer, Christian N., Helleberg, Hans, Johansson, Eva, Nishimura, Erica, Schluckebier, Gerd, Steensgaard, Dorte Bjerre, Sturis, Jeppe, Kjeldsen, Thomas B.

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Engineering of Orally Available, Ultralong-Acting Insulin Analogues: Discovery of OI338 and OI320 von Kjeldsen, Thomas B., Hubalek, Frantisek, Tagmose, Tina M., Pridal, Lone, Refsgaard, Hanne H. F., Porsgaard, Trine, Gram-Nielsen, Sanne, Hovgaard, Lars, Valore, Henrik, Munzel, Martin, Hjorringgaard, Claudia U., Jeppesen, Claus Bekker, Manfe, Valentina, Hoeg-Jensen, Thomas, Ludvigsen, Svend, Nielsen, Peter Kresten, Lautrup-Larsen, Inger, Stidsen, Carsten E., Wulff, Erik M., Garibay, Patrick W., Kodra, Janos T., Nishimura, Erica, Madsen, Peter

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A microneedle platform for buccal macromolecule delivery von Caffarel-Salvador, Ester, Kim, Soyoung, Soares, Vance, Tian, Ryan Yu, Stern, Sarah R., Minahan, Daniel, Yona, Raissa, Lu, Xiaoya, Zakaria, Fauziah R., Collins, Joy, Wainer, Jacob, Wong, Jessica, McManus, Rebecca, Tamang, Siddartha, McDonnell, Shane, Ishida, Keiko, Hayward, Alison, Liu, Xiewen, Hubalek, Frantisek, Fels, Johannes, Vegge, Andreas, Frederiksen, Morten Revsgaard, Rahbek, Ulrik, Yoshitake, Tadayuki, Fujimoto, James, Roxhed, Niclas, Langer, Robert, Traverso, Giovanni

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The role of citric acid in oral peptide and protein formulations: Relationship between calcium chelation and proteolysis inhibition von Welling, Søren H., Hubálek, František, Jacobsen, Jette, Brayden, David J., Rahbek, Ulrik L., Buckley, Stephen T.

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Chemically modified peptides and proteins - critical considerations for oral delivery von Buckley, Stephen T., Hubálek, František, Rahbek, Ulrik Lytt

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Binding of Rasagiline-Related Inhibitors to Human Monoamine Oxidases:  A Kinetic and Crystallographic Analysis von Binda, Claudia, Hubálek, Frantisek, Li, Min, Herzig, Yaacov, Sterling, Jeffrey, Edmondson, Dale E, Mattevi, Andrea

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