Copper-Catalyzed C–N Coupling in the Synthesis of Integrase Inhibitors of Immunodeficiency Viruses von Lin, Jinguan, Houpis, Ioannis N, Liu, Renmao, Wang, Youchu, Zhang, Jianqian

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Efficient Large-Scale Synthesis of BILN 2061, a Potent HCV Protease Inhibitor, by a Convergent Approach Based on Ring-Closing Metathesis von Yee, Nathan K, Farina, Vittorio, Houpis, Ioannis N, Haddad, Nizar, Frutos, Rogelio P, Gallou, Fabrice, Wang, Xiao-jun, Wei, Xudong, Simpson, Robert D, Feng, Xuwu, Fuchs, Victor, Xu, Yibo, Tan, Jonathan, Zhang, Li, Xu, Jinghua, Smith-Keenan, Lana L, Vitous, Jana, Ridges, Michael D, Spinelli, Earl M, Johnson, Michael, Donsbach, Kai, Nicola, Thomas, Brenner, Michael, Winter, Eric, Kreye, Paul, Samstag, Wendelin

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Amination of aryl halides using copper catalysis von Lang, Fengrui, Zewge, Daniel, Houpis, Ioannis N, Volante, R.P

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Efficient Synthesis of (S)-2-(Cyclopentyloxycarbonyl)-amino-8-nonenoic Acid:  Key Building Block for BILN 2061, an HCV NS3 Protease Inhibitor von Wang, Xiao-jun, Zhang, Li, Smith-Keenan, Lana L, Houpis, Ioannis N, Farina, Vittorio

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Stereoselective C-Glycosylation Reactions with Arylzinc Reagents von Lemaire, Sébastien, Houpis, Ioannis N, Xiao, Tingting, Li, Juanjuan, Digard, Eric, Gozlan, Charlotte, Liu, Renmao, Gavryushin, Andrey, Diène, Coura, Wang, Youchu, Farina, Vittorio, Knochel, Paul

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Synthesis of 4,4′-Disubstituted Azepines via Ring-Closing Metathesis Reaction and Asymmetric Arylation of Lactones von Delhaye, Laurent, Merschaert, Alain, Diker, Khalid, Houpis, Ioannis N.

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Synthesis of a Muscarinic Receptor Antagonist via a Diastereoselective Michael Reaction, Selective Deoxyfluorination and Aromatic Metal−Halogen Exchange Reaction von Mase, Toshiaki, Houpis, Ioannis N, Akao, Atsushi, Dorziotis, Ilias, Emerson, Khateeta, Hoang, Thoa, Iida, Takehiko, Itoh, Takahiro, Kamei, Keisuke, Kato, Shinji, Kato, Yoshiaki, Kawasaki, Masashi, Lang, Fengrui, Lee, Jaemoon, Lynch, Joseph, Maligres, Peter, Molina, Audrey, Nemoto, Takayuki, Okada, Shigemitsu, Reamer, Robert, Song, Jake Z, Tschaen, David, Wada, Toshihiro, Zewge, Daniel, Volante, R. P, Reider, Paul J, Tomimoto, Koji

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Total synthesis of glycinoeclepin A von Corey, E. J, Houpis, Ioannis N

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Regioselective Cross-Coupling Reactions of Boronic Acids with Dihalo Heterocycles von Houpis, Ioannis N, Liu, Renmao, Wu, Yanfei, Yuan, Yukuan, Wang, Youchu, Nettekoven, Ulrike

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Carboxylate Directed Cross-Coupling Reactions in the Synthesis of Trisubstituted Benzoic Acids von Houpis, Ioannis N, Huang, Changkang, Nettekoven, Ulrike, Chen, Jason G, Liu, Renmao, Canters, Martine

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Utilization of Sequential Palladium-Catalyzed Cross-Coupling Reactions in the Stereospecific Synthesis of Trisubstituted Olefins von Houpis, Ioannis N, Shilds, Didier, Nettekoven, Ulrike, Schnyder, Anita, Bappert, Erhart, Weerts, Koen, Canters, Martine, Vermuelen, Wim

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Condensation of 2-methylbenzoxazole with aromatic aldehydes bearing acidic protons. A convenient coupling in the synthesis of the HIV-reverse transcriptase inhibitor L-696,229 von Houpis, Ioannis N, Molina, Audrey, Lynch, Joseph, Reamer, Robert A, Volante, R. P, Reider, Paul J

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Palladium- and Copper-Catalyzed Site Selective Monoamination of Dibromobenzoic Acid von Houpis, Ioannis N., Weerts, Koen, Nettekoven, Ulrike, Canters, Martine, Tan, Hongyu, Liu, Renmao, Wang, Youchu

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Palladium(II)-catalyzed coupling of 2-carboxyethyl enol triflates with organostannanes von Houpis, Ioannis N.

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Synthesis of PPAR Agonist via Asymmetric Hydrogenation of a Cinnamic Acid Derivative and Stereospecific Displacement of (S)-2-Chloropropionic Acid von Houpis, Ioannis N, Patterson, Lawrence E, Alt, Charles A, Rizzo, John R, Zhang, Tony Y, Haurez, Michael

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Nickel Catalyzed Reactions of Nucleophiles with Unactivated and Partially Activated Olefins and Acetylenes von Houpis, Ioannis N., Lee, Jaemoon

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The control of diastereoselectivity in the Michael reaction of ketonic enolates with crotonic acid derivatives von Corey, E.J., Houpis, Ioannis N.

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Utilization of Sequential Palladium-Catalyzed Cross-Coupling Reactions in the Stereospecific Synthesis of Trisubstituted Olefins von Houpis, Ioannis N, Schils, Didier, Nettekoven, Ulrike, Schnyder, Anita, Bappert, Erhart, Weerts, Koen, Canters, Martine, Vermeulen, Wim

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Synthesis of a Peroxime Proliferator Activated Receptor (PPAR) α/γ Agonist via Stereocontrolled Williamson Ether Synthesis and Stereospecific SN2 Reaction of S-2-Chloro Propionic A... von Aikins, James A, Haurez, Michael, Rizzo, John R, Van Hoeck, Jean-Pierre, Brione, Willy, Kestemont, Jean-Paul, Stevens, Christophe, Lemair, Xavier, Stephenson, Gregory A, Marlot, Eric, Forst, Mindy, Houpis, Ioannis N

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Metal-halogen exchange-initiated cyclization of iodo carbonyl compounds von Cooke, Manning P., Houpis, Ioannis N.

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