GPCRdb: an information system for G protein-coupled receptors von Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S, Vroling, Bas, Bojarski, Andrzej J, Vriend, Gert, Gloriam, David E

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Structural insights into the lipid and ligand regulation of serotonin receptors von Xu, Peiyu, Huang, Sijie, Zhang, Huibing, Mao, Chunyou, Zhou, X. Edward, Cheng, Xi, Simon, Icaro A., Shen, Dan-Dan, Yen, Hsin-Yung, Robinson, Carol V., Harpsøe, Kasper, Svensson, Bo, Guo, Jia, Jiang, Hualiang, Gloriam, David E., Melcher, Karsten, Jiang, Yi, Zhang, Yan, Xu, H. Eric

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GPCRdb in 2018: adding GPCR structure models and ligands von Pándy-Szekeres, Gáspár, Munk, Christian, Tsonkov, Tsonko M, Mordalski, Stefan, Harpsøe, Kasper, Hauser, Alexander S, Bojarski, Andrzej J, Gloriam, David E

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GPCRs steer Gi and Gs selectivity via TM5-TM6 switches as revealed by structures of serotonin receptors von Huang, Sijie, Xu, Peiyu, Shen, Dan-Dan, Simon, Icaro A., Mao, Chunyou, Tan, Yangxia, Zhang, Huibing, Harpsøe, Kasper, Li, Huadong, Zhang, Yumu, You, Chongzhao, Yu, Xuekui, Jiang, Yi, Zhang, Yan, Gloriam, David E., Xu, H. Eric

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Molecular insights into ligand recognition and G protein coupling of the neuromodulatory orphan receptor GPR139 von Zhou, Yali, Daver, Henrik, Trapkov, Boris, Wu, Lijie, Wu, Meng, Harpsøe, Kasper, Gentry, Patrick R., Liu, Kaiwen, Larionova, Marina, Liu, Junlin, Chen, Na, Bräuner-Osborne, Hans, Gloriam, David E., Hua, Tian, Liu, Zhi-Jie

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Total synthesis and structure–activity relationship studies of a series of selective G protein inhibitors von Xiong, Xiao-Feng, Zhang, Hang, Underwood, Christina R., Harpsøe, Kasper, Gardella, Thomas J., Wöldike, Mie F., Mannstadt, Michael, Gloriam, David E., Bräuner-Osborne, Hans, Strømgaard, Kristian

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GPCRdb: an information system for G protein-coupled receptors von Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S, Vroling, Bas, Bojarski, Andrzej J, Vriend, Gert, Gloriam, David E

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A novel red fluorescence dopamine biosensor selectively detects dopamine in the presence of norepinephrine in vitro von Nakamoto, Chihiro, Goto, Yuhei, Tomizawa, Yoko, Fukata, Yuko, Fukata, Masaki, Harpsoe, Kasper, Gloriam, David E., Aoki, Kazuhiro, Takeuchi, Tomonori

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Ligand selectivity hotspots in serotonin GPCRs von Simon, Icaro A, Bjørn-Yoshimoto, Walden E, Harpsøe, Kasper, Iliadis, Stylianos, Svensson, Bo, Jensen, Anders A, Gloriam, David E

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A community Biased Signaling Atlas von Caroli, Jimmy, Mamyrbekov, Alibek, Harpsøe, Kasper, Gardizi, Sahar, Dörries, Linda, Ghosh, Eshan, Hauser, Alexander S., Kooistra, Albert J., Gloriam, David E.

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Discovery of a new class of orthosteric antagonists with nanomolar potency at extrasynaptic GABAA receptors von Falk-Petersen, Christina Birkedahl, Tsonkov, Tsonko M., Nielsen, Malene Sofie, Harpsøe, Kasper, Bundgaard, Christoffer, Frølund, Bente, Kristiansen, Uffe, Gloriam, David E., Wellendorph, Petrine

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Structure–activity relationship and conformational studies of the natural product cyclic depsipeptides YM-254890 and FR900359 von Zhang, Hang, Nielsen, Alexander L., Boesgaard, Michael W., Harpsøe, Kasper, Daly, Norelle L., Xiong, Xiao-Feng, Underwood, Christina R., Haugaard-Kedström, Linda M., Bräuner-Osborne, Hans, Gloriam, David E., Strømgaard, Kristian

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GPCRdb in 2018: adding GPCR structure models and ligands von Pándy-Szekeres, Gáspár, Munk, Christian, Tsonkov, Tsonko M, Mordalski, Stefan, Harpsøe, Kasper, Hauser, Alexander S, Bojarski, Andrzej J, Gloriam, David E

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Integrating structural and mutagenesis data to elucidate GPCR ligand binding von Munk, Christian, Harpsøe, Kasper, Hauser, Alexander S, Isberg, Vignir, Gloriam, David E

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Development of a human vasopressin V1a-receptor antagonist from an evolutionary-related insect neuropeptide von Di Giglio, Maria Giulia, Muttenthaler, Markus, Harpsøe, Kasper, Liutkeviciute, Zita, Keov, Peter, Eder, Thomas, Rattei, Thomas, Arrowsmith, Sarah, Wray, Susan, Marek, Ales, Elbert, Tomas, Alewood, Paul F., Gloriam, David E., Gruber, Christian W.

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Unraveling the high- and low-sensitivity agonist responses of nicotinic acetylcholine receptors von Harpsøe, Kasper, Ahring, Philip K, Christensen, Jeppe K, Jensen, Marianne L, Peters, Dan, Balle, Thomas

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Selective Negative Allosteric Modulation Of Metabotropic Glutamate Receptors – A Structural Perspective of Ligands and Mutants von Harpsøe, Kasper, Isberg, Vignir, Tehan, Benjamin G., Weiss, Dahlia, Arsova, Angela, Marshall, Fiona H., Bräuner-Osborne, Hans, Gloriam, David E.

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Molecular Determinants Underlying Delta Selective Compound 2 Activity at delta-Containing GABA(A) Receptors von Falk-Petersen, Christina B., Rostrup, Frederik, Loffler, Rebekka, Buchleithner, Stine, Harpsoe, Kasper, Gloriam, David E., Frolund, Bente, Wellendorph, Petrine

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Pharmacological characterization of novel small molecule agonists and antagonists for the orphan receptor GPR139 von Pallareti, Lisa, Rath, Tine F., Trapkov, Boris, Tsonkov, Tsonko, Nielsen, Anders Thorup, Harpsøe, Kasper, Gentry, Patrick R., Bräuner-Osborne, Hans, Gloriam, David E., Foster, Simon R.

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Comprehensive Peptide Cyclization Examination Yields Optimized APP Scaffolds with Improved Affinity toward Mint2 von Bartling, Christian R. O., Alexopoulou, Flora, Kuschert, Sarah, Chin, Yanni K.-Y., Jia, Xinying, Sereikaite, Vita, Özcelik, Dennis, Jensen, Thomas M., Jain, Palash, Nygaard, Mads M., Harpsøe, Kasper, Gloriam, David E., Mobli, Mehdi, Strømgaard, Kristian

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