Alleviation of arthritis through prevention of neutrophil extracellular traps by an orally available inhibitor of protein arginine deiminase 4 von Gajendran, Chandru, Fukui, Shoichi, Sadhu, Naveen M., Zainuddin, Mohammed, Rajagopal, Sridharan, Gosu, Ramachandraiah, Gutch, Sarah, Fukui, Saeko, Sheehy, Casey E., Chu, Long, Vishwakarma, Santosh, Jeyaraj, D. A., Hallur, Gurulingappa, Wagner, Denisa D., Sivanandhan, Dhanalakshmi

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Design, Synthesis, and Evaluation of Novel Boronic-Chalcone Derivatives as Antitumor Agents von Kumar, Srinivas K, Hager, Erin, Pettit, Catherine, Gurulingappa, Hallur, Davidson, Nancy E, Khan, Saeed R

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Palladium-Catalyzed Direct α‑Arylation of Indane-1,3-dione to 2‑Substituted Indene-1,3-diones von Tamizharasan, Natarajan, Hallur, Gurulingappa, Suresh, Palaniswamy

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Silver-Promoted Rapid Synthesis of 3‑Arylindan-1-ones: Microwave-Assisted Reductive Coupling of N‑Tosylhydrazone and Boronic Acids von Tamizharasan, Natarajan, Santhoshkumar, Pandeeswaran, Devarajan, Nainamalai, Hallur, Mahanandeesha S., Hallur, Gurulingappa, Suresh, Palaniswamy

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Development of two novel benzoylphenylurea sulfur analogues and evidence that the microtubule-associated protein tau is predictive of their activity in pancreatic cancer von Jimeno, Antonio, Hallur, Gurulingappa, Chan, Audrey, Zhang, Xiangfeng, Cusatis, George, Chan, Fonda, Shah, Preeti, Chen, Rongbing, Hamel, Ernest, Garrett-Mayer, Elizabeth, Khan, Saeed, Hidalgo, Manuel

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Three New Tetranortriterpenoids from Neem Seed Oil von Hallur, Gurulingappa, Sivramakrishnan, Apoorba, Bhat, Sujata V

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Validation of an LC-ESI–MS/MS method for the determination of apalutamide, a novel non-steroidal anti-androgen in mice plasma and its application to a pharmacokinetic study in mice... von Hallur, Gurulingappa, Purra, Buchi Reddy, Sulochana, Suresh P, Saini, Neeraj Kumar, Daram, Prasanthi, Zainuddin, Mohd, Mullangi, Ramesh

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LC-ESI–MS/MS determination of defactinib, a novel FAK inhibitor in mice plasma and its application to a pharmacokinetic study in mice von Hallur, Gurulingappa, Tamizharasan, Natarajan, Sulochana, Suresh P., Saini, Neeraj Kumar, Zainuddin, Mohd, Mullangi, Ramesh

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In vitro and In vivo Clinical Pharmacology of Dimethyl Benzoylphenylurea, a Novel Oral Tubulin-Interactive Agent von Rudek, Michelle A, Zhao, Ming, Smith, Nicola F, Robey, Robert W, He, Ping, Hallur, Gurulingappa, Khan, Saeed, Hidalgo, Manuel, Jimeno, Antonio, Colevas, A Dimitrios, Messersmith, Wells A, Wolff, Antonio C, Baker, Sharyn D

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Discovery and optimization of novel phenyldiazepine and pyridodiazepine based Aurora kinase inhibitors von Tamizharasan, Natarajan, Gajendran, Chandru, Kristam, Rajendra, Sulochana, Suresh P., Sivanandhan, Dhanalakshmi, Mullangi, Ramesh, Mathivathanan, Logesh, Hallur, Gurulingappa, Suresh, Palaniswamy

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Abstract 3332: LNG-451 is a potent, CNS-penetrant, wild-type EGFR sparing inhibitor of EGFR exon 20 insertion mutations von Murray, Brion W., Pandey, Anjali, Roth, Bruce, Saxton, Tracy, Estes, Daniel J., Agrawal, Himanshu, Vishwakarma, Santosh, Hallur, Gurulingappa, Ahmad, Ishtiyaque, Trivedi, Ravi, Jenkins, Helen, Pearson, Paul G.

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Abstract 3261: LNG-451, a potent inhibitor of EGFR exon 20 insertion mutations with high CNS exposure von Pearson, Paul G., Pandey, Anjali, Roth, Bruce, Saxton, Tracy, Estes, Daniel J., Trivedi, Ravi, Agrawal, Himanshu, Hallur, Gurulingappa, Ahmad, Ishtiyaque, Jenkins, Helen, Murray, Brion W.

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Validation of an LC–MS/MS Method for Simultaneous Detection of Five Selective KCNQ Channel Openers: ICA-27243, ML-213, PF-05020182, SF-0034 and Flupirtine in Mice Plasma and its Ap... von Todmal, Umesh, Sulochana, Suresh P., Zainuddin, Mohd, Bhamidipati, Ravi Kanth, Samanta, Swapan Kumar, Hallur, Gurulingappa, Rajagopal, Sridharan, Rajagopal, Sriram, Mullangi, Ramesh

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Abstract 2646: Novel, isoform selective PAD4 inhibitors for the treatment of cancer von Sivanandhan, Dhanalakshmi, Rajagopal, Sridharan, G, Chandru, Zainuddin, Mohd, Sadhu, Naveen, Gosu, Ramachandraiah, Rastelli, Luca, Siddiqui, Amir, Singh, Sharad, G, Rudresh, Mullurwar, Sadanand, Kandan, Saravanan, Vishwakarma, Santosh, Hallur, Gurulingappa, Trivedi, Ravi, A, Jeyaraj D

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Validated LC–MS-MS Method for Determination of SF0034 in Mice Plasma: Application to a Pharmacokinetic Study in Mice von Todmal, Umesh, Suresh, P. S., Zainuddin, Mohd, Kanth Bhamidipati, Ravi, Samanta, Swapan Kumar, Hallur, Gurulingappa, Rajagopal, Sridharan, Rajagopal, Sriram, Mullangi, Ramesh

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Novel Microtubule-Interacting Phenoxy Pyridine and Phenyl Sulfanyl Pyridine Analogues for Cancer Therapy von Anchoori, Ravi Kumar, Kortenhorst, Madeleine Susanne Quirine, Hidalgo, Manuel, Sarkar, Taradas, Hallur, Gurulingappa, Bai, Ruoli, Diest, Paul J. Van, Hamel, Ernest, Khan, Saeed R

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Targeting Vascular and Avascular Compartments of Tumors with C. novyi-NT and Anti-microtubule Agents von Dang, L.H., Bettegowda, C., Agrawal, N., Cheong, I., Huso, D., Frost, P., Loganzo, F., Greenberger, L., Barkoczy, J., Pettit, G.R., Smith, A.B., Gurulingappa, H., Khan, S., Parmigiani, G., Kinzler, K.W., Zhou, S., Vogelstein, B.

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Benzoylphenylurea Sulfur Analogues with Potent Antitumor Activity von Hallur, Gurulingappa, Jimeno, Antonio, Dalrymple, Susan, Zhu, Tao, Jung, M. Katherine, Hidalgo, Manuel, Isaacs, John T, Sukumar, Saraswati, Hamel, Ernest, Khan, Saeed R

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Rational design of novel antiandrogens for neutralizing androgen receptor function in hormone refractory prostate cancer von Singh, Pratap, Hallur, Gurulingappa, Anchoori, Ravi K., Bakare, Oladapo, Kageyama, Yukio, Khan, Saeed R., Isaacs, John T.

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Susceptibility of Aedes aegypti and Culex quinquefasciatus Larvae to Gedunin-Related Limonoids von Gurulingappa, Hallur, Tare, Vrushali, Pawar, Pushpa, Tungikar, Vijay, Jorapur, Yogesh R., Madhavi, Sriram, Bhat, Sujata V.

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