Discovery of bioactive molecules from CuAAC click-chemistry-based combinatorial libraries von Wang, Xueshun, Huang, Boshi, Liu, Xinyong, Zhan, Peng

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First discovery of novel 3-hydroxy-quinazoline-2,4(1H,3H)-diones as specific anti-vaccinia and adenovirus agents via ‘privileged scaffold’ refining approach von Kang, Dongwei, Zhang, Heng, Zhou, Zhongxia, Huang, Boshi, Naesens, Lieve, Zhan, Peng, Liu, Xinyong

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Newly Emerging Strategies in Antiviral Drug Discovery: Dedicated to Prof. Dr. Erik De Clercq on Occasion of His 80th Anniversary von Xu, Shujing, Ding, Dang, Zhang, Xujie, Sun, Lin, Kang, Dongwei, Huang, Boshi, Liu, Xinyong, Zhan, Peng

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Teaching an old dog new tricks: Drug discovery by repositioning natural products and their derivatives von Huang, Boshi, Zhang, Yan

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Discovery of non-peptide small molecular CXCR4 antagonists as anti-HIV agents: Recent advances and future opportunities von Zhang, Heng, Kang, Dongwei, Huang, Boshi, Liu, Na, Zhao, Fabao, Zhan, Peng, Liu, Xinyong

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VZHE-039, a novel antisickling agent that prevents erythrocyte sickling under both hypoxic and anoxic conditions von Abdulmalik, Osheiza, Pagare, Piyusha P., Huang, Boshi, Xu, Guoyan G., Ghatge, Mohini S., Xu, Xiaomeng, Chen, Qiukan, Anabaraonye, Nancy, Musayev, Faik N., Omar, Abdelsattar M., Venitz, Jürgen, Zhang, Yan, Safo, Martin K.

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Discovery of GluN2A subtype-selective N -methyl-d-aspartate (NMDA) receptor ligands von Jiang, Liyang, Liu, Na, Zhao, Fabao, Huang, Boshi, Kang, Dongwei, Zhan, Peng, Liu, Xinyong

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Medicinal chemistry insights in the discovery of novel LSD1 inhibitors von Wang, Xueshun, Huang, Boshi, Suzuki, Takayoshi, Liu, Xinyong, Zhan, Peng

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Exploring the hydrophobic channel of NNIBP leads to the discovery of novel piperidine-substituted thiophene[3,2-d]pyrimidine derivatives as potent HIV-1 NNRTIs von Kang, Dongwei, Feng, Da, Ginex, Tiziana, Zou, Jinmi, Wei, Fenju, Zhao, Tong, Huang, Boshi, Sun, Yanying, Desta, Samuel, De Clercq, Erik, Pannecouque, Christophe, Zhan, Peng, Liu, Xinyong

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Design, Synthesis, and Investigation of Novel Nitric Oxide (NO)-Releasing Aromatic Aldehydes as Drug Candidates for the Treatment of Sickle Cell Disease von Huang, Boshi, Ghatge, Mohini S., Donkor, Akua K., Musayev, Faik N., Deshpande, Tanvi M., Al-Awadh, Mohammed, Alhashimi, Rana T., Zhu, Hongmei, Omar, Abdelsattar M., Telen, Marilyn J., Zhang, Yan, McMahon, Tim J., Abdulmalik, Osheiza, Safo, Martin K.

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An improved synthesis approach of the HIV-1 inhibitor RDEA427, a pyrrolo[2,3-d]pyrimidine derivative von Huang, Boshi, Liu, Xinhao, Li, Wanzhuo, Chen, Zihui, Kang, Dongwei, Zhan, Peng, Liu, Xinyong

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Design, Synthesis, and Antisickling Investigation of a Thiazolidine Prodrug of TD-7 That Prolongs the Duration of Action of Antisickling Aromatic Aldehyde von Alhashimi, Rana T., Ahmed, Tarek A., Alghanem, Lamya, Pagare, Piyusha P., Huang, Boshi, Ghatge, Mohini S., Omar, Abdelsattar M., Abdulmalik, Osheiza, Zhang, Yan, Safo, Martin K.

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Discovery of diarylpyrimidine derivatives bearing piperazine sulfonyl as potent HIV-1 nonnucleoside reverse transcriptase inhibitors von Jiang, Xiangyi, Huang, Boshi, Rumrill, Shawn, Pople, David, Zalloum, Waleed A., Kang, Dongwei, Zhao, Fabao, Ji, Xiangkai, Gao, Zhen, Hu, Lide, Wang, Zhao, Xie, Minghui, De Clercq, Erik, Ruiz, Francesc X., Arnold, Eddy, Pannecouque, Christophe, Liu, Xinyong, Zhan, Peng

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The development of an effective synthetic route of lesinurad (RDEA594) von Meng, Qing, Zhao, Tong, Kang, Dongwei, Huang, Boshi, Zhan, Peng, Liu, Xinyong

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Effective and Versatile Synthesis of Ginkgotoxin and Its 4′-O-Derivatives through Regioselective 4′-O-Alkylation and 4′-O-Chlorination of 3,5′-O-Dibenzylpyridoxine von Huang, Boshi, Danso-Danquah, Richmond, Safo, Martin K., Zhang, Yan

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Discovery of piperidine-substituted thiazolo[5,4-d]pyrimidine derivatives as potent and orally bioavailable HIV-1 non-nucleoside reverse transcriptase inhibitors von Kang, Dongwei, Zhao, Tong, Wang, Zhao, Feng, Da, Zhang, Heng, Huang, Boshi, Wu, Gaochan, Wei, Fenju, Zhou, Zhongxia, Jing, Lanlan, Zuo, Xiaofang, Tian, Ye, Poongavanam, Vasanthanathan, Kongsted, Jacob, De Clercq, Erik, Pannecouque, Christophe, Zhan, Peng, Liu, Xinyong

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Design, Synthesis, and Antisickling Investigation of a Nitric Oxide-Releasing Prodrug of 5HMF for the Treatment of Sickle Cell Disease von Alhashimi, Rana T, Ghatge, Mohini S, Donkor, Akua K, Deshpande, Tanvi M, Anabaraonye, Nancy, Alramadhani, Dina, Danso-Danquah, Richmond, Huang, Boshi, Zhang, Yan, Musayev, Faik N, Abdulmalik, Osheiza, Safo, Martin K

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Recent advances in multitarget-directed ligands targeting G-protein-coupled receptors von Ma, Hongguang, Huang, Boshi, Zhang, Yan

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Inhibitors of Influenza Virus Polymerase Acidic (PA) Endonuclease: Contemporary Developments and Perspectives von Ju, Han, Zhang, Jian, Huang, Boshi, Kang, Dongwei, Huang, Bing, Liu, Xinyong, Zhan, Peng

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Determination of Cadmium in Water Samples by FR-PAN Fluorescence Method von Wang, Xinqing, Lin, Dongying, Liu, Jingjing, Xiao, Xilin, Ren, Lanxing, Huang, Boshi, Xue, Jinhua

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