Metallaphotoredox aryl and alkyl radiomethylation for PET ligand discovery von Pipal, Robert W., Stout, Kenneth T., Musacchio, Patricia Z., Ren, Sumei, Graham, Thomas J. A., Verhoog, Stefan, Gantert, Liza, Lohith, Talakad G., Schmitz, Alexander, Lee, Hsiaoju S., Hesk, David, Hostetler, Eric D., Davies, Ian W., MacMillan, David W. C.

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Discovery of 6‑(Fluoro-18 F)‑3-(1H‑pyrrolo[2,3‑c]pyridin-1-yl)isoquinolin-5-amine ([18F]-MK-6240): A Positron Emission Tomography (PET) Imaging Agent for Quantification of Neurofib... von Walji, Abbas M, Hostetler, Eric D, Selnick, Harold, Zeng, Zhizhen, Miller, Patricia, Bennacef, Idriss, Salinas, Cristian, Connolly, Brett, Gantert, Liza, Holahan, Marie, O’Malley, Stacey, Purcell, Mona, Riffel, Kerry, Li, Jing, Balsells, Jaume, OBrien, Julie A, Melquist, Stacey, Soriano, Aileen, Zhang, Xiaoping, Ogawa, Aimie, Xu, Serena, Joshi, Elizabeth, Della Rocca, Joseph, Hess, Fred J, Schachter, Joel, Hesk, David, Schenk, David, Struyk, Arie, Babaoglu, Kerim, Lohith, Talakad G, Wang, Yaode, Yang, Kun, Fu, Jianmin, Evelhoch, Jeffrey L, Coleman, Paul J

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In vivo quantification of calcitonin gene-related peptide receptor occupancy by telcagepant in rhesus monkey and human brain using the positron emission tomography tracer [11C]MK-4... von Hostetler, Eric D, Joshi, Aniket D, Sanabria-Bohórquez, Sandra, Fan, Hong, Zeng, Zhizhen, Purcell, Mona, Gantert, Liza, Riffel, Kerry, Williams, Mangay, O'Malley, Stacey, Miller, Patricia, Selnick, Harold G, Gallicchio, Steven N, Bell, Ian M, Salvatore, Christopher A, Kane, Stefanie A, Li, Chi-Chung, Hargreaves, Richard J, de Groot, Tjibbe, Bormans, Guy, Van Hecken, Anne, Derdelinckx, Inge, de Hoon, Jan, Reynders, Tom, Declercq, Ruben, De Lepeleire, Inge, Kennedy, W P, Blanchard, Rebecca, Marcantonio, Eugene E, Sur, Cyrille, Cook, Jacquelynn J, Van Laere, Koen, Evelhoch, Jeffrey L

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Preclinical Safety Evaluation and Human Dosimetry of [18F]MK-6240, a Novel PET Tracer for Imaging Neurofibrillary Tangles von Koole, Michel, Lohith, Talakad G., Valentine, John L., Bennacef, Idriss, Declercq, Ruben, Reynders, Tom, Riffel, Kerry, Celen, Sofie, Serdons, Kim, Bormans, Guy, Ferry-Martin, Sandrine, Laroque, Philippe, Walji, Abbas, Hostetler, Eric D., Briscoe, Richard J., de Hoon, Jan, Sur, Cyrille, Van Laere, Koen, Struyk, Arie

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A dual-time-window protocol to reduce acquisition time of dynamic tau PET imaging using [18F]MK-6240 von Kolinger, Guilherme D., Vállez García, David, Lohith, Talakad G., Hostetler, Eric D., Sur, Cyrille, Struyk, Arie, Boellaard, Ronald, Koole, Michel

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In Vivo Evaluation and Dosimetry Estimate for a High Affinity Affibody PET Tracer Targeting PD-L1 von Rubins, Daniel J, Meng, Xiangjun, McQuade, Paul, Klimas, Michael, Getty, Krista, Lin, Shu-An, Connolly, Brett M., O’Malley, Stacey S., Haley, Hyking, Purcell, Mona, Gantert, Liza, Holahan, Marie, Lindgren, Joel, Eklund, Pär, Ekblad, Caroline, Frejd, Fredrik Y., Hostetler, Eric D., González Trotter, Dinko E., Evelhoch, Jeffrey L.

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MK-8719, a Novel and Selective O-GlcNAcase Inhibitor That Reduces the Formation of Pathological Tau and Ameliorates Neurodegeneration in a Mouse Model of Tauopathy von Wang, Xiaohai, Li, Wenping, Marcus, Jacob, Pearson, Michelle, Song, Lixin, Smith, Karen, Terracina, Giuseppe, Lee, Julie, Hong, Kwok-Lam Karen, Lu, Sherry X., Hyde, Lynn, Chen, Shu-Cheng, Kinsley, David, Melchor, Jerry P., Rubins, Daniel J., Meng, Xiangjun, Hostetler, Eric, Sur, Cyrille, Zhang, Lili, Schachter, Joel B., Hess, J. Fred, Selnick, Harold G., Vocadlo, David J., McEachern, Ernest J., Uslaner, Jason M., Duffy, Joseph L., Smith, Sean M.

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cGMP production of the radiopharmaceutical [18F]MK‐6240 for PET imaging of human neurofibrillary tangles von Collier, Thomas Lee, Yokell, Daniel L., Livni, Eli, Rice, Peter A., Celen, Sofie, Serdons, Kim, Neelamegam, Ramesh, Bormans, Guy, Harris, Dawn, Walji, Abbas, Hostetler, Eric D., Bennacef, Idriss, Vasdev, Neil

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Discovery of pyrazolopyrimidine phosphodiesterase 10A inhibitors for the treatment of schizophrenia von Raheem, Izzat T., Schreier, John D., Fuerst, Joy, Gantert, Liza, Hostetler, Eric D., Huszar, Sarah, Joshi, Aniket, Kandebo, Monika, Kim, Somang H., Li, Jing, Ma, Bennett, McGaughey, Georgia, Sharma, Sujata, Shipe, William D., Uslaner, Jason, Vandeveer, George H., Yan, Youwei, Renger, John J., Smith, Sean M., Coleman, Paul J., Cox, Christopher D.

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Continuous Microwave-Assisted Gas–Liquid Segmented Flow Reactor for Controlled Nucleation and Growth of Nanocrystals von Kim, Ki-Joong, Oleksak, Richard P, Hostetler, Eric B, Peterson, Daniel A, Chandran, Padmavathi, Schut, David M, Paul, Brian K, Herman, Gregory S, Chang, Chih-Hung

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Discovery of [11C]MK-8193 as a PET tracer to measure target engagement of phosphodiesterase 10A (PDE10A) inhibitors von Cox, Christopher D., Hostetler, Eric D., Flores, Broc A., Evelhoch, Jeffrey L., Fan, Hong, Gantert, Liza, Holahan, Marie, Eng, Waisi, Joshi, Aniket, McGaughey, Georgia, Meng, Xiangjun, Purcell, Mona, Raheem, Izzat T., Riffel, Kerry, Yan, Youwei, Renger, John J., Smith, Sean M., Coleman, Paul J.

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Brain Imaging of Alzheimer Dementia Patients and Elderly Controls with 18 F-MK-6240, a PET Tracer Targeting Neurofibrillary Tangles von Lohith, Talakad G, Bennacef, Idriss, Vandenberghe, Rik, Vandenbulcke, Mathieu, Salinas, Cristian A, Declercq, Ruben, Reynders, Tom, Telan-Choing, N Florestina, Riffel, Kerry, Celen, Sofie, Serdons, Kim, Bormans, Guy, Tsai, Kuenhi, Walji, Abbas, Hostetler, Eric D, Evelhoch, Jeffrey L, Van Laere, Koen, Forman, Mark, Stoch, Aubrey, Sur, Cyrille, Struyk, Arie

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Training the next generation of radiopharmaceutical scientists von Gee, Antony D., Andersson, Jan, Bhalla, Rajiv, Choe, Yearn Seong, Dick, David W., Herth, Matthias M., Hostetler, Eric D., Jáuregui-Haza, Ulises J., Huang, Ya-Yao, James, Michelle L., Jeong, Jae Min, Korde, Aruna, Kuge, Yuji, Kung, Hank F., Lapi, Suzanne E., Osso, Joao Alberto, Parent, Ephraim, Patt, Marianne, Pricile, Ekoume Fany, Riss, Patrick J., Santos-Oliveira, Ralph, Taylor, Stephen, Vasdev, Neil, Vercouillie, Johnny, Wadsak, Wolfgang, Yang, Zhi, Zhu, Hua, Scott, Peter J.H.

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PET/CT Imaging of 89Zr-N-sucDf-Pembrolizumab in Healthy Cynomolgus Monkeys von Li, Wenping, Wang, Yuchuan, Rubins, Daniel, Bennacef, Idriss, Holahan, Marie, Haley, Hyking, Purcell, Mona, Gantert, Liza, Hseih, SuChun, Judo, Michael, Seghezzi, Wolfgang, Zhang, Shuli, van der Veen, Elly L., Lub-de Hooge, Marjolijn N., de Vries, Elisabeth G.E., Evelhoch, Jeffrey L., Klimas, Michael, Hostetler, Eric D.

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Preclinical evaluation of [11C]L‐235 as a radioligand for Positron Emission Tomography cathepsin K imaging in bone von Bennacef, Idriss, Rubins, Daniel, Riffel, Kerry, Williams, Mangay, Posavec, Diane J., Holahan, Marie A., Purcell, Mona L., Haley, Hyking D., Wolf, Mary, Stachel, Shawn J., Lubbers, Laura S., Wesolowski, Gregg A., Duong, Le T., Hamill, Terence G., Evelhoch, Jeffrey L., Hostetler, Eric D.

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In Vivo Imaging of the Programmed Death Ligand 1 by 18 F PET von González Trotter, Dinko E, Meng, Xiangjun, McQuade, Paul, Rubins, Daniel, Klimas, Michael, Zeng, Zhizhen, Connolly, Brett M, Miller, Patricia J, O'Malley, Stacey S, Lin, Shu-An, Getty, Krista L, Fayadat-Dilman, Laurence, Liang, Linda, Wahlberg, Elisabet, Widmark, Olof, Ekblad, Caroline, Frejd, Fredrik Y, Hostetler, Eric D, Evelhoch, Jeffrey L

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Synthesis, characterization, and monkey PET studies of [18F]MK-1312, a PET tracer for quantification of mGluR1 receptor occupancy by MK-5435 von Hostetler, Eric D., Eng, Waisi, Joshi, Aniket D., Sanabria-Bohórquez, Sandra, Kawamoto, Hiroshi, Ito, Satoru, O'Malley, Stacey, Krause, Stephen, Ryan, Christine, Patel, Shil, Williams, Mangay, Riffel, Kerry, Suzuki, Gentaroh, Ozaki, Satoshi, Ohta, Hisashi, Cook, Jacquelynn, Burns, H. Donald, Hargreaves, Richard

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Evaluation of [18F]MK-0911, a positron emission tomography (PET) tracer for opioid receptor-like 1 (ORL1), in rhesus monkey and human von Hostetler, Eric D., Sanabria-Bohórquez, Sandra, Eng, Waisi, Joshi, Aniket D., Patel, Shailendra, Gibson, Raymond E., O'Malley, Stacey, Krause, Stephen M., Ryan, Christine, Riffel, Kerry, Bi, Sheng, Okamoto, Osamu, Kawamoto, Hiroshi, Ozaki, Satoshi, Ohta, Hisashi, de Groot, Tjibbe, Bormans, Guy, Depré, Marleen, de Hoon, Jan, De Lepeleire, Inge, Reynders, Tom, Cook, Jacquelynn J., Burns, H. Donald, Egan, Michael, Cho, William, van Laere, Koen, Hargreaves, Richard J.

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Synthesis, characterization, and monkey positron emission tomography (PET) studies of [18F]Y1-973, a PET tracer for the neuropeptide Y Y1 receptor von Hostetler, Eric D., Sanabria-Bohórquez, Sandra, Fan, Hong, Zeng, Zhizhen, Gantert, Liza, Williams, Mangay, Miller, Patricia, O'Malley, Stacey, Kameda, Minoru, Ando, Makoto, Sato, Nagaaki, Ozaki, Satoshi, Tokita, Shigeru, Ohta, Hisashi, Williams, David, Sur, Cyrille, Cook, Jacquelynn J., Burns, H. Donald, Hargreaves, Richard

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Ex Vivo Imaging of Pancreatic Beta Cells using a Radiolabeled GLP-1 Receptor Agonist von Connolly, Brett M., Vanko, Amy, McQuade, Paul, Guenther, Ilonka, Meng, Xiangjun, Rubins, Daniel, Waterhouse, Rikki, Hargreaves, Richard, Sur, Cyrille, Hostetler, Eric

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