Enantiopure bicyclic piperidinones: stereoselectivity in lactam enolate alkylations von Brewster, Andrew G, Broady, Simon, Davies, Catherine E, Heightman, Thomas D, Hermitage, Stephen A, Hughes, Mark, Moloney, Mark G, Woods, Gordon

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Synthesis of Galactose- and N-Acetylglucosamine-Derived Tetrazoles and their evaluation as β-glycosidase inhibitors von Heightman, Thomas D., Ermert, Philipp, Klein, Daniela, Vasella, Andrea

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Convenient preparations of racemic and enantiopure methyl 6-oxopipecolate von Davies, Catherine E., Heightman, Thomas D., Hermitage, Stephen A., Moloney, Mark G.

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Diastereoselectivity in the alkylations of bicyclic piperidinones von Mills (née Davis), Catherine E., Heightman, Thomas D., Hermitage, Stephen A., Moloney, Mark G., Woods, Gordon A.

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Tetrahydrobenzazepines as Histamine H3 Receptor Ligands von HEIGHTMAN THOMAS D, WILSON DAVID M

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Substituted piperazines (1,4) diaszepines, and 2,5-diazabicyclo (2.2.1) heptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists von ANCLIFF RANCHAEL,ELDRED COLIN D.,FOGDEN YVONNE C.,HANCOCK ASHLEY P.,HEIGHTMAN THOMAS D.,HOBBS HEATHER,HODGSON SIMON T.,LINDON MATTHEW J.,WILSON DAVIDM

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Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists von ANCLIFF RANCHAEL A.,ELDRED COLIN D.,FOGDEN YVONNEC.,HANCOCK ASHLEY P.,HEIGHTMAN THOMAS D.,HOBBS HEATHER,HODGSON SIMON T.,LINDON MATTHEW J.,WILSON DAVID M

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Isoquinoline and quinazoline derivatives having a combined 5HT1A, 5HT1B, and 5HT1D receptor activity von HEIGHTMAN THOMAS D, GASTER LARAMIE M, PILLEUX JEAN-PIERRE

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Benzazepine derivatives for the treatment of neurological and psychiatric disorders von HEIGHTMAN THOMAS D, BAMFORD MARK J, WILSON DAVID M, WITHERINGTON JASON

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Phenyl substituted triazoles and their use as selective inhibitors of AKL5 kinase von HARLING, JOHN, D, ASTER, LARAMIE, M, PAYNE, ANDREW, H, HEER, JAG, P, HEIGHTMAN, THOMAS, D

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Aryloxyalkylamine derivatives as h3 receptor ligands von HEIGHTMAN THOMAS D, BRUTON GORDON, ORLEK BARRY S, BEST DESMOND J

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Enantiopure Bicyclic Piperidinones: Stereoselectivity in Lactam Enolate Alkylations von Brewster, Andrew G., Broady, Simon, Davies, Catherine E., Heightman, Thomas D., Hermitage, Stephen A., Hughes, Mark, Moloney, Mark G., Woods, Gordon

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Substituted piperazines (1,4) diaszepines, and 2,5-diazabicyclo (2.2.1) heptanes as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists von ELDRED, COLIN, D, LINDON, MATTHEW, J, FOGDEN, YVONNE, C, WILSON, DAVID, M, RACHAEL ANCLIFF, HEATHER HOBBS, HODGSON, SIMON, T, HANCOCK, ASHLEY, P, HEIGHTMAN, THOMAS, D

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Compounds von HEIGHTMAN THOMAS D, HODGSON SIMON T, LINDON MATTHEW J, FOGDEN YVONNE C, ELDRED COLIN D, HANCOCK ASHLEY P, HOBBS HEATHER, WILSON DAVID M, ANCLIFF RANCHAEL A

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Patterns of myocardial injury in recovered troponin-positive COVID-19 patients assessed by cardiovascular magnetic resonance von Kotecha, Tushar, Knight, Daniel S, Razvi, Yousuf, Kumar, Kartik, Vimalesvaran, Kavitha, Thornton, George, Patel, Rishi, Chacko, Liza, Brown, James T, Coyle, Clare, Leith, Donald, Shetye, Abhishek, Ariff, Ben, Bell, Robert, Captur, Gabriella, Coleman, Meg, Goldring, James, Gopalan, Deepa, Heightman, Melissa, Hillman, Toby, Howard, Luke, Jacobs, Michael, Jeetley, Paramjit S, Kanagaratnam, Prapa, Kon, Onn Min, Lamb, Lucy E, Manisty, Charlotte H, Mathurdas, Palmira, Mayet, Jamil, Negus, Rupert, Patel, Niket, Pierce, Iain, Russell, Georgina, Wolff, Anthony, Xue, Hui, Kellman, Peter, Moon, James C, Treibel, Thomas A, Cole, Graham D, Fontana, Marianna

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Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2‑Related Factor 2 (KEAP1:NRF2) Protein–Protein Interaction with High Cell Potency Identi... von Davies, Thomas G, Wixted, William E, Coyle, Joseph E, Griffiths-Jones, Charlotte, Hearn, Keisha, McMenamin, Rachel, Norton, David, Rich, Sharna J, Richardson, Caroline, Saxty, Gordon, Willems, Henriëtte M. G, Woolford, Alison J.-A, Cottom, Joshua E, Kou, Jen-Pyng, Yonchuk, John G, Feldser, Heidi G, Sanchez, Yolanda, Foley, Joseph P, Bolognese, Brian J, Logan, Gregory, Podolin, Patricia L, Yan, Hongxing, Callahan, James F, Heightman, Tom D, Kerns, Jeffrey K

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Structure–Activity and Structure–Conformation Relationships of Aryl Propionic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1/Nuclear Factor Erythroid 2‑Related Factor 2... von Heightman, Tom D, Callahan, James F, Chiarparin, Elisabetta, Coyle, Joseph E, Griffiths-Jones, Charlotte, Lakdawala, Ami S, McMenamin, Rachel, Mortenson, Paul N, Norton, David, Peakman, Torren M, Rich, Sharna J, Richardson, Caroline, Rumsey, William L, Sanchez, Yolanda, Saxty, Gordon, Willems, Henriëtte M. G, Wolfe, Lawrence, Woolford, Alison J.-A, Wu, Zining, Yan, Hongxing, Kerns, Jeffrey K, Davies, Thomas G

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Fragment-Guided Discovery of Pyrazole Carboxylic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2 Related Factor 2 (KEAP1:NRF2) Protein−Protei... von Norton, David, Bonnette, William G, Callahan, James F, Carr, Maria G, Griffiths-Jones, Charlotte M, Heightman, Tom D, Kerns, Jeffrey K, Nie, Hong, Rich, Sharna J, Richardson, Caroline, Rumsey, William, Sanchez, Yolanda, Verdonk, Marcel L, Willems, Henriëtte M. G, Wixted, William E, Woolford, Alison J.-A, Wu, Zining, Davies, Thomas G

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Cardiopulmonary Fitness, Skeletal Muscle Oxidative Capacity And Microvascular Function In People Living With Long Covid Compared With Healthy Controls: 2494 von Jamieson, Alexandra, Astin, Ronan, Bell, Robert, Hamer, Mark, Howes, Lee Hamill, Heightman, Melissa, Hillman, Toby, Montgomery, Hugh, Al Saikhan, Lamia, Scully, Marie Ann, Treibel, Thomas, Hughes, Alun D., Jones, Siana

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Mechanisms underlying exercise intolerance in long COVID: An accumulation of multisystem dysfunction von Jamieson, Alexandra, Al Saikhan, Lamia, Alghamdi, Lamis, Hamill Howes, Lee, Purcell, Helen, Hillman, Toby, Heightman, Melissa, Treibel, Thomas, Orini, Michele, Bell, Robert, Scully, Marie, Hamer, Mark, Chaturvedi, Nishi, Montgomery, Hugh, Hughes, Alun D., Astin, Ronan, Jones, Siana

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