triple helix: 50 years later, the outcome von Duca, Maria, Vekhoff, Pierre, Oussedik, Kahina, Halby, Ludovic, Arimondo, Paola B

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DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge von Castillo-Aguilera, Omar, Depreux, Patrick, Halby, Ludovic, Arimondo, Paola B, Goossens, Laurence

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Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein von Bon, Corentin, Si, Yang, Pernak, Melanie, Barbachowska, Magdalena, Levi-Acobas, Eva, Daniel, Veronique Cadet, Jallet, Corinne, Ruzic, Dusan, Djokovic, Nemanja, Djikic, Teodora, Nikolic, Katarina, Halby, Ludovic, Arimondo, Paola B.

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Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors von Halby, Ludovic, Marechal, Nils, Pechalrieu, Dany, Cura, Vincent, Franchini, Don-Marc, Faux, Céline, Alby, Fréderic, Troffer-Charlier, Nathalie, Kudithipudi, Srikanth, Jeltsch, Albert, Aouadi, Wahiba, Decroly, Etienne, Guillemot, Jean-Claude, Page, Patrick, Ferroud, Clotilde, Bonnefond, Luc, Guianvarc'h, Dominique, Cavarelli, Jean, Arimondo, Paola B.

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Direct Synthesis of Allyl Amines with 2‐Nitrosulfonamide Derivatives via the Tsuji‐Trost Reaction von Bon, Corentin, Arimondo, Paola B., Halby, Ludovic

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DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites von Nardella, Flore, Halby, Ludovic, Hammam, Elie, Erdmann, Diane, Cadet-Daniel, Véronique, Peronet, Roger, Ménard, Didier, Witkowski, Benoit, Mecheri, Salah, Scherf, Artur, Arimondo, Paola B

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Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum von Nardella, Flore, Dobrescu, Irina, Hassan, Haitham, Rodrigues, Fabien, Thiberge, Sabine, Mancio-Silva, Liliana, Tafit, Ambre, Jallet, Corinne, Cadet-Daniel, Véronique, Goussin, Stéphane, Lorthiois, Audrey, Menon, Yoann, Molinier, Nicolas, Pechalrieu, Dany, Long, Christophe, Sautel, François, Matondo, Mariette, Duchateau, Magalie, Médard, Guillaume, Witkowski, Benoit, Scherf, Artur, Halby, Ludovic, Arimondo, Paola B.

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Targeting DNA Methylation with Small Molecules: What’s Next?: Miniperspective von Erdmann, Alexandre, Halby, Ludovic, Fahy, Jacques, Arimondo, Paola B

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Targeting DNA methylation with small molecules: what's next? von Erdmann, Alexandre, Halby, Ludovic, Fahy, Jacques, Arimondo, Paola B

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Sequence-specific targeting of IGF-I and IGF-IR genes by camptothecins von Oussedik, Kahina, François, Jean-Christophe, Halby, Ludovic, Senamaud-Beaufort, Catherine, Toutirais, Géraldine, Dallavalle, Sabrina, Pommier, Yves, Pisano, Claudio, Arimondo, Paola B

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Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic ‘writers’ von Bon, Corentin, Halby, Ludovic, Arimondo, Paola Barbara

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Editorial : Bisubstrate inhibitors: the promise of a selective and potent chemical inhibition of epigenetic “writers von Bon, Corentin, Halby, Ludovic, Arimondo, Paola B, Arimondo, Paola B

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Towards the sustainable discovery and development of new antibiotics von Miethke, Marcus, Pieroni, Marco, Weber, Tilmann, Brönstrup, Mark, Hammann, Peter, Halby, Ludovic, Arimondo, Paola B., Glaser, Philippe, Aigle, Bertrand, Bode, Helge B., Moreira, Rui, Li, Yanyan, Luzhetskyy, Andriy, Medema, Marnix H., Pernodet, Jean-Luc, Stadler, Marc, Tormo, José Rubén, Genilloud, Olga, Truman, Andrew W., Weissman, Kira J., Takano, Eriko, Sabatini, Stefano, Stegmann, Evi, Brötz-Oesterhelt, Heike, Wohlleben, Wolfgang, Seemann, Myriam, Empting, Martin, Hirsch, Anna K. H., Loretz, Brigitta, Lehr, Claus-Michael, Titz, Alexander, Herrmann, Jennifer, Jaeger, Timo, Alt, Silke, Hesterkamp, Thomas, Winterhalter, Mathias, Schiefer, Andrea, Pfarr, Kenneth, Hoerauf, Achim, Graz, Heather, Graz, Michael, Lindvall, Mika, Ramurthy, Savithri, Karlén, Anders, van Dongen, Maarten, Petkovic, Hrvoje, Keller, Andreas, Peyrane, Frédéric, Donadio, Stefano, Fraisse, Laurent, Piddock, Laura J. V., Gilbert, Ian H., Moser, Heinz E., Müller, Rolf

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Exploring the Cellular Activity of Camptothecin-Triple-Helix-Forming Oligonucleotide Conjugates von Arimondo, Paola B., Thomas, Craig J., Oussedik, Kahina, Baldeyrou, Brigitte, Mahieu, Christine, Halby, Ludovic, Guianvarc'h, Dominique, Lansiaux, Amélie, Hecht, Sidney M., Bailly, Christian, Giovannangeli, Carine

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Targeting MDR1 Gene: Synthesis and Cellular Study of Modified Daunomycin-Triplex-Forming Oligonucleotide Conjugates Able to Inhibit Gene Expression in Resistant Cell Lines von Stierlé, Vérène, Duca, Maria, Halby, Ludovic, Senamaud-Beaufort, Catherine, Capobianco, Massimo L, Laigle, Alain, Jollès, Béatrice, Arimondo, Paola B

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Optimized Synthesis and Enhanced Efficacy of Novel Triplex-Forming Camptothecin Derivatives Based on Gimatecan von Vekhoff, Pierre, Halby, Ludovic, Oussedik, Kahina, Dallavalle, Sabrina, Merlini, Lucio, Mahieu, Christine, Lansiaux, Amélie, Bailly, Christian, Boutorine, Alexandre, Pisano, Claudio, Giannini, Giuseppe, Alloatti, Domenico, Arimondo, Paola B

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DNA methylation inhibitors in cancer: Recent and future approaches von Gros, Christina, Fahy, Jacques, Halby, Ludovic, Dufau, Isabelle, Erdmann, Alexandre, Gregoire, Jean-Marc, Ausseil, Fréderic, Vispé, Stéphane, Arimondo, Paola B.

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Procainamide–SAHA Fused Inhibitors of hHDAC6 Tackle Multidrug-Resistant Malaria Parasites von Nardella, Flore, Halby, Ludovic, Dobrescu, Irina, Viluma, Johanna, Bon, Corentin, Claes, Aurélie, Cadet-Daniel, Véronique, Tafit, Ambre, Roesch, Camille, Hammam, Elie, Erdmann, Diane, Mairet-Khedim, Melissa, Peronet, Roger, Mecheri, Salah, Witkowski, Benoit, Scherf, Artur, Arimondo, Paola B

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Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells von Halby, Ludovic, Menon, Yoann, Rilova, Elodie, Pechalrieu, Dany, Masson, Véronique, Faux, Celine, Bouhlel, Mohamed Amine, David-Cordonnier, Marie-Hélène, Novosad, Natacha, Aussagues, Yannick, Samson, Arnaud, Lacroix, Laurent, Ausseil, Fréderic, Fleury, Laurence, Guianvarc’h, Dominique, Ferroud, Clotilde, Arimondo, Paola B

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Regioselective and efficient halogenation of 4,5-unsubstituted alkyl 3-hydroxypyrrole/3-hydroxythiophene-2-yl-carboxylates von Castillo-Aguilera, Omar, Depreux, Patrick, Halby, Ludovic, Azaroual, Nathalie, Arimondo, Paola B., Goossens, Laurence

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