Small-Molecule Inhibitors and Probes for Ubiquitin- and Ubiquitin-Like-Specific Proteases von Borodovsky, Anna, Ovaa, Huib, Meester, Wim J.N, Venanzi, Emily S, Bogyo, Matthew S, Hekking, Brian G, Ploegh, Hidde L, Kessler, Benedikt M, Overkleeft, Herman S

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Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic β-subunits von Kessler, Benedikt M, Tortorella, Domenico, Altun, Mikael, Kisselev, Alexei F, Fiebiger, Edda, Hekking, Brian G, Ploegh, Hidde L, Overkleeft, Herman S

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Solid phase synthesis of peptide vinyl sulfone and peptide epoxyketone proteasome inhibitors von Overkleeft, Herman S, Bos, Pepijn R, Hekking, Brian G, Gordon, Eva J, Ploegh, Hidde L, Kessler, Benedikt M

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Development of Potent Mcl‑1 Inhibitors: Structural Investigations on Macrocycles Originating from a DNA-Encoded Chemical Library Screen von Hekking, Koen F. W., Maroto, Sergio, van Kekem, Kees, Haasjes, Frank S., Slootweg, Jack C., Oude Alink, Patrick G. B., Dirks, Ron, Sardana, Malvika, Bolster, Marjon G., Kuijpers, Brian, Smith, Dennis, Doodeman, Robin, Scheepstra, Marcel, Zech, Birgit, Mulvihill, Mark, Renzetti, Louis M., Babiss, Lee, Centrella, Paolo A., Clark, Matthew A., Cuozzo, John W., Guié, Marie-Aude, Sigel, Eric, Habeshian, Sevan, Hupp, Christopher D., Liu, Julie, Thomson, Heather A., Zhang, Ying, Keefe, Anthony D., Müller, Gerhard, Gremmen, Stijn

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