BU08073 a buprenorphine analogue with partial agonist activity at μ‐receptors in vitro but long‐lasting opioid antagonist activity in vivo in mice von Khroyan, T V, Wu, J, Polgar, W E, Cami‐Kobeci, G, Fotaki, N, Husbands, S M, Toll, L

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Activities of mixed NOP and μ‐opioid receptor ligands von Spagnolo, B, Calo, G, Polgar, W E, Jiang, F, Olsen, C M, Berzetei‐Gurske, I, Khroyan, T V, Husbands, S M, Lewis, J W, Toll, L, Zaveri, N T

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Pyrrolo- and pyridomorphinans: Non-selective opioid antagonists and delta opioid agonists/mu opioid partial agonists von Kumar, V., Clark, M.J., Traynor, J.R., Lewis, J.W., Husbands, S.M.

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Characterization of [3H]Harmane Binding to Rat Whole Brain Membranes von ANDERSON, N J., ROBINSON, ES J., HUSBANDS, S M., DELAGRANGE, P, NUTT, D J., HUDSON, A L.

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3-Deoxyclocinnamox:  The First High-Affinity, Nonpeptide μ-Opioid Antagonist Lacking a Phenolic Hydroxyl Group von Derrick, Ian, Neilan, Claire L, Andes, Jennifer, Husbands, Stephen M, Woods, James H, Traynor, John R, Lewis, John W

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Structure−Activity Relationships at the Monoamine Transporters and σ Receptors for a Novel Series of 9-[3-(cis-3,5-Dimethyl-1-piperazinyl)-propyl]carbazole (Rimcazole) Analogues von Husbands, Stephen M, Izenwasser, Sari, Kopajtic, Theresa, Bowen, Wayne D, Vilner, Bertold J, Katz, Jonathan L, Newman, Amy Hauck

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Design and Synthesis of [(2,3-Dichlorophenyl)piperazin-1-yl]alkylfluorenylcarboxamides as Novel Ligands Selective for the Dopamine D3 Receptor Subtype von Robarge, Michael J, Husbands, Stephen M, Kieltyka, Andrzej, Brodbeck, Robbin, Thurkauf, Andrew, Newman, Amy Hauck

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14β-O-Cinnamoylnaltrexone and Related Dihydrocodeinones are Mu Opioid Receptor Partial Agonists with Predominant Antagonist Activity von Moynihan, H, Jales, A. R, Greedy, B. M, Rennison, D, Broadbear, J. H, Purington, L, Traynor, J. R, Woods, J. H, Lewis, J. W, Husbands, S. M

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14 beta-O-cinnamoylnaltrexone and related dihydrocodeinones are mu opioid receptor partial agonists with predominant antagonist activity von Moynihan, H, Jales, A R, Greedy, B M, Rennison, D, Broadbear, J H, Purington, L, Traynor, J R, Woods, J H, Lewis, J W, Husbands, S M

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Ring constrained analogues of the orvinols: The furanomorphides von Husbands, Stephen M., Breeden, Simon W., Grivas, Konstantinos, Lewis, John W.

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Structural Determinants of Efficacy for κ Opioid Receptors in the Orvinol Series:  7,7-Spiro Analogues of Buprenorphine von Husbands, Stephen M, Lewis, John W

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β -carboline binding to imidazoline receptors von Husbands, Stephen M., Glennon, Richard A., Gorgerat, Stephane, Gough, Rhianon, Tyacke, Robin, Crosby, John, Nutt, David J., Lewis, John W., Hudson, Alan L.

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Isothiocyanate Derivatives of 9-[3-(cis-3,5-Dimethyl-1-piperazinyl)propyl]- carbazole (Rimcazole):  Irreversible Ligands for the Dopamine Transporter von Husbands, Stephen M, Izenwasser, Sari, Loeloff, Richard J, Katz, Jonathan L, Bowen, Wayne D, Vilner, Bertold J, Newman, Amy Hauck

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3-Alkyl Ethers of Clocinnamox:  Delayed Long-Term μ-Antagonists with Variable μ Efficacy von Husbands, Stephen M, Sadd, John, Broadbear, Jillian H, Woods, James H, Martin, Jason, Traynor, John R, Aceto, Mario D, Bowman, Edward R, Harris, Louis S, Lewis, John W

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Rimcazole analogs attenuate the convulsive effects of cocaine: correlation with binding to sigma receptors rather than dopamine transporters von Matsumoto, Rae R, Hewett, Kizzy L, Pouw, Buddy, Bowen, Wayne D, Husbands, Stephen M, Cao, Jian Jing, Hauck Newman, Amy

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Characterization of the complex morphinan derivative BU72 as a high efficacy, long-lasting mu-opioid receptor agonist von Neilan, Claire L., Husbands, Stephen M., Breeden, Simon, Ko, M.C. (Holden), Aceto, Mario D., Lewis, John W., Woods, James H., Traynor, John R.

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Major Effect of Pyrrolic N-Benzylation in Norbinaltorphimine, the Selective κ-Opioid Receptor Antagonist von Chauvignac, Cédric, Miller, Carl N, Srivastava, Sanjay K, Lewis, John W, Husbands, Stephen M, Traynor, John R

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A novel orvinol analog, BU08028, as a safe opioid analgesic without abuse liability in primates von Ding, Huiping, Czoty, Paul W., Kiguchi, Norikazu, Cami-Kobeci, Gerta, Sukhtankar, Devki D., Nader, Michael A., Husbands, Stephen M., Ko, Mei-Chuan

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Probes for imidazoline binding sites : Synthesis and evaluation of a selective, irreversible I2 ligand von COATES, P. A, GRUNDT, P, ROBINSON, E. S. J, NUTT, D. J, TYACKE, R, HUDSON, A. L, LEWIS, J. W, HUSBANDS, S. M

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BU10038 as a safe opioid analgesic with fewer side-effects after systemic and intrathecal administration in primates von Kiguchi, Norikazu, Ding, Huiping, Cami-Kobeci, Gerta, Sukhtankar, Devki D., Czoty, Paul W., DeLoid, Heather B., Hsu, Fang-Chi, Toll, Lawrence, Husbands, Stephen M., Ko, Mei-Chuan

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