E7766, a Macrocycle‐Bridged Stimulator of Interferon Genes (STING) Agonist with Potent Pan‐Genotypic Activity von Kim, Dae‐Shik, Endo, Atsushi, Fang, Francis G., Huang, Kuan‐Chun, Bao, Xingfeng, Choi, Hyeong‐wook, Majumder, Utpal, Shen, Young Y., Mathieu, Steven, Zhu, Xiaojie, Sanders, Kristen, Noland, Thomas, Hao, Ming‐Hong, Chen, Yu, Wang, John Y., Yasui, So, TenDyke, Karen, Wu, Jiayi, Ingersoll, Christy, Loiacono, Kara A., Hutz, Janna E., Sarwar, Nadeem

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Building C(sp3)-rich complexity by combining cycloaddition and C–C cross-coupling reactions von Chen, Tie–Gen, Barton, Lisa M., Lin, Yutong, Tsien, Jet, Kossler, David, Bastida, Iñaki, Asai, Shota, Bi, Cheng, Chen, Jason S., Shan, Mingde, Fang, Hui, Fang, Francis G., Choi, Hyeong-wook, Hawkins, Lynn, Qin, Tian, Baran, Phil S.

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Apratoxin A Shows Novel Pancreas-Targeting Activity through the Binding of Sec 61 von Huang, Kuan-Chun, Chen, Zhihong, Jiang, Yimin, Akare, Sandeep, Kolber-Simonds, Donna, Condon, Krista, Agoulnik, Sergei, Tendyke, Karen, Shen, Yongchun, Wu, Kuo-Ming, Mathieu, Steven, Choi, Hyeong-Wook, Zhu, Xiaojie, Shimizu, Hajime, Kotake, Yoshihiko, Gerwick, William H, Uenaka, Toshimitsu, Woodall-Jappe, Mary, Nomoto, Kenichi

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M-COPA, a Golgi Disruptor, Inhibits Cell Surface Expression of MET Protein and Exhibits Antitumor Activity against MET-Addicted Gastric Cancers von Ohashi, Yoshimi, Okamura, Mutsumi, Hirosawa, Asaka, Tamaki, Naomi, Akatsuka, Akinobu, Wu, Kuo-Ming, Choi, Hyeong-Wook, Yoshimatsu, Kentaro, Shiina, Isamu, Yamori, Takao, Dan, Shingo

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Targeting the Golgi apparatus to overcome acquired resistance of non-small cell lung cancer cells to EGFR tyrosine kinase inhibitors von Ohashi, Yoshimi, Okamura, Mutsumi, Katayama, Ryohei, Fang, Siyang, Tsutsui, Saki, Akatsuka, Akinobu, Shan, Mingde, Choi, Hyeong-Wook, Fujita, Naoya, Yoshimatsu, Kentaro, Shiina, Isamu, Yamori, Takao, Dan, Shingo

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Synthesis of a Polycyclic Halichondrin C1–C14 Fragment via Intermolecular Oxy-Michael/Trans-Ketalization von Kim, Dae-Shik, Fang, Francis G, Choi, Hyeong-wook, Fang, Hui

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Synthesis of the Halichondrin C1–C15 Fragment from a Halaven C27–C35 Byproduct: Stereospecific Intramolecular Kishi Reduction von Kim, Dae-Shik, Fang, Francis G, Choi, Hyeong-wook, Fang, Hui

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Asymmetric Ni(II)/Cr(II)-Mediated Coupling Reaction:  Catalytic Process von Choi, Hyeong-wook, Nakajima, Katsumasa, Demeke, Damtew, Kang, Fu-An, Jun, Hyuk-Sang, Wan, Zhao-Kui, Kishi, Yoshito

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Asymmetric Ni(II)/Cr(II)-Mediated Coupling Reaction:  Stoichiometric Process von Wan, Zhao-Kui, Choi, Hyeong-wook, Kang, Fu-An, Nakajima, Katsumasa, Demeke, Damtew, Kishi, Yoshito

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EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity von Campbell, John E, Kuntz, Kevin W, Knutson, Sarah K, Warholic, Natalie M, Keilhack, Heike, Wigle, Tim J, Raimondi, Alejandra, Klaus, Christine R, Rioux, Nathalie, Yokoi, Akira, Kawano, Satoshi, Minoshima, Yukinori, Choi, Hyeong-Wook, Porter Scott, Margaret, Waters, Nigel J, Smith, Jesse J, Chesworth, Richard, Moyer, Mikel P, Copeland, Robert A

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Prins Reaction of Homoallenyl Alcohols: Access to Substituted Pyrans in the Halichondrin Series von Choi, Hyeong-wook, Fang, Francis G., Fang, Hui, Kim, Dae-Shik, Mathieu, Steven R., Yu, Robert T.

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Discovery and characterization of stereodefined PMO-gapmers targeting tau von Kanatsu, Kunihiko, Takahashi, Yoshinori, Sakaguchi, Tetsuya, Kim, Dae-Shik, Murota, Miki, Shan, Mingde, Fukami, Kazuki, Itano, Wataru, Kikuta, Kenji, Yoshimura, Hikaru, Kurokawa, Toshiki, Nagayama, Yuko, Ishikawa, Rena, Dairiki, Ryo, Zhou, Zhi, Sanders, Kristen, Stupalski, Jacob, Yasui, So, Liu, Diana, Benayoud, Farid, Fang, Hui, Jing, Enxuan, Ogo, Makoto, Fang, Francis G., Wang, John, Choi, Hyeong-wook

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Synthetic studies on the marine natural product halichondrins von Choi, Hyeong-wook, Demeke, Damtew, Kang, F.-A., Kishi, Y., Nakajima, K., Nowak, P., Wan, Z.-K., Xie, C.

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Total Synthesis of Natural (+)-Lasonolide A von Kang, Sung Ho, Kang, Suk Youn, Kim, Chul Min, Choi, Hyeong-wook, Jun, Hyuk-Sang, Lee, Byeong Moon, Park, Chul Min, Jeong, Joon Won

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Mixed-mode separation of antisense oligonucleotides using a single column with complementary anion-exchange and hydrophobic interaction chromatography approaches von Kazarian, Artaches A., Lee, Jung Hwa, Mitasev, Branko, Choi, Hyeong-wook

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Efficient Activation of Zinc: Application of the Blaise Reaction to an Expedient Synthesis of a Statin Intermediate von Shin, Hyunik, Choi, Bo Seung, Lee, Ki Kon, Choi, Hyeong-wook, Chang, Jay Hyok, Lee, Kyu Woong, Nam, Do Hyun, Kim, No-Soo

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Abstract 592: Demonstration of E7766, a novel STING agonist, as a potent immunotherapy in BCG-insensitive non-muscle invasive bladder cancer models via intravesical administration von Huang, Kuan-Chun, Zhang, Chi, Yu, Kun, Kim, Dae-Shik, Dixit, Vaishali, Hukkanen, Renee, Choi, Hyeong-Wook, Hutz, Janna, Fang, Frank, Bao, Xingfeng

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Stereoselective Total Synthesis of the Natural (+)-Lasonolide A von Kang, Sung Ho, Kang, Suk Youn, Choi, Hyeong-wook, Kim, Chul Min, Jun, Hyuk-Sang, Youn, Joo-Hack

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Development of a Scalable Synthetic Route towards a Thrombin Inhibitor, LB30057 von Kim, Bong Chan, Hwang, Sang Yeul, Lee, Tae Hee, Chang, Jay Hyok, Choi, Hyeong-wook, Lee, Kyu Woong, Choi, Bo Seung, Kim, Young Keun, Lee, Jae Hoon, Kim, Won Sup, Oh, Yeong Soo, Lee, Hee Bong, Kim, Kyu Young, Shin, Hyunik

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Efficient Synthesis of Clitocine via 1,3-N (endo) to N (exo) Migration: A Revision to Kini’s Work von Choi, Hyeong-wook, Choi, Bo Seung, Chang, Jay Hyok, Lee, Kyu Woong, Nam, Do Hyun, Kim, Young Keun, Lee, Jae Hoon, Heo, Taeho, Shin, Hyunik, Kim, No-Soo

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