SUBSTITUTED 1H-PYRROLO[3,2-B]PYRIDINE COMPOUNDS AND METHODS OF USE THEREOF von Schulze, Volker, Bömer, Ulf, Lechner, Christian, Mengel, Anne, Furst, Laura, Berger, Markus, Faria Alvares De Lemos, Adelaide Clara, Brezezinka, Krzysztof, Mortier, Jérémie Xavier, Lienau, Philip, Rupaimoole, Rajesha, Christian, Sven, Orsi, Douglas, Hillig, v, Madec, Amael, Corsello, Steven, Shekhar, Mrinal, Handing, Katarzyna, Kaulfuss, Stefan, McKinney, David

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Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2 von Eggert, Erik, Hillig, Roman C, Koehr, Silke, Stöckigt, Detlef, Weiske, Jörg, Barak, Naomi, Mowat, Jeffrey, Brumby, Thomas, Christ, Clara D, ter Laak, Antonius, Lang, Tina, Fernandez-Montalvan, Amaury E, Badock, Volker, Weinmann, Hilmar, Hartung, Ingo V, Barsyte-Lovejoy, Dalia, Szewczyk, Magdalena, Kennedy, Steven, Li, Fengling, Vedadi, Masoud, Brown, Peter J, Santhakumar, Vijayaratnam, Arrowsmith, Cheryl H, Stellfeld, Timo, Stresemann, Carlo

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Discovery and Characterization of BAY-184: A New Potent and Selective Acylsulfonamide-Benzofuran In Vivo-Active KAT6AB Inhibitor von ter Laak, Antonius, Hillig, Roman C., Ferrara, Steven J., Korr, Daniel, Barak, Naomi, Lienau, Philip, Herbert, Simon, Fernández-Montalván, Amaury Ernesto, Neuhaus, Roland, Gorjánácz, Mátyás, Puetter, Vera, Badock, Volker, Bone, Wilhelm, Strathdee, Craig, Siegel, Franziska, Schatz, Christoph, Nowak-Reppel, Katrin, Doehr, Olaf, Gradl, Stefan, Hartung, Ingo V., Meyerson, Matthew, Bouché, Léa

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BAY 2927088: The first non-covalent, potent, and selective tyrosine kinase inhibitor targeting EGFR exon 20 insertions and C797S resistance mutations in NSCLC von Siegel, F., Siegel, S., Graham, K., Karsli-Uzunbas, G., Korr, D., Schroeder, J., Boemer, U., Hillig, R.C., Mortier, J., Niehues, M., Golfier, S., Schulze, V., Menz, S., Kamburov, A., Hermsen, M., Cherniak, A., Eis, K., Eheim, A., Meyerson, M., Greulich, H.

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Gene Expression–Based Molecular Test as Diagnostic Aid for the Differential Diagnosis of Psoriasis and Eczema in Formalin-Fixed and Paraffin-Embedded Tissue, Microbiopsies, and Tap... von Fischer, Felix, Doll, Anais, Uereyener, Deniz, Roenneberg, Sophie, Hillig, Christina, Weber, Lucca, Hackert, Verena, Meinel, Martin, Farnoud, Ali, Seiringer, Peter, Thomas, Jenny, Anand, Philipp, Graner, Larissa, Schlenker, Franziska, Zengerle, Roland, Jonsson, Pontus, Jargosch, Manja, Theis, Fabian J., Schmidt-Weber, Carsten B., Biedermann, Tilo, Howell, Michael, Reich, Kristian, Eyerich, Kilian, Menden, Michael, Garzorz-Stark, Natalie, Lauffer, Felix, Eyerich, Stefanie

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Optimization of allosteric MEK inhibitors. Part 2: Taming the sulfamide group balances compound distribution properties von Hartung, Ingo V., Hammer, Stefanie, Hitchcock, Marion, Neuhaus, Roland, Scholz, Arne, Siemeister, Gerhard, Bohlmann, Rolf, Hillig, Roman C., Pühler, Florian

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Optimization of allosteric MEK inhibitors. Part 1: Venturing into underexplored SAR territories von Hartung, Ingo V., Hitchcock, Marion, Pühler, Florian, Neuhaus, Roland, Scholz, Arne, Hammer, Stefanie, Petersen, Kirstin, Siemeister, Gerhard, Brittain, Dominic, Hillig, Roman C.

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Modular Assembly of Allosteric MEK Inhibitor Structural Elements Unravels Potency and Feedback-Modulation Handles von Hartung, Ingo V., Pühler, Florian, Neuhaus, Roland, Scholz, Arne, Siemeister, Gerhard, Geisler, Jens, Hillig, Roman C., von Ahsen, Oliver, Hitchcock, Marion

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Back Cover: Modular Assembly of Allosteric MEK Inhibitor Structural Elements Unravels Potency and Feedback-Modulation Handles (ChemMedChem 12/2015) von Hartung, Ingo V., Pühler, Florian, Neuhaus, Roland, Scholz, Arne, Siemeister, Gerhard, Geisler, Jens, Hillig, Roman C., von Ahsen, Oliver, Hitchcock, Marion

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Abstract 5239: Probing the cancer epigenome: empowering target validation by open innovation von Hartung, Ingo V., Arrowsmith, Cheryl, Badock, Volker, Barak, Naomi, Berger, Markus, Brown, Peter J., Christ, Clara D., Eggert, Erik, Egner, Ursula, Fedorov, Oleg, Fernandez-Montalvan, Amaury E., Gorjanacz, Matyas, Haegebarth, Andrea, Haendler, Bernard, Hillig, Roman C., Holton, Simon H., Huber, Kilian V., Koo, Seong J., Laak, Antonius ter, Mueller, Susanne, Mueller-Fahrnow, Anke, Scholten, Cora, Siegel, Stephan, Stellfeld, Timo, Stoeckigt, Detlef, Stresemann, Carlo, Vedadi, Masoud, Weiske, Joerg, Weinmann, Hilmar

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The crystal structure of rna1p: a new fold for a GTPase-activating protein von Hillig, R C, Renault, L, Vetter, I R, Drell, 4th, T, Wittinghofer, A, Becker, J

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High-resolution structure of HLA-A0201 in complex with a tumour-specific antigenic peptide encoded by the MAGE-A4 gene von Hillig, R C, Coulie, P G, Stroobant, V, Saenger, W, Ziegler, A, Hülsmeyer, M

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Adição de aparas de papel reciclável na fabricação de chapas de madeira aglomerada von Calegari, Leandro, Haselein, Clovis R., Barros, Marcos V., Scaravelli, Tobias L., Dacosta, Lourdes Patricia E., Pedrazzi, Cristiane, Hillig, Everton

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Structure of wild type Plk1 kinase domain in complex with a selective DARPin von Carrondo, M.A., Hillig, R.C., Bandeiras, T.M., Matias, P.M., Eberspaecher, U., Fanghanel, J., Thomaz, M., Miranda, S., Crusius, K., Putter, V., Amstutz, P., Gulotti-Georgieva, M., Binz, K., Holz, C., Schmitz, A.A., Lang, C.

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Adição de aparas de papel reciclável na fabricação de chapas de madeira aglomerada von Leandro Calegari, Clovis R. Haselein, Marcos V. Barros, Tobias L. Scaravelli, Lourdes Patricia E. Dacosta, Cristiane Pedrazzi, Everton Hillig

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Avaliação da degradação não-isotérmica de madeira através de termogravimetria-TGA von Bianchi, Otávio, Dal Castel, Charles, Oliveira, Ricardo V. B. de, Bertuoli, Paula T., Hillig, Everton

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Avaliação da degradação não-isotérmica de madeira através de termogravimetria-TGA Nonisothermal degradation of wood using thermogravimetric measurements von Otávio Bianchi, Charles Dal Castel, Ricardo V. B. de Oliveira, Paula T. Bertuoli, Everton Hillig

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ADIÇÃO DE APARAS DE PAPEL RECICLÁVEL NA FABRICAÇÃO DE CHAPAS DE MADEIRA AGLOMERADA von Everton Hillig, Cristiane Pedrazzi, Lourdes Patricia E. Dacosta, Tobias L. Scaravelli, Marcos V. Barros, Clovis R. Haselein, Leandro Calegari

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Adição de aparas de papel reciclável na fabricação de chapas de madeiraaglomerada von Leandro Calegari, Clovis R. Haselein, Marcos V. Barros, Tobias L. Scaravelli, Lourdes Patricia E. Dacosta, Cristiane Pedrazzi, Everton Hillig

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Avaliação da degradação não-isotérmica de madeira através de termogravimetria-TGA von Otávio Bianchi, Charles Dal Castel, Ricardo V. B. de Oliveira, Paula T. Bertuoli, Everton Hillig

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