Cryo-EM structure of GABA transporter 1 reveals substrate recognition and transport mechanism von Nayak, Smruti Ranjan, Joseph, Deepthi, Höfner, Georg, Dakua, Archishman, Athreya, Arunabh, Wanner, Klaus T., Kanner, Baruch I., Penmatsa, Aravind

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Development of a Potent Nurr1 Agonist Tool for In Vivo Applications von Vietor, Jan, Gege, Christian, Stiller, Tanja, Busch, Romy, Schallmayer, Espen, Kohlhof, Hella, Höfner, Georg, Pabel, Jörg, Marschner, Julian A., Merk, Daniel

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Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation von Arifi, Silvia, Marschner, Julian A., Pollinger, Julius, Isigkeit, Laura, Heitel, Pascal, Kaiser, Astrid, Obeser, Lennart, Höfner, Georg, Proschak, Ewgenij, Knapp, Stefan, Chaikuad, Apirat, Heering, Jan, Merk, Daniel

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Synthesis of 4-substituted nipecotic acid derivatives and their evaluation as potential GABA uptake inhibitors von Hellenbrand, Tim, Höfner, Georg, Wein, Thomas, Wanner, Klaus T.

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MS Binding Assays for D1 and D5 Dopamine Receptors von Neiens, Patrick, Höfner, Georg, Wanner, Klaus Theodor

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Novel Allosteric Ligands of γ‑Aminobutyric Acid Transporter 1 (GAT1) by MS Based Screening of Pseudostatic Hydrazone Libraries von Hauke, Tobias J, Wein, Thomas, Höfner, Georg, Wanner, Klaus T

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Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives with N‐Arylalkynyl Substituents von Lutz, Toni, Wein, Thomas, Höfner, Georg, Wanner, Klaus T.

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Identification of ligands binding to MB327-PAM-1, a binding pocket relevant for resensitization of nAChRs von Kaiser, Jesko, Gertzen, Christoph G.W., Bernauer, Tamara, Nitsche, Valentin, Höfner, Georg, Niessen, Karin V., Seeger, Thomas, Paintner, Franz F., Wanner, Klaus T., Steinritz, Dirk, Worek, Franz, Gohlke, Holger

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MS Transport Assays for γ‑Aminobutyric Acid TransportersAn Efficient Alternative for Radiometric Assays von Schmitt, Sebastian, Höfner, Georg, Wanner, Klaus T

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Structure-Guided Design of Nurr1 Agonists Derived from the Natural Ligand Dihydroxyindole von Sai, Minh, Vietor, Jan, Kornmayer, Moritz, Egner, Markus, López-García, Úrsula, Höfner, Georg, Pabel, Jörg, Marschner, Julian A., Wein, Thomas, Merk, Daniel

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Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors von Quandt, Gabriele, Höfner, Georg, Wanner, Klaus T.

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Simultaneous LC-ESI-MS/MS Quantification of Levosimendan and Its Metabolites for Therapeutic Drug Monitoring of Cardiac Surgery Patients von Kipka, Hannah, Tomasi, Roland, Hübner, Max, Liebchen, Uwe, Hagl, Christian, Wanner, Klaus T., Mannell, Hanna, Höfner, Georg

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MS Binding Assays for the Three Monoamine Transporters Using the Triple Reuptake Inhibitor (1R,3S)-Indatraline as Native Marker von Grimm, Stefanie H., Höfner, Georg, Wanner, Klaus T.

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Development of New Photoswitchable Azobenzene Based γ‑Aminobutyric Acid (GABA) Uptake Inhibitors with Distinctly Enhanced Potency upon Photoactivation von Lutz, Toni, Wein, Thomas, Höfner, Georg, Pabel, Jörg, Eder, Matthias, Dine, Julien, Wanner, Klaus T

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Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease... von Zaręba, Paula, Łątka, Kamil, Mazur, Gabriela, Gryzło, Beata, Pasieka, Anna, Godyń, Justyna, Panek, Dawid, Skrzypczak-Wiercioch, Anna, Höfner, Georg C., Latacz, Gniewomir, Maj, Maciej, Espargaró, Alba, Sabaté, Raimon, Jóźwiak, Krzysztof, Wanner, Klaus T., Sałat, Kinga, Malawska, Barbara, Kulig, Katarzyna, Bajda, Marek

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Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions von Petrera, Marilena, Wein, Thomas, Allmendinger, Lars, Sindelar, Miriam, Pabel, Jörg, Höfner, Georg, Wanner, Klaus T.

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Simultaneous Multiple MS Binding Assays Addressing D1 and D2 Dopamine Receptors von Schuller, Marion, Höfner, Georg, Wanner, Klaus T.

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Different Binding Modes of Small and Large Binders of GAT1 von Wein, Thomas, Petrera, Marilena, Allmendinger, Lars, Höfner, Georg, Pabel, Jörg, Wanner, Klaus T.

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Development and validation of an LC-ESI-MS/MS method for the triple reuptake inhibitor indatraline enabling its quantification in MS Binding Assays von Grimm, Stefanie H., Höfner, Georg, Wanner, Klaus T.

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Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity von Gryzło, Beata, Zaręba, Paula, Malawska, Katarzyna, Mazur, Gabriela, Rapacz, Anna, Ła̧tka, Kamil, Höfner, Georg C, Latacz, Gniewomir, Bajda, Marek, Sałat, Kinga, Wanner, Klaus T, Malawska, Barbara, Kulig, Katarzyna

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