Identification and characterization of the new generation soluble guanylate cyclase stimulator BAY‐747 designed for the treatment of resistant hypertension von Wunder, Frank, Stasch, Johannes‐Peter, Knorr, Andreas, Mondritzki, Thomas, Brockschnieder, Damian, Becker‐Pelster, Eva‐Maria, Sandner, Peter, Tinel, Hanna, Redlich, Gorden, Hartung, Ingo V., Vakalopoulos, Alexandros, Follmann, Markus

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Discovery of Molidustat (BAY 85‐3934): A Small‐Molecule Oral HIF‐Prolyl Hydroxylase (HIF‐PH) Inhibitor for the Treatment of Renal Anemia von Beck, Hartmut, Jeske, Mario, Thede, Kai, Stoll, Friederike, Flamme, Ingo, Akbaba, Metin, Ergüden, Jens‐Kerim, Karig, Gunter, Keldenich, Jörg, Oehme, Felix, Militzer, Hans‐Christian, Hartung, Ingo V., Thuss, Uwe

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A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition von Falkenstern, Lilia, Georgi, Victoria, Bunse, Stefanie, Badock, Volker, Husemann, Manfred, Roehn, Ulrike, Stellfeld, Timo, Fitzgerald, Mark, Ferrara, Steven, Stöckigt, Detlef, Stresemann, Carlo, Hartung, Ingo V., Fernández-Montalván, Amaury

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Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2 von Eggert, Erik, Hillig, Roman C, Koehr, Silke, Stöckigt, Detlef, Weiske, Jörg, Barak, Naomi, Mowat, Jeffrey, Brumby, Thomas, Christ, Clara D, ter Laak, Antonius, Lang, Tina, Fernandez-Montalvan, Amaury E, Badock, Volker, Weinmann, Hilmar, Hartung, Ingo V, Barsyte-Lovejoy, Dalia, Szewczyk, Magdalena, Kennedy, Steven, Li, Fengling, Vedadi, Masoud, Brown, Peter J, Santhakumar, Vijayaratnam, Arrowsmith, Cheryl H, Stellfeld, Timo, Stresemann, Carlo

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Electronic and Steric Control of Regioselectivities in Rh(I)-Catalyzed (5 + 2) Cycloadditions: Experiment and Theory von Liu, Peng, Sirois, Lauren E, Cheong, Paul Ha-Yeon, Yu, Zhi-Xiang, Hartung, Ingo V, Rieck, Heiko, Wender, Paul A, Houk, K. N

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No shortcuts to SARS-CoV-2 antivirals von Edwards, Aled, Hartung, Ingo V.

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Targeting the aryl hydrocarbon receptor (AhR) with BAY 2416964: a selective small molecule inhibitor for cancer immunotherapy von Kober, Christina, Roewe, Julian, Schmees, Norbert, Roese, Lars, Roehn, Ulrike, Bader, Benjamin, Stoeckigt, Detlef, Prinz, Florian, Gorjánácz, Mátyás, Roider, Helge Gottfried, Olesch, Catherine, Leder, Gabriele, Irlbacher, Horst, Lesche, Ralf, Lefranc, Julien, Oezcan-Wahlbrink, Mine, Batra, Ankita Sati, Elmadany, Nirmeen, Carretero, Rafael, Sahm, Katharina, Oezen, Iris, Cichon, Frederik, Baumann, Daniel, Sadik, Ahmed, Opitz, Christiane A, Weinmann, Hilmar, Hartung, Ingo V, Kreft, Bertolt, Offringa, Rienk, Platten, Michael, Gutcher, Ilona

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8-Oxabicyclo[3.2.1]oct-6-en-3-ones: Application to the Asymmetric Synthesis of Polyoxygenated Building Blocks von Hartung, Ingo V., Hoffmann, H. Martin R.

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Expanding Chemical Probe Space: Quality Criteria for Covalent and Degrader Probes von Hartung, Ingo V., Rudolph, Joachim, Mader, Mary M., Mulder, Monique P. C., Workman, Paul

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Rules were made to be broken von Hartung, Ingo V., Huck, Bayard R., Crespo, Alejandro

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Which Small Molecule? Selecting Chemical Probes for Use in Cancer Research and Target Validation von Mader, Mary M, Rudolph, Joachim, Hartung, Ingo V, Uehling, David, Workman, Paul, Zuercher, William

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Discovery of BAY-405: An Azaindole-Based MAP4K1 Inhibitor for the Enhancement of T‑Cell Immunity against Cancer von Mowat, Jeffrey, Carretero, Rafael, Leder, Gabriele, Aiguabella Font, Nuria, Neuhaus, Roland, Berndt, Sandra, Günther, Judith, Friberg, Anders, Schäfer, Martina, Briem, Hans, Raschke, Marian, Miyatake Ondozabal, Hideki, Buchmann, Bernd, Boemer, Ulf, Kreft, Bertolt, Hartung, Ingo V., Offringa, Rienk

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New Generation of sGC Stimulators: Discovery of Imidazo[1,2‑a]pyridine Carboxamide BAY 1165747 (BAY-747), a Long-Acting Soluble Guanylate Cyclase Stimulator for the Treatment of Re... von Vakalopoulos, Alexandros, Wunder, Frank, Hartung, Ingo V., Redlich, Gorden, Jautelat, Rolf, Buchgraber, Philipp, Hassfeld, Jorma, Gromov, Alexey V., Lindner, Niels, Bierer, Donald, Gries, Jörg, Kroh, Walter, Paulsen, Holger, Mittendorf, Joachim, Lang, Dieter, Becker-Pelster, Eva, Brockschnieder, Damian, Geiss, Volker, Li, Volkhart, Straub, Alexander, Knorr, Andreas, Mondritzki, Thomas, Trübel, Hubert, Raschke, Marian, Schaefer, Martina, Thomas, Dirk, Sandner, Peter, Stasch, Johannes-Peter, Follmann, Markus

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Systematic Potency and Property Assessment of VHL Ligands and Implications on PROTAC Design von Krieger, Johannes, Sorrell, Fiona J., Wegener, Ansgar A., Leuthner, Birgitta, Machrouhi‐Porcher, Fouzia, Hecht, Martin, Leibrock, Eva M., Müller, Juliane E., Eisert, Jonathan, Hartung, Ingo V., Schlesiger, Sarah

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Discovery and Characterization of BAY-184: A New Potent and Selective Acylsulfonamide-Benzofuran In Vivo-Active KAT6AB Inhibitor von ter Laak, Antonius, Hillig, Roman C., Ferrara, Steven J., Korr, Daniel, Barak, Naomi, Lienau, Philip, Herbert, Simon, Fernández-Montalván, Amaury Ernesto, Neuhaus, Roland, Gorjánácz, Mátyás, Puetter, Vera, Badock, Volker, Bone, Wilhelm, Strathdee, Craig, Siegel, Franziska, Schatz, Christoph, Nowak-Reppel, Katrin, Doehr, Olaf, Gradl, Stefan, Hartung, Ingo V., Meyerson, Matthew, Bouché, Léa

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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation von Quancard, Jean, Vulpetti, Anna, Bach, Anders, Cox, Brian, Guéret, Stéphanie M., Hartung, Ingo V., Koolman, Hannes F., Laufer, Stefan, Messinger, Josef, Sbardella, Gianluca, Craft, Russell

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The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes von Quancard, Jean, Cox, Brian, Finsinger, Dirk, Guéret, Stéphanie M., Hartung, Ingo V., Koolman, Hannes F., Messinger, Josef, Sbardella, Gianluca, Laufer, Stefan

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The 17th EFMC Short Course on Medicinal Chemistry on Small Molecule Protein Degraders von Ciulli, Alessio, O'Connor, Suzanne, Chung, Chun‐Wa, Hartung, Ingo V., Testa, Andrea, Daniels, Danette L., Heitman, Laura H.

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Workflow for E3 Ligase Ligand Validation for PROTAC Development von Miletić, Nebojša, Weckesser, Janik, Mosler, Thorsten, Rathore, Rajeshwari, Hoffmann, Marina E, Gehrtz, Paul, Schlesiger, Sarah, Hartung, Ingo V, Berner, Nicola, Wilhelm, Stephanie, Müller, Juliane, Adhikari, Bikash, Němec, Václav, Sivashanmugam, Saran Aswathaman, Elson, Lewis, Holzmann, Hanna, Schwalm, Martin P, Hoffmann, Lasse, Abdul Azeez, Kamal Rayees, Müller, Susanne, Kuster, Bernhard, Wolf, Elmar, Đikić, Ivan, Knapp, Stefan

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Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains von Bouché, Léa, Christ, Clara D, Siegel, Stephan, Fernández-Montalván, Amaury E, Holton, Simon J, Fedorov, Oleg, ter Laak, Antonius, Sugawara, Tatsuo, Stöckigt, Detlef, Tallant, Cynthia, Bennett, James, Monteiro, Octovia, Díaz-Sáez, Laura, Siejka, Paulina, Meier, Julia, Pütter, Vera, Weiske, Jörg, Müller, Susanne, Huber, Kilian V. M, Hartung, Ingo V, Haendler, Bernard

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