IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: improved PK, hERG and metabolic profiles von Nair, Anilkumar G, Wong, Michael K C, Shu, Youheng, Jiang, Yueheng, Jenh, Chung-Her, Kim, Seong Heon, Yang, De-Yi, Zeng, Qingbei, Shao, Yuefei, Zawacki, Lisa Guise, Duo, Jingqi, McGuinness, Brian F, Carroll, Carolyn Diianni, Hobbs, Doug W, Shih, Neng-Yang, Rosenblum, Stuart B, Kozlowski, Joseph A

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Deriving Knowledge through Data Mining High-Throughput Screening Data von Diller, David J, Hobbs, Doug W

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Understanding hERG inhibition with QSAR models based on a one-dimensional molecular representation von Diller, David J, Hobbs, Doug W

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Design, synthesis, and evaluation of tetrahydroquinoline and pyrrolidine sulfonamide carbamates as γ-secretase inhibitors von Guo, Tao, Gu, Huizhong, Hobbs, Doug W., Rokosz, Laura L., Stauffer, Tara M., Jacob, Biji, Clader, John W.

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III. Identification of novel CXCR3 chemokine receptor antagonists with a pyrazinyl–piperazinyl–piperidine scaffold von Kim, Seong Heon, Anilkumar, Gopinadhan N., Zawacki, Lisa Guise, Zeng, Qingbei, Yang, De-Yi, Shao, Yuefei, Dong, Guizhen, Xu, Xiaolian, Yu, Wensheng, Jiang, Yueheng, Jenh, Chung-Her, Hall, James W., Carroll, Carolyn DiIanni, Hobbs, Doug W., Baldwin, John J., McGuinness, Brian F., Rosenblum, Stuart B., Kozlowski, Joseph A., Shankar, Bandarpalle B., Shih, Neng-Yang

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II. SAR studies of pyridyl–piperazinyl-piperidine derivatives as CXCR3 chemokine antagonists von Shao, Yuefei, Anilkumar, Gopinadhan N., Carroll, Carolyn DiIanni, Dong, Guizhen, Hall, James W., Hobbs, Doug W., Jiang, Yueheng, Jenh, Chung-Her, Kim, Seong Heon, Kozlowski, Joseph A., McGuinness, Brian F., Rosenblum, Stuart B., Schulman, Inna, Shih, Neng-Yang, Shu, Youheng, Wong, Michael K.C., Yu, Wensheng, Zawacki, Lisa Guise, Zeng, Qingbei

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Novel CXCR3 antagonists with a piperazinyl-piperidine core von McGuinness, Brian F., Carroll, Carolyn DiIanni, Zawacki, Lisa Guise, Dong, Guizhen, Yang, Cangming, Hobbs, Doug W., Jacob-Samuel, Biji, Hall, James W., Jenh, Chung-Her, Kozlowski, Joseph A., Anilkumar, Gopinadhan N., Rosenblum, Stuart B.

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Privileged structure-based combinatorial libraries targeting G protein-coupled receptors von Guo, Tao, Hobbs, Doug W

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Orally active, nonpeptide oxytocin antagonists von Evans, Ben E, Leighton, James L, Rittle, Kenneth E, Gilbert, Kevin F, Lundell, George F, Gould, Norman P, Hobbs, Doug W, DiPardo, Robert M, Veber, Daniel F, Pettibone, Douglas J, Clineschmidt, Bradley V, Anderson, Paul S, Freidinger, Roger M

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Discovery and SAR of 4-amino-2-biarylbutylurea MCH 1 receptor antagonists through solid-phase parallel synthesis von Guo, Tao, Hunter, Rachael C., Gu, Huizhong, Rokosz, Laura L., Stauffer, Tara M., Hobbs, Doug W.

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Discovery of tetralin ureas as potent melanin concentrating hormone 1 receptor antagonists von Guo, Tao, Gu, Huizhong, Hobbs, Doug W., Busler, Dennis E., Rokosz, Laura L.

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Discovery and SAR of biaryl piperidine MCH1 receptor antagonists through solid-phase encoded combinatorial synthesis von Guo, Tao, Shao, Yuefei, Qian, Gang, Rokosz, Laura L., Stauffer, Tara M., Hunter, Rachael C., Babu, Suresh D., Gu, Huizhong, Hobbs, Doug W.

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Development of Orally Active Oxytocin Antagonists:  Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d... von Bell, Ian M, Erb, Jill M, Freidinger, Roger M, Gallicchio, Steven N, Guare, James P, Guidotti, Maribeth T, Halpin, Rita A, Hobbs, Doug W, Homnick, Carl F, Kuo, Michelle S, Lis, Edward V, Mathre, David J, Michelson, Stuart R, Pawluczyk, Joseph M, Pettibone, Douglas J, Reiss, Duane R, Vickers, Stanley, Williams, Peter D, Woyden, Carla J

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Synthesis of diphenyl thioether derivatives of peptides and aminoacids von Hobbs, Doug W., Still, W.Clark

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Synthesis and anti-herpes virus activity of acyclic 2'-deoxyguanosine analogs related to 9-[(1,3-dihydroxy-2-propoxy)methyl]guanine von Martin, John C, McGee, Danny P. C, Jeffrey, Gary A, Hobbs, Doug W, Smee, Donald F, Matthews, Thomas R, Verheyden, Julian P. H

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Discovery and SAR of 4-amino-2-biarylbutylurea MCH 1 receptor antagonists through solid-phase parallel synthesis: G-protein-coupled receptors in drug discovery von TAO GUO, HUNTER, Rachael C, HUIZHONG GU, ROKOSZ, Laura L, STAUFFER, Tara M, HOBBS, Doug W

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LIBRARY DESIGN CONCEPTS AND IMPLEMENTATION STRATEGIES1 von Hobbs, Doug W., Guo, Tao

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Discovery and SAR of biaryl piperidine MCH1 receptor antagonists through solid-phase encoded combinatorial synthesis: G-protein-coupled receptors in drug discovery von TAO GUO, YUEFEI SHAO, GANG QIAN, ROKOSZ, Laura L, STAUFFER, Tara M, HUNTER, Rachael C, BABU, Suresh D, HUIZHONG GU, HOBBS, Doug W

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LIBRARY DESIGN CONCEPTS AND IMPLEMENTATION STRATEGIES von Hobbs, Doug W., Guo, Tao

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Combinatorial library methods and protocols von English, Lisa Bellavance

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