Optimization of Hydroxyethylamine Transition State Isosteres as Aspartic Protease Inhibitors by Exploiting Conformational Preferences von Bueno, Ana B., Agejas, Javier, Broughton, Howard, Dally, Robert, Durham, Timothy B., Espinosa, Juan Félix, González, Rosario, Hahn, Patric J., Marcos, Alicia, Rodríguez, Ramón, Sanz, Gema, Soriano, José F., Timm, David, Vidal, Paloma, Yang, Hsiu-Chiung, McCarthy, James R.

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Gaussian Conversion Protocols for Cubic Phase State Generation von Zheng, Yu, Hahn, Oliver, Stadler, Pascal, Holmvall, Patric, Quijandría, Fernando, Ferraro, Alessandro, Ferrini, Giulia

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Design and Synthesis of α-Aryloxy-α-methylhydrocinnamic Acids:  A Novel Class of Dual Peroxisome Proliferator-Activated Receptor α/γ Agonists von Xu, Yanping, Rito, Christopher J, Etgen, Garret J, Ardecky, Robert J, Bean, James S, Bensch, William R, Bosley, Jacob R, Broderick, Carol L, Brooks, Dawn A, Dominianni, Samuel J, Hahn, Patric J, Liu, Sha, Mais, Dale E, Montrose-Rafizadeh, Chahrzad, Ogilvie, Kathy M, Oldham, Brian A, Peters, Mary, Rungta, Deepa K, Shuker, Anthony J, Stephenson, Gregory A, Tripp, Allie E, Wilson, Sarah B, Winneroski, Leonard L, Zink, Richard, Kauffman, Raymond F, McCarthy, James R

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Use of solid supported nucleophiles and electrophiles for the purification of non-peptide small molecule libraries von Kaldor, Stephen W., Siegel, Miles G., Fritz, James E., Dressman, Bruce A., Hahn, Patric J.

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Discovery of the First α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ‑8... von Gardinier, Kevin M, Gernert, Douglas L, Porter, Warren J, Reel, Jon K, Ornstein, Paul L, Spinazze, Patrick, Stevens, F. Craig, Hahn, Patric, Hollinshead, Sean P, Mayhugh, Daniel, Schkeryantz, Jeff, Khilevich, Albert, De Frutos, Oscar, Gleason, Scott D, Kato, Akihiko S, Luffer-Atlas, Debra, Desai, Prashant V, Swanson, Steven, Burris, Kevin D, Ding, Chunjin, Heinz, Beverly A, Need, Anne B, Barth, Vanessa N, Stephenson, Gregory A, Diseroad, Benjamin A, Woods, Tim A, Yu, Hong, Bredt, David, Witkin, Jeffrey M

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Abstract LB-274: Identification and characterization of LY3410738, a novel covalent inhibitor of cancer-associated mutant Isocitrate Dehydrogenase 1 (IDH1) von Brooks, Nathan, DeWalt, Robin, Boulet, Serge, Lu, ZhaoHai, Kays, Lisa, cavitt, Rachel, Gomez, Sandra, Strelow, John, Milligan, Paul, Roth, Kenneth, Bauer, Renato, Antonysamy, Stephen, Hahn, Patric, Rankovic, Zoran, McCann, Denis, Mo, Gary, Tiu, Ramon, Burkholder, Timothy, Geeganage, Sandaruwan, Gilmour, Raymond

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Fully Printed Inverters using Metal‐Oxide Semiconductor and Graphene Passives on Flexible Substrates von Singaraju, Surya Abhishek, Marques, Gabriel Cadilha, Gruber, Patric, Kruk, Robert, Hahn, Horst, Breitung, Ben, Aghassi-Hagmann, Jasmin

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physica status solidi (RRL) - Rapid Research Letters von Surya Abhishek Singaraju, Marques, Gabriel Cadilha, Gruber, Patric, Kruk, Robert, Hahn, Horst, Breitung, Ben, Aghassi-Hagmann, Jasmin

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Fully Printed Inverters using Metal‐Oxide Semiconductor and Graphene Passives on Flexible Substrates von Singaraju, Surya Abhishek, Marques, Gabriel Cadilha, Gruber, Patric, Kruk, Robert, Hahn, Horst, Breitung, Ben, Aghassi-Hagmann, Jasmin

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Rapid purification of small molecule libraries by ion exchange chromatography von Siegel, Miles G., Hahn, Patric J., Dressman, Bruce A., Fritz, James E., Grunwell, Jocelyn R., Kaldor, Stephen W.

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7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS MUTANT IDH1 AND IDH2 INHIBITORS von BURKHOLDER, Timothy Paul, RANKOVIC, Zoran, BOULET, Serge Louis, BAUER, Renato Alejandro, HAHN, Patric James, GILMOUR, Raymond

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7-PHENYLETHLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS MUTANT IDH1 AND IDH2 INHIBITORS von BURKHOLDER, Timothy Paul, RANKOVIC, Zoran, BOULET, Serge Louis, BAUER, Renato Alejandro, HAHN, Patric James, GILMOUR, Raymond

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7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitors von Rankovic, Zoran, Burkholder, Timothy Paul, Bauer, Renato Alejandro, Boulet, Serge Louis, Hahn, Patric James

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7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitors von Gilmour, Raymond, Rankovic, Zoran, Burkholder, Timothy Paul, Bauer, Renato Alejandro, Boulet, Serge Louis, Hahn, Patric James

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PYRIDO[4,3-D][1,3]OXAZIN-2-ONE COMPOUNDS AS MUTANT IDH1 AND IDH2 INHIBITORS von BURKHOLDER, Timothy Paul, RANKOVIC, Zoran, BOULET, Serge Louis, BAUER, Renato Alejandro, HAHN, Patric James, GILMOUR, Raymond

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Deterministic Gaussian conversion protocols for non-Gaussian single-mode resources von Hahn, Oliver, Holmvall, Patric, Stadler, Pascal, Ferrini, Giulia, Ferraro, Alessandro

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7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS MUTANT IDH1 AND IDH2 INHIBITORS von GILMOUR, RAYMOND, HAHN, PATRIC JAMES, RANKOVIC, ZORAN, BAUER, RENATO ALEJANDRO, BOULET, SERGE LOUIS, BURKHOLDER, TIMOTHY PAUL

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DÉRIVÉS DE PYRIDO[4,3-D][1,3]OXAZIN-2-ONE EN TANT QU'INHIBITEURS DE LA FORME MUTÉE DES PROTÉINES IDH1 ET IDH2 von BURKHOLDER, Timothy Paul, RANKOVIC, Zoran, BOULET, Serge Louis, BAUER, Renato Alejandro, HAHN, Patric James, GILMOUR, Raymond

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7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as mutant IDH1 and IDH2 inhibitors von Gilmour, Raymond, Rankovic, Zoran, Burkholder, Timothy Paul, Bauer, Renato Alejandro, Boulet, Serge Louis, Hahn, Patric James

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O1-06-02: The design and synthesis of an efficacious BACE inhibitor von McCarthy, James R., Agejas, Javier, Bender, David M., Broughton, Howard, Bueno, Ana, Dally, Robert D., Durham, Timothy, Erickson, Jon A., Espinosa, Juan F., Gonzalez, Rosario, Hahn, Patric J., Laigle, Debra K., Kohn, Todd J., May, Patrick C., Rodriguez, Juan R., Sanz, Gema, Shepherd, Timothy A., Timm, David, Vidal, Paloma, Yang, Hsiu-Chiung

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