Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity von Gryzło, Beata, Zaręba, Paula, Malawska, Katarzyna, Mazur, Gabriela, Rapacz, Anna, Ła̧tka, Kamil, Höfner, Georg C, Latacz, Gniewomir, Bajda, Marek, Sałat, Kinga, Wanner, Klaus T, Malawska, Barbara, Kulig, Katarzyna

Volltext

Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease... von Zaręba, Paula, Łątka, Kamil, Mazur, Gabriela, Gryzło, Beata, Pasieka, Anna, Godyń, Justyna, Panek, Dawid, Skrzypczak-Wiercioch, Anna, Höfner, Georg C., Latacz, Gniewomir, Maj, Maciej, Espargaró, Alba, Sabaté, Raimon, Jóźwiak, Krzysztof, Wanner, Klaus T., Sałat, Kinga, Malawska, Barbara, Kulig, Katarzyna, Bajda, Marek

Volltext

Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity von Zaręba, Paula, Sałat, Kinga, Höfner, Georg C., Łątka, Kamil, Bajda, Marek, Latacz, Gniewomir, Kotniewicz, Krzysztof, Rapacz, Anna, Podkowa, Adrian, Maj, Maciej, Jóźwiak, Krzysztof, Filipek, Barbara, Wanner, Klaus T., Malawska, Barbara, Kulig, Katarzyna

Volltext

Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice von Zaręba, Paula, Gryzło, Beata, Malawska, Katarzyna, Sałat, Kinga, Höfner, Georg C., Nowaczyk, Alicja, Fijałkowski, Łukasz, Rapacz, Anna, Podkowa, Adrian, Furgała, Anna, Żmudzki, Paweł, Wanner, Klaus T., Malawska, Barbara, Kulig, Katarzyna

Volltext

Development, validation and application of a 96-well enzymatic assay based on LC-ESI-MS/MS quantification for the screening of selective inhibitors against Mycobacterium tuberculos... von Cattaneo, Giulia, Ubiali, Daniela, Calleri, Enrica, Rabuffetti, Marco, Höfner, Georg C., Wanner, Klaus T., De Moraes, Marcela C., Martinelli, Leonardo K.B., Santos, Diógenes Santiago, Speranza, Giovanna, Massolini, Gabriella

Volltext

2-Substituted 4-hydroxybutanamides as potential inhibitors of γ-aminobutyric acid transporters mGAT1–mGAT4: Synthesis and biological evaluation von Kowalczyk, Paula, Sałat, Kinga, Höfner, Georg C., Guzior, Natalia, Filipek, Barbara, Wanner, Klaus T., Kulig, Katarzyna

Volltext

Synthesis, biological evaluation and structure–activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides von Kowalczyk, Paula, Sałat, Kinga, Höfner, Georg C., Mucha, Marta, Rapacz, Anna, Podkowa, Adrian, Filipek, Barbara, Wanner, Klaus T., Kulig, Katarzyna

Volltext

Synthesis and biological evaluation of 4-hydroxy-4-(4-methoxyphenyl)-substituted proline and pyrrolidin-2-ylacetic acid derivatives as GABA uptake inhibitors von Zhao, Xueqing, Pabel, Jörg, Höfner, Georg C., Wanner, Klaus T.

Volltext

Synthesis and biological evaluation of new derivatives of 2-substituted 4-hydroxybutanamides as GABA uptake inhibitors von Kulig, Katarzyna, Więckowski, Krzysztof, Więckowska, Anna, Gajda, Justyna, Pochwat, Bartłomiej, Höfner, Georg C., Wanner, Klaus T., Malawska, Barbara

Volltext

Synthesis and pharmacological properties of new GABA uptake inhibitors von Sałat, Kinga, Więckowska, Anna, Więckowski, Krzysztof, Höfner, Georg C., Kamiński, Jacek, Wanner, Klaus T., Malawska, Barbara, Filipek, Barbara, Kulig, Katarzyna

Volltext

Synthesis and biological evaluation of α- and β-hydroxy substituted amino acid derivatives as potential mGAT1–4 inhibitors von Andreß, Janina C., Böck, Michael C., Höfner, Georg, Wanner, Klaus T.

Volltext

Azidobupramine, an Antidepressant-Derived Bifunctional Neurotransmitter Transporter Ligand Allowing Covalent Labeling and Attachment of Fluorophores von Kirmeier, Thomas, Gopalakrishnan, Ranganath, Gormanns, Vanessa, Werner, Anna M, Cuboni, Serena, Rudolf, Georg C, Höfner, Georg, Wanner, Klaus T, Sieber, Stephan A, Schmidt, Ulrike, Holsboer, Florian, Rein, Theo, Hausch, Felix

Volltext

N‐Substituted Nipecotic Acids as (S)‐SNAP‐5114 Analogues with Modified Lipophilic Domains von Böck, Michael C., Höfner, Georg, Wanner, Klaus T.

Volltext

Deletion of the γ-Aminobutyric Acid Transporter 2 (GAT2 and SLC6A13) Gene in Mice Leads to Changes in Liver and Brain Taurine Contents von Zhou, Yun, Holmseth, Silvia, Guo, Caiying, Hassel, Bjørnar, Höfner, Georg, Huitfeldt, Henrik S., Wanner, Klaus T., Danbolt, Niels C.

Volltext

Withdrawal: K.T. Wanner et al. “MS‐based screening of small amino acid derived oxime libraries for hGAT3 inhibitors” von Andreß, Janina C., Höfner, Georg, Wanner, Klaus T.

Volltext

Parsing and Printing of and with Triples von Joosten, Sebastiaan J. C.

Volltext

Algebra for Quantitative Information Flow von McIver, A. K., Morgan, C. C., Rabehaja, T.

Volltext

N‐Substituted Nipecotic Acids as (S )‐SNAP‐5114 Analogues with Modified Lipophilic Domains von Böck, Michael C, Höfner, Georg, Wanner, Klaus T

Volltext bestellen

Synthesis and biological evaluation of α- and β-hydroxy substituted amino acid derivatives as potential mGAT1-4 inhibitors von Andreß, Janina C, Böck, Michael C, Höfner, Georg, Wanner, Klaus T

Volltext bestellen

NMDA-NR2B subtype selectivity of stereoisomeric 2-(1,2,3,4-tetrahydro-1-isoquinolyl)ethanol derivatives von Höfner, Georg, Hoesl, Cornelia E., Parsons, Chris, Quack, Günther, Wanner, Klaus T.

Volltext