N-Nitrosamine Formation in Pharmaceutical Solid Drug Products: Experimental Observations von Moser, Justin, Ashworth, Ian W., Harris, Laurence, Hillier, Michael C., Nanda, Kausik K., Scrivens, Garry

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Synthesis of hydantoins and dihydrouracils via thermally-promoted cyclization of ureidoacetamides von Hillier, Michael C., Gong, Hai-Hua, Clyne, Dean S., Babcock, Martin J.

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Stereoselective Formation of Carbon−Carbon Bonds via SN2-Displacement:  Synthesis of Substituted Cycloalkyl[b]indoles von Hillier, Michael C, Marcoux, Jean-François, Zhao, Dalian, Grabowski, Edward J. J, McKeown, Arlene E, Tillyer, Richard D

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Enantioselective Total Syntheses of Ircinal A and Related Manzamine Alkaloids von Martin, Stephen F, Humphrey, John M, Ali, Amjad, Hillier, Michael C

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Stereoselective Carbon−Carbon Bond Formation via the Mitsunobu Displacement of Chiral Secondary Benzylic Alcohols von Hillier, Michael C, Desrosiers, Jean-Nicolas, Marcoux, Jean-François, Grabowski, Edward J. J

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Risk Assessment of the Leachables’ Profile for Small-Molecule Pharmaceutical Drug Substances von Reddy, Rajarathnam E, Hu, Wenbin, Lowry, Brian R, Fogle, Jace L, Malick, Robert E, Erexson, Greg, Westerberg, John M, Carragher, Adelia L, Robinson, Emily E, Orihuela, Carlos A, Hillier, Michael C, Davis, Steven R, Kruk, Paul E, Ide, Nathan D, Mlinar, Laurie, Mulhern, Mathew M, Engstrom, Kenneth M, Chaaya, Elie, McKee, Laura A, Manning, Patrick E, Tirino, Pasquale, Joudioux, Roberta, Cornelio, Lisa

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Stereoselective Preparation of a Cyclopentane-Based NK1 Receptor Antagonist Bearing an Unsymmetrically Substituted Sec−Sec Ether von Kuethe, Jeffrey T, Marcoux, Jean-Francois, Wong, Audrey, Wu, Jimmy, Hillier, Michael C, Dormer, Peter G, Davies, Ian W, Hughes, David L

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Asymmetric Synthesis of 1,2,3-Trisubstituted Cyclopentanes and Cyclohexanes as Key Components of Substance P Antagonists von Kuethe, Jeffrey T, Wong, Audrey, Wu, Jimmy, Davies, Ian W, Dormer, Peter G, Welch, Christopher J, Hillier, Michael C, Hughes, David L, Reider, Paul J

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A One-Pot Preparation of 1,3-Disubstituted Azetidines von Hillier, Michael C, Chen, Cheng-yi

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Practical, Highly Convergent, Asymmetric Synthesis of a Selective PPARγ Modulator von Maligres, Peter E, Humphrey, Guy R, Marcoux, Jean-François, Hillier, Michael C, Zhao, Dalian, Krska, Shane, Grabowski, Edward J. J

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Stereoselective synthesis from a process research perspective von Hillier, Michael C, Reider, Paul J

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Cyclopropane-Derived Peptidomimetics. Design, Synthesis, Evaluation, and Structure of Novel HIV-1 Protease Inhibitors von Martin, Stephen F, Dorsey, Gordon O, Gane, Todd, Hillier, Michael C, Kessler, Horst, Baur, Matthias, Mathä, Barbara, Erickson, John W, Bhat, T. Nagarajan, Munshi, Sanjeev, Gulnik, Sergei V, Topol, Igor A

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Diastereodifferentiation in intramolecular cyclopropanations of chiral secondary allylic diazoacetates von Martin, Stephen F, Hillier, Michael C

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ChemInform Abstract: Synthesis of Hydantoins and Dihydrouracils via Thermally-Promoted Cyclization of Ureidoacetamides von Hillier, Michael C., Gong, Hai-Hua, Clyne, Dean S., Babcock, Martin J.

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Cyclopropane-Derived Peptidomimetics. Design, Synthesis, and Evaluation of Novel Ras Farnesyltransferase Inhibitors von Hillier, Michael C., Davidson, James P., Martin, Stephen F.

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Selective displacement of aryl fluorides with hydroquinone: synthesis of 4-phenoxyphenols von Marcune, Benjamin F., Hillier, Michael C., Marcoux, Jean-François, Humphrey, Guy R.

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Stereoselective Formation of Carbon−Carbon Bonds via S N 2-Displacement:  Synthesis of Substituted Cycloalkyl[ b ]indoles von Hillier, Michael C., Marcoux, Jean-François, Zhao, Dalian, Grabowski, Edward J. J., McKeown, Arlene E., Tillyer, Richard D.

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Applications of Intramolecular Cyclopropanations of Chiral Secondary Allylic Diazoacetates von Martin, Stephen F., Hillier, Michael C.

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Cyclopropane-Derived Peptidomimetics. Design, Synthesis, and Evaluation of Novel Ras Farnesyltransferase Inhibitors von HILLIER, Michael C., DAVIDSON, James P., MARTIN, Stephen F.

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ETHYL 5-CHLORO-3-PHENYLINDOLE-2-CARBOXYLATE

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