Synthesis and Evaluation of a Series of Novel 2-[(4-Chlorophenoxy)methyl]- benzimidazoles as Selective Neuropeptide Y Y1 Receptor Antagonists von Zarrinmayeh, Hamideh, Nunes, Anne M, Ornstein, Paul L, Zimmerman, Dennis M, Arnold, M. Brian, Schober, Douglas A, Gackenheimer, Susan L, Bruns, Robert F, Hipskind, Philip A, Britton, Thomas C, Cantrell, Buddy E, Gehlert, Donald R

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Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists von Zarrinmayeh, Hamideh, Zimmerman, Dennis M., Cantrell, Buddy E., Schober, Douglas A., Bruns, Robert E., Gackenheimer, Susan L., Ornstein, Paul L., Hipskind, Philip A., Britton, Thomas C., Gehlert, Donald R.

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Acyl Sulfonamide Anti-Proliferatives:  Benzene Substituent Structure−Activity Relationships for a Novel Class of Antitumor Agents von Lobb, Karen L, Hipskind, Philip A, Aikins, James A, Alvarez, Enrique, Cheung, Yiu-Yin, Considine, Eileen L, De Dios, Alfonso, Durst, Gregory L, Ferritto, Rafael, Grossman, Cora Sue, Giera, Deborah D, Hollister, Beth A, Huang, Zhongping, Iversen, Philip W, Law, Kevin L, Li, Tiechao, Lin, Ho-Shen, Lopez, Beatriz, Lopez, Jose E, Cabrejas, Luisa M. Martin, McCann, Denis J, Molero, Victoriano, Reilly, John E, Richett, Michael E, Shih, Chuan, Teicher, Beverly, Wikel, James H, White, Wesley T, Mader, Mary M

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[3H]LY303870, a Novel Nonpeptide Radioligand for the NK‐1 Receptor von Gehlert, D. R., Schober, D. A., Hipskind, P. A., Gitter, B. D., Howbert, J. J.

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Structure-activity relationships of a series of benzothiophene-derived NPY Y1 antagonists: Optimization of the C-2 side chain von Britton, Thomas C., Spinazze, Patrick G., Hipskind, Philip A., Zimmerman, Dennis M., Zarrinmayeh, Hamideh, Schober, Douglas A., Gehlert, Donald R., Bruns, Robert F.

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Structure-activity relationships of a series of 1-substituted-4-methylbenzimidazole neuropeptide Y-1 receptor antagonists von Zimmerman, Dennis M., Cantrell, Buddy E., Smith, Edward C.R., Nixon, James A., Bruns, Robert F., Gitter, Bruce, Hipskind, Philip A., Ornstein, Paul L., Zarrinmayeh, Hamideh, Britton, Thomas C., Schober, Douglas A., Gehlert, Donald R.

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Potent and Selective 1,2,3-Trisubstituted Indole NPY Y-1 Antagonists von Hipskind, Philip A, Lobb, Karen L, Nixon, James A, Britton, Thomas C, Bruns, Robert F, Catlow, John, Dieckman-McGinty, Donna K, Gackenheimer, Susan L, Gitter, Bruce D, Iyengar, Smriti, Schober, Douglas A, Simmons, Rosa M. A, Swanson, Steve, Zarrinmayeh, Hamideh, Zimmerman, Dennis M, Gehlert, Donald R

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Neuropeptide Y receptor antagonists in obesity von Gehlert, Donald R, Hipskind, Philip A

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Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs von Vieth, Michal, Siegel, Miles G, Higgs, Richard E, Watson, Ian A, Robertson, Daniel H, Savin, Kenneth A, Durst, Gregory L, Hipskind, Philip A

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Recent developments in our understanding of the physiological role of PP-fold peptide receptor subtypes von Berglund, Magnus M, Hipskind, Philip A, Gehlert, Donald R

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A novel cephalosporin dehydrothiazine ring cleavage mode von Lunn, W.H.W., Hipskind, Philip A.

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Expedited discovery of second generation NK-1 antagonists: identification of a nonbasic aryloxy substituent von Fritz, James E., Hipskind, Philip A., Lobb, Karen L., Nixon, James A., Threlkeld, Penny G., Gitter, Bruce D., McMillian, Carl L., Kaldor, Stephen W.

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The non-peptide NK-1 receptor antagonist LY303870 inhibits neurogenic dural inflammation in guinea pigs von Phebus, L A, Johnson, K W, Stengel, P W, Lobb, K L, Nixon, J A, Hipskind, P A

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3-Aryl-1,2-diacetamidopropane Derivatives as Novel and Potent NK-1 Receptor Antagonists von Hipskind, Philip A, Howbert, J. Jeffry, Bruns, Robert F, Cho, Steven S. Y, Crowell, Thomas A, Foreman, Mark M, Gehlert, Donald R, Iyengar, Smriti, Johnson, Kirk W, Krushinski, Joseph H, Li, Dominic L, Lobb, Karen L, Mason, Norman R, Muehl, Brian S, Nixon, James A, Phebus, Lee A, Regoli, Domenico, Simmons, Rosa M, Threlkeld, Penny G, Waters, Diane C, Gitter, Bruce D

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Stress and central Urocortin increase anxiety-like behavior in the social interaction test via the CRF1 receptor von GEHLERT, Donald R, SHEKHAR, Anantha, MORIN, S. Michelle, HIPSKIND, Phillip A, ZINK, Charity, GACKENHEIMER, Susan L, SHAW, Janice, FITZ, Stephanie D, SAJDYK, Tammy J

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Peripheral effects of three novel non-peptide tachykinin NK1 receptor antagonists in the anaesthetized rat von Cellier, E, Fayolle, C, Hipskind, P A, Iyengar, S, Couture, R

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Substance P Regulates PTH Secretion through the Neurokinin-1 Receptor von Sells Galvin, Rachelle J., Babbey, Lael E., Hipskind, Philip A., Lamar, Tiffanie, George, Carolyn A., Baez, Melvyn, Gitter, Bruce D.

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Stress-related neuropeptides and alcoholism: CRH, NPY, and beyond von Ciccocioppo, Roberto, Gehlert, Donald R, Ryabinin, Andrey, Kaur, Simranjit, Cippitelli, Andrea, Thorsell, Annika, Lê, Anh D, Hipskind, Philip A, Hamdouchi, Chafiq, Lu, Jianliang, Hembre, Erik J, Cramer, Jeffrey, Song, Min, McKinzie, David, Morin, Michelle, Economidou, Daina, Stopponi, Serena, Cannella, Nazzareno, Braconi, Simone, Kallupi, Marsida, de Guglielmo, Giordano, Massi, Maurizio, George, David T, Gilman, Jody, Hersh, Jacqueline, Tauscher, Johannes T, Hunt, Stephen P, Hommer, Daniel, Heilig, Markus

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A total asymmetric synthesis of the isolactarane sesquiterpene (−)-merulidial von Trost, Barry M., Hipskind, Philip A.

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NEUROPEPTIDEY (NPY) AND OBESITY: POTENT AND SELECTIVE NONPEPTIDEY1 RECEPTOR ANTAGONISTS REDUCE FOOD CONSUMPTION AND BODY WEIGHT IN RODENTS von Gehlert, D R, Tinsley, F C, Zimmerman, D, Hipskind, P A, Zarrinmayeh, H, Britton, T, Bruns, R F, Iyengar, S

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