Synthesis and Activity of New Aryl- and Heteroaryl-Substituted Pyrazole Inhibitors of the Transforming Growth Factor-β Type I Receptor Kinase Domain von Sawyer, J. Scott, Anderson, Bryan D, Beight, Douglas W, Campbell, Robert M, Jones, Michael L, Herron, David K, Lampe, John W, McCowan, Jefferson R, McMillen, William T, Mort, Nicholas, Parsons, Stephen, Smith, Edward C. R, Vieth, Michal, Weir, Leonard C, Yan, Lei, Zhang, Faming, Yingling, Jonathan M

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Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain von SAWYER, J. Scott, BEIGHT, Douglas W, PARSONS, Stephen, SMITH, Edward C. R, WAGNER, Jill R, LEI YAN, FAMING ZHANG, YINGLING, Jonathan M, BRITT, Karen S, ANDERSON, Bryan D, CAMPBELL, Robert M, GOODSON, Theodore JR, HERRON, David K, LI, Hong-Yu, MCMILLEN, William T, MORT, Nicholas

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Kinetic Characterization of Novel Pyrazole TGF-β Receptor I Kinase Inhibitors and Their Blockade of the Epithelial−Mesenchymal Transition von Peng, Sheng-Bin, Yan, Lei, Xia, Xiaoling, Watkins, Scott A, Brooks, Harold B, Beight, Douglas, Herron, David K, Jones, Michael L, Lampe, John W, McMillen, William T, Mort, Nicholas, Sawyer, J. Scott, Yingling, Jonathan M

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Anthranilamide inhibitors of factor Xa von Mendel, David, Marquart, Angela L., Joseph, Sajan, Waid, Philip, Yee, Ying K., Tebbe, Anne Louise, Ratz, Andrew M., Herron, David K., Goodson, Theodore, Masters, John J., Franciskovich, Jeffry B., Tinsley, Jennifer M., Wiley, Michael R., Weir, Leonard C., Kyle, Jeffrey A., Klimkowski, Valentine J., Smith, Gerald F., Towner, Richard D., Froelich, Larry L., Buben, John, Craft, Trelia J.

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N 2-Aroylanthranilamide Inhibitors of Human Factor Xa von Yee, Ying K, Tebbe, Anne Louise, Linebarger, Jared H, Beight, Douglas W, Craft, Trelia J, Gifford-Moore, Donetta, Goodson, Theodore, Herron, David K, Klimkowski, Valentine J, Kyle, Jeffrey A, Sawyer, J. Scott, Smith, Gerald F, Tinsley, Jennifer M, Towner, Richard D, Weir, Leonard, Wiley, Michael R

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High-Affinity Aptamers Selectively Inhibit Human Nonpancreatic Secretory Phospholipase A2 (hnps-PLA2) von Bridonneau, Philippe, Chang, Ying-Fon, O'Connell, Dan, Gill, Stanley C, Snyder, David W, Johnson, Lea, Goodson, Theodore, Herron, David K, Parma, David H

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Leukotriene B4 (LTB4) Receptor Antagonists: A Series of (Hydroxyphenyl)pyrazoles von Harper, Richard W, Jackson, William T, Froelich, Larry L, Boyd, Robert J, Aldridge, Timothy E, Herron, David K

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Leukotriene B4 receptor antagonists: the LY255283 series of hydroxyacetophenones von Herron, David K, Goodson, Theodore, Bollinger, Nancy G, Swanson-Bean, Dorothy, Wright, Ian G, Staten, Gilbert S, Thompson, Alan R, Froelich, Larry L, Jackson, William T

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Development of a series of phenyltetrazole leukotriene D4(LTD4) receptor antagonists von Harper, Richard W, Herron, David K, Bollinger, Nancy G, Sawyer, J. Scott, Baldwin, Ronald F, Roman, Carlos R, Rinkema, Lynn E, Fleisch, Jerome H

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New stereospecific synthetic routes to trisubstituted olefins von Corey, Elias J, Yamamoto, Hisashi, Herron, David K, Achiwa, Kazuo

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Electronic structures of cephalosporins and penicillins. 11. Parabolic relationships between antibacterial activity of cephalosporins and .beta.-lactam reactivity predicted from mo... von Boyd, Donald B, Herron, David K, Lunn, W. H. W, Spitzer, Wayne A

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Pulmonary actions of LY255283, a leukotriene B4 receptor antagonist von SILBAUGH, S. A, STENGEL, P. W, COCKERHAM, S. L, ROMAN, C. R, SAUSSY, D. L, SPAETHE, S. M, GOODSON, T. JR, HERRON, D. K, FLEISCH, J. H

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N(2)-Aroylanthranilamide inhibitors of human factor Xa von Yee, Y K, Tebbe, A L, Linebarger, J H, Beight, D W, Craft, T J, Gifford-Moore, D, Goodson, Jr, T, Herron, D K, Klimkowski, V J, Kyle, J A, Sawyer, J S, Smith, G F, Tinsley, J M, Towner, R D, Weir, L, Wiley, M R

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Solution photolysis of camphor von Agosta, William C, Herron, David K

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Convenient synthesis of 2,2-dimethylcyclobutanone von Agosta, William C, Herron, David K

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Non-Amidine-Containing 1,2-Dibenzamidobenzene Inhibitors of Human Factor Xa with Potent Anticoagulant and Antithrombotic Activity von Masters, John J, Franciskovich, Jeffry B, Tinsley, Jennifer M, Campbell, Charles, Campbell, Jack B, Craft, Trelia J, Froelich, Larry L, Gifford-Moore, Donetta S, Hay, Lynne A, Herron, David K, Klimkowski, Valentine J, Kurz, Kenneth D, Metz, James T, Ratz, Andrew M, Shuman, Robert T, Smith, Gerald F, Smith, Tommy, Towner, Richard D, Wiley, Michael R, Wilson, Alex, Yee, Ying K

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Structure-Based Design of Potent, Amidine-Derived Inhibitors of Factor Xa:  Evaluation of Selectivity, Anticoagulant Activity, and Antithrombotic Activity von Wiley, Michael R, Weir, Leonard C, Briggs, Steven, Bryan, Nancy A, Buben, John, Campbell, Charles, Chirgadze, Nickolay Y, Conrad, Richard C, Craft, Trelia J, Ficorilli, James V, Franciskovich, Jeffry B, Froelich, Larry L, Gifford-Moore, Donetta S, Goodson, Theodore, Herron, David K, Klimkowski, Valentine J, Kurz, Kenneth D, Kyle, Jeffery A, Masters, John J, Ratz, Andrew M, Milot, Guy, Shuman, Robert T, Smith, Tommy, Smith, Gerald F, Tebbe, Ann Louise, Tinsley, Jennifer M, Towner, Richard D, Wilson, Alexander, Yee, Ying K

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Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4 H-pyrrolo[1,2- b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain von Scott Sawyer, J., Beight, Douglas W., Britt, Karen S., Anderson, Bryan D., Campbell, Robert M., Goodson, Theodore, Herron, David K., Li, Hong-Yu, McMillen, William T., Mort, Nicholas, Parsons, Stephen, Smith, Edward C.R., Wagner, Jill R., Yan, Lei, Zhang, Faming, Yingling, Jonathan M.

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OVID and SUPER: two overlap programs for drug design von Hermann, R B, Herron, D K

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1,2-Dibenzamidobenzene Inhibitors of Human Factor Xa von Herron, David K, Goodson, Theodore, Wiley, Michael R, Weir, Leonard C, Kyle, Jeffrey A, Yee, Ying K, Tebbe, Ann Louise, Tinsley, Jennifer M, Mendel, David, Masters, John J, Franciskovich, Jeffry B, Sawyer, J. Scott, Beight, Douglas W, Ratz, Andrew M, Milot, Guy, Hall, Steven E, Klimkowski, Valentine J, Wikel, James H, Eastwood, Brian J, Towner, Richard D, Gifford-Moore, Donetta S, Craft, Trelia J, Smith, Gerald F

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