selective antagonist EPPTB reveals TAAR1-mediated regulatory mechanisms in dopaminergic neurons of the mesolimbic system von Bradaia, Amyaouch, Trube, Gerhard, Stalder, Henri, Norcross, Roger D, Ozmen, Laurence, Wettstein, Joseph G, Pinard, Audrée, Buchy, Danièle, Gassmann, Martin, Hoener, Marius C, Bettler, Bernhard

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Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): Discovery of EPPTB ( RO5212773) von Stalder, Henri, Hoener, Marius C., Norcross, Roger D.

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Selective GlyT1 Inhibitors: Discovery of [4-(3-Fluoro-5-trifluoromethylpyridin-2-yl)piperazin-1-yl][5-methanesulfonyl-2-((S)-2,2,2-trifluoro-1-methylethoxy)phenyl]methanone (RG1678... von Pinard, Emmanuel, Alanine, Alexander, Alberati, Daniela, Bender, Markus, Borroni, Edilio, Bourdeaux, Patrick, Brom, Virginie, Burner, Serge, Fischer, Holger, Hainzl, Dominik, Halm, Remy, Hauser, Nicole, Jolidon, Synese, Lengyel, Judith, Marty, Hans-Peter, Meyer, Thierry, Moreau, Jean-Luc, Mory, Roland, Narquizian, Robert, Nettekoven, Mathias, Norcross, Roger D, Puellmann, Bernd, Schmid, Philipp, Schmitt, Sebastien, Stalder, Henri, Wermuth, Roger, Wettstein, Joseph G, Zimmerli, Daniel

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Optimisation of imidazole compounds as selective TAAR1 agonists: Discovery of RO5073012 von Galley, Guido, Stalder, Henri, Goergler, Annick, Hoener, Marius C., Norcross, Roger D.

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Modulation of Pharmacologically Relevant Properties of Piperidine Derivatives by Functional Groups in an Equatorial or Axial β‐Position to the Amino Group von Schnider, Patrick, Dolente, Cosimo, Stalder, Henri, Martin, Rainer E., Reinmüller, Viktoria, Marty, Roman, Wyss Gramberg, Caroline, Wagner, Björn, Fischer, Holger, Alker, André M., Müller, Klaus

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Development of a Virtual Screening Method for Identification of “Frequent Hitters” in Compound Libraries von Roche, Olivier, Schneider, Petra, Zuegge, Jochen, Guba, Wolfgang, Kansy, Manfred, Alanine, Alexander, Bleicher, Konrad, Danel, Franck, Gutknecht, Eva-Maria, Rogers-Evans, Mark, Neidhart, Werner, Stalder, Henri, Dillon, Michael, Sjögren, Eric, Fotouhi, Nader, Gillespie, Paul, Goodnow, Robert, Harris, William, Jones, Phil, Taniguchi, Mikio, Tsujii, Shinji, von der Saal, Wolfgang, Zimmermann, Gerd, Schneider, Gisbert

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3‑Amido-3-aryl-piperidines: A Novel Class of Potent, Selective, and Orally Active GlyT1 Inhibitors von Pinard, Emmanuel, Alberati, Daniela, Alvarez-Sanchez, Ruben, Brom, Virginie, Burner, Serge, Fischer, Holger, Hauser, Nicole, Kolczewski, Sabine, Lengyel, Judith, Mory, Roland, Saladin, Christian, Schulz-Gasch, Tanja, Stalder, Henri

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Discovery of benzoylpiperazines as a novel class of potent and selective GlyT1 inhibitors von Pinard, Emmanuel, Alberati, Daniela, Borroni, Edilio, Fischer, Holger, Hainzl, Dominik, Jolidon, Synèse, Moreau, Jean-Luc, Narquizian, Robert, Nettekoven, Matthias, Norcross, Roger D., Stalder, Henri, Thomas, Andrew W.

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Discovery of N-(2-hydroxy-2-aryl-cyclohexyl) substituted spiropiperidines as GlyT1 antagonists with improved pharmacological profile von Ceccarelli, Simona M., Pinard, Emmanuel, Stalder, Henri, Alberati, Daniela

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Discovery of N-(2-aryl-cyclohexyl) substituted spiropiperidines as a novel class of GlyT1 inhibitors von Pinard, Emmanuel, Ceccarelli, Simona M., Stalder, Henri, Alberati, Daniela

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Tetrahydrolipstatin: Degradation products produced by human carboxyl-ester lipase von Stalder, Henri, Oesterhelt, Gottfried, Borgström, Bengt

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Joint Meeting on Medicinal Chemistry in Vienna von Martin, Rainer E., Mohr, Peter, Palmer, Wylie, Stalder, Henri

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Design and synthesis of 4-substituted-8-(2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one as a novel class of GlyT1 inhibitors: Achieving selectivity against the μ opioid and n... von Alberati, Daniela, Ceccarelli, Simona M., Jolidon, Synèse, Krafft, Eva A., Kurt, Anke, Maier, Axel, Pinard, Emmanuel, Stalder, Henri, Studer, Deborah, Thomas, Andrew W., Zimmerli, Daniel

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2-(2-Oxo-1,4-dihydro-2H-quinazolin-3-yl)- and 2-(2,2-Dioxo-1,4-dihydro-2H-2λ6-benzo[1,2,6]thiadiazin-3-yl)-N-hydroxy-acetamides as Potent and Selective Peptide Deformylase Inhibito... von Apfel, Christian, Banner, David W, Bur, Daniel, Dietz, Michel, Hubschwerlen, Christian, Locher, Hans, Marlin, Frédéric, Masciadri, Raffaello, Pirson, Wolfgang, Stalder, Henri

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Tetrahydrolipstatin: Thermal and Hydrolytic Degradation von Stalder, Henri, Schneider, Pierre R., Oesterhelt, Gottfried

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Fachtagung medizinische Chemie in Wien von Martin, Rainer E., Mohr, Peter, Palmer, Wylie, Stalder, Henri

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piperidinas aroilamino- e heteroaroilamino-substituídas como inibidores de glyt-1 von EMMANUEL PINARD, HENRI STALDER, SABINE KOLCZEWSKI

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aminas ou amido alcoóis como inibidores de glyt1 von Emmanuel Pinard, Henri Stalder, Sabine Kolczewski, Hans-Peter Marty, Robert Narquizian

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Metaboliten der 1,5‐Dihydroimidazo[2,1‐b]chinazolin‐2(3H)‐one. Synthese und Reaktionen einiger 1,5‐Dihydro‐3‐hydroxyimidazo[2,1‐b]chinazolin‐2(3H)‐one von Stalder, Henri

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Piperidine derivatives von STALDER HENRI, PINARD EMMANUEL, KOLCZEWSKI SABINE

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