Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279 von Leit, Silvana, Greenwood, Jeremy, Carriero, Samantha, Mondal, Sayan, Abel, Robert, Ashwell, Mark, Blanchette, Heather, Boyles, Nicholas A., Cartwright, Mark, Collis, Alan, Feng, Shulu, Ghanakota, Phani, Harriman, Geraldine C., Hosagrahara, Vinayak, Kaila, Neelu, Kapeller, Rosanna, Rafi, Salma B., Romero, Donna L., Tarantino, Paul M., Timaniya, Jignesh, Toms, Angela V., Wester, Ronald T., Westlin, William, Srivastava, Bhaskar, Miao, Wenyan, Tummino, Peter, McElwee, Joshua J., Edmondson, Scott D., Masse, Craig E.

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Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis von Leit, Silvana, Greenwood, Jeremy R., Mondal, Sayan, Carriero, Samantha, Dahlgren, Markus, Harriman, Geraldine C., Kennedy-Smith, Joshua J., Kapeller, Rosana, Lawson, Jon P., Romero, Donna L., Toms, Angela V., Shelley, Mee, Wester, Ronald T., Westlin, William, McElwee, Joshua J., Miao, Wenyan, Edmondson, Scott D., Masse, Craig E.

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Design, Synthesis, and Evaluation of Naphthalene-Sulfonamide Antagonists of Human CCR8 von Jenkins, Tracy J, Guan, Bing, Dai, Mingshi, Li, Gang, Lightburn, Thomas E, Huang, Shan, Freeze, B. Scott, Burdi, Douglas F, Jacutin-Porte, Swanee, Bennett, Robert, Chen, Weirong, Minor, Charles, Ghosh, Shomir, Blackburn, Christopher, Gigstad, Kenneth M, Jones, Matthew, Kolbeck, Roland, Yin, Wei, Smith, Sean, Cardillo, Daniel, Ocain, Timothy D, Harriman, Geraldine C

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Selective cell adhesion inhibitors: Barbituric acid based α4β7—MAdCAM inhibitors von Harriman, Geraldine C., Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R., Briskin, Michael J.

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Selective cell adhesion inhibitors: Barbituric acid based alpha 4 beta 7 - MAdCAM inhibitors von Harriman, Geraldine C, Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R, Briskin, Michael J

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The Chemistry of the Taxane Diterpene:  Stereoselective Reductions of Taxanes von Georg, Gunda I, Harriman, Geraldine C. B, Datta, Apurba, Ali, Syed, Cheruvallath, Zacharia, Dutta, Dinah, Vander Velde, David G, Himes, Richard H

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A Facile One-Flask Conversion of Aldehydes and Ketones to N-Sulfonyl Imines von Georg, Gunda I, Harriman, Geraldine C. B, Peterson, Scott A

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Synthesis, Conformational Analysis, and Biological Evaluation of Heteroaromatic Taxanes von Georg, Gunda I, Harriman, Geraldine C. B, Hepperle, Michael, Clowers, Jamie S, Vander Velde, David G, Himes, Richard H

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Synthesis of a Photoaffinity Taxol Analog and Its Use in Labeling Tubulin von Dasgupta, Debjani, Park, Haeil, Harriman, Geraldine C. B, Georg, Gunda I, Himes, Richard H

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Adenosine deaminase inhibitors. Synthesis and biological evaluation of 4-amino-1-[2(S)-hydroxy-3(R)-nonyl]-1H-imidazo[4,5-c]pyridine [3-deaza-(+)-EHNA] and certain C1' derivatives von Harriman, Geraldine C. B, Abushanab, Elie, Stoeckler, Johanna D

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Adenosine deaminase inhibitors. Synthesis and biological evaluation of C1' and nor-C1' derivatives of (+)-erythro-9-[2(S)-hydroxy-3(R)-nonyl]adenine von Harriman, Geraldine C. B, Poirot, Anne F, Abushanab, Elie, Midgett, Rose Marie, Stoeckler, Johanna D

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PYRAZOLE ACC INHIBITORS AND USES THEREOF von HARRIMAN, GERALDINE C, GREENWOOD, JEREMY ROBERT, LEIT DE MORADEI, SILVANA MARCEL, GHOSH, SHOMIR

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TRIAZOLE ACC INHIBITORS AND USES THEREOF von HARRIMAN, GERALDINE C, GREENWOOD, JEREMY ROBERT, LEIT DE MORADEI, SILVANA MARCEL, GHOSH, SHOMIR

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ESTER ACC INHIBITORS AND USES THEREOF von HARRIMAN, GERALDINE C, GREENWOOD, JEREMY ROBERT, LEIT DE MORADEI, SILVANA MARCEL, GHOSH, SHOMIR

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Solid forms for a thienopyrimidinedione ACC inhibitor and methods for production thereof von Lawson, Jon P, Yang, Xiaowei, Harriman, Geraldine C

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PYRAZOLE ACC INHIBITORS AND USES THEREOF von HARRIMAN, Geraldine C, LEIT DE MORADEI, Silvana Marcel, GHOSH, Shomir, GREENWOOD, Jeremy Robert

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TRIAZOLE ACC INHIBITORS AND USES THEREOF von HARRIMAN, Geraldine C, LEIT DE MORADEI, Silvana Marcel, GHOSH, Shomir, GREENWOOD, Jeremy Robert

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ACC INHIBITORS AND USES THEREOF von Ghosh Shomir, Harriman Geraldine C

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ACC INHIBITORS AND USES THEREOF von HARRIMAN, Geraldine C, GHOSH, Shomir

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ACC INHIBITORS AND USES THEREOF von HARRIMAN, GERALDINE C, HARWOOD, JAMES, GREENWOOD, JEREMY ROBERT, MASSE, CRAIG E, BHAT, SATHESH

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