The β-d-Glucose Scaffold as a β-Turn Mimetic von Hirschmann, Ralph F, Nicolaou, K. C, Angeles, Angie R, Chen, Jason S, Smith, Amos B

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Medicinal Chemistry in the Golden Age of Biology: Lessons from Steroid and Peptide Research von Hirschmann, Ralph

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Peptide Synthesis Catalyzed by an Antibody Containing a Binding Site for Variable Amino Acids von Hirschmann, Ralph, Smith, Amos B., Taylor, Carol M., Benkovic, Patricia A., Taylor, Scott D., Yager, Kraig M., Sprengeler, Paul A., Benkovic, Stephen J.

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Pyrrolinone-Based Peptidomimetics.“Let the Enzyme or Receptor be the Judge” von Smith, Amos B, Charnley, Adam K, Hirschmann, Ralph

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De novo design and synthesis of somatostatin non-peptide peptidomimetics utilizing .beta.-D-glucose as a novel scaffolding von Hirschmann, Ralph, Nicolaou, K. C, Pietranico, Sherrie, Leahy, Ellen M, Salvino, Joseph, Arison, Byron, Cichy, Maria A, Spoors, P. Grant, Shakespeare, William C

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Modulation of Receptor and Receptor Subtype Affinities Using Diastereomeric and Enantiomeric Monosaccharide Scaffolds as a Means to Structural and Biological Diversity. A New Route... von Hirschmann, Ralph, Hynes, John, Cichy-Knight, Maria A, van Rijn, Rachel D, Sprengeler, Paul A, Spoors, P. Grant, Shakespeare, William C, Pietranico-Cole, Sherrie, Barbosa, Joseph, Liu, Josephine, Yao, Wenqing, Rohrer, Susan, Smith, Amos B

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The cortisone era: aspects of its impact. Some contributions of the Merck Laboratories von Hirschmann, Ralph

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Novel Ligands Lacking a Positive Charge for the δ- and μ-Opioid Receptors von Schiller, Peter W, Berezowska, Irena, Nguyen, Thi M.-D, Schmidt, Ralf, Lemieux, Carole, Chung, Nga N, Falcone-Hindley, Margaret L, Yao, Wenqing, Liu, Josephine, Iwama, Seiji, Smith, Amos B, Hirschmann, Ralph

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Design, synthesis, and crystal structure of a pyrrolinone-based peptidomimetic possessing the conformation of a .beta.-strand: potential application to the design of novel inhibito... von Smith, Amos B., Keenan, Terence P., Holcomb, Ryan C., Sprengeler, Paul A., Guzman, Mark C., Wood, John L., Carroll, Patrick J., Hirschmann, Ralph

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Peptide bond formation via catalytic antibodies: Synthesis of a novel phosphonate diester hapten von Smith, Amos B., Taylor, Carol M., Benkovic, Stephen J., Hirschmann, Ralph

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Design, Synthesis, and Evaluation of a Pyrrolinone-Based Matrix Metalloprotease Inhibitor von Smith, Amos B, Nittoli, Thomas, Sprengeler, Paul A, Duan, James J.-W, Liu, Rui-Qin, Hirschmann, Ralph F

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Pyrrolinone-Based Peptidomimetics: “ von Smith, Amos B., Charnley, Adam K., Hirschmann, Ralph

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The Crystal Structure of a Pyrrolinone−Peptide Hybrid Ligand Bound to the Human Class II MHC Protein HLA-DR1 von Lee, Kon Ho, Olson, Gary L, Bolin, David R, Benowitz, Andrew B, Sprengeler, Paul A, Smith, Amos B, Hirschmann, Ralph F, Wiley, Don C

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The first design and synthesis of a steroidal peptidomimetic. The potential value of peptidomimetics in elucidating the bioactive conformation of peptide ligands von Hirschmann, Ralph, Sprengeler, Paul A, Kawasaki, Tomomi, Leahy, James W, Shakespeare, William C, Smith, Amos B

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Cyclic Peptide Formation Catalyzed by an Antibody Ligase von Smithrud, David B., Benkovic, Patricia A., Benkovic, Stephen J., Roberts, Victoria, Liu, Josephine, Neagu, Irina, Iwama, Seiji, Phillips, Barton W., Smith, Amos B., Hirschmann, Ralph

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Synthesis of a Substance P Antagonist with a Somatostatin Scaffold:  Factors Affecting Agonism/Antagonism at GPCRs and the Role of Pseudosymmetry von Liu, Josephine, Underwood, Dennis J, Cascieri, Margaret A, Rohrer, Susan P, Cantin, Louis-David, Chicchi, Gary, Smith, Amos B, Hirschmann, Ralph

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Design, Synthesis, and Structural Analysis of d,l-Mixed Polypyrrolinones. 1. From Nonpeptide Peptidomimetics to Nanotubes von Smith, III, Amos B, Wang, Wenyong, Charnley, Adam K, Carroll, Patrick J, Kenesky, Craig S, Hirschmann, Ralph

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Azide and Cyanide Displacements via Hypervalent Silicate Intermediates von Soli, Eric D, Manoso, Amy S, Patterson, Michael C, DeShong, Philip, Favor, David A, Hirschmann, Ralph, Smith, Amos B

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Design, Synthesis, and Structural Analysis of d,l-Mixed Polypyrrolinones. 2. Macrocyclic Hexapyrrolinones von Smith, III, Amos B, Xiong, Hui, Charnley, Adam K, Brenner, Meinrad, Mesaros, Eugen F, Kenesky, Craig S, Di Costanzo, Luigi, Christianson, David W, Hirschmann, Ralph

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Development of an Efficient, Regio- and Stereoselective Route to Libraries Based on the β-d-Glucose Scaffold von Hirschmann, Ralph, Ducry, Laurent, Smith, Amos B

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