A straightforward approach towards cyclic peptides via ring-closing metathesis--scope and limitations von Kazmaier, Uli, Hebach, Christina, Watzke, Anja, Maier, Sabine, Mues, Heike, Huch, Volker

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Design, Synthesis, and In Vitro and In Vivo Evaluation of Cereblon Binding Bruton’s Tyrosine Kinase (BTK) Degrader CD79b Targeted Antibody–Drug Conjugates von Zhang, Alan, Seiss, Katherine, Laborde, Laurent, Palacio-Ramirez, Sebastian, Guthy, Daniel, Lanter, Mylene, Lorber, Julien, Vulpetti, Anna, Arista, Luca, Zoller, Thomas, Radimerski, Thomas, Thoma, Claudio, Hebach, Christina, Tschantz, William R., Karpov, Alexei, Hollingworth, Gregory J., D’Alessio, Joseph A., Ferretti, Stephane, Burger, Matthew T.

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Via Ugi reactions to conformationally fixed cyclic peptidesDedicated to Professor Dr D. Seebach on the occasion of his 65th birthday von Hebach, Christina, Kazmaier, Uli

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Via Ugi reactions to conformationally fixed cyclic peptides von Hebach, Christina, Kazmaier, Uli

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Discovery of novel pyrrolidineoxy-substituted heteroaromatics as potent and selective PI3K delta inhibitors with improved physicochemical properties von Hoegenauer, Klemens, Soldermann, Nicolas, Hebach, Christina, Hollingworth, Gregory J., Lewis, Ian, von Matt, Anette, Smith, Alexander B., Wolf, Romain M., Wilcken, Rainer, Haasen, Dorothea, Burkhart, Christoph, Zécri, Frédéric

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Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors von Hoegenauer, Klemens, Soldermann, Nicolas, Stauffer, Frédéric, Furet, Pascal, Graveleau, Nadege, Smith, Alexander B, Hebach, Christina, Hollingworth, Gregory J, Lewis, Ian, Gutmann, Sascha, Rummel, Gabriele, Knapp, Mark, Wolf, Romain M, Blanz, Joachim, Feifel, Roland, Burkhart, Christoph, Zécri, Frédéric

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A straightforward approach towards glycoamino acids and glycopeptides via Pd-catalysed allylic alkylation von Krämer, Katja, Deska, Jan, Hebach, Christina, Kazmaier, Uli

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Ammonia in Ugi Reactions - Four-Component versus Six-Component Couplings von Pick, Rigobert, Bauer, Michael, Kazmaier, Uli, Hebach, Christina

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A straightforward approach towards glycoamino acids and glycopeptidesviaPd-catalysed allylic alkylation von Krämer, Katja, Deska, Jan, Hebach, Christina, Kazmaier, Uli

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Carboxylate-stabilised sulfur ylides (thetin salts) in asymmetric epoxidation for the synthesis of glycidic acids. Mechanism and implications von Aggarwal, Varinder K, Hebach, Christina

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Peptide Syntheses via Ugi Reactionswith Ammonia von Kazmaier, Uli, Hebach, Christina

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Readily Synthesized Chiral Sulfides as Reagents for Asymmetric Epoxidation von Badine, D. Michael, Hebach, Christina, Aggarwal, Varinder K.

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INTERMEDIATES OF N-(3-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)PHENYL)BENZAMIDE DERIVATIVES von ZOLLER, Thomas, MACHAUER, Rainer, ARISTA, Luca, VULPETTI, Anna, LORBER, Julien, IMBACH-WEESE, Patricia, HOLZER, Philipp, SCHMIEDEBERG, Niko, HEBACH, Christina, HOLLINGWORTH, Gregory John

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3-hydroxy-N-(3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)pyrrolidine-1-carboxamide Derivatives von ZOLLER, Thomas, MACHAUER, Rainer, ARISTA, Luca, VULPETTI, Anna, IMBACH-WEESE, Patricia, HOLZER, Philipp, SCHMIEDEBERG, Niko, HEBACH, Christina, HOLLINGWORTH, Gregory John

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N-(3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)benzamide Derivatives von ZOLLER, Thomas, MACHAUER, Rainer, ARISTA, Luca, VULPETTI, Anna, LORBER, Julien, IMBACH-WEESE, Patricia, HOLZER, Philipp, SCHMIEDEBERG, Niko, HEBACH, Christina, HOLLINGWORTH, Gregory John

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3-hydroxy-N-(3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)pyrrolidine-1-carboxamide derivatives von Arista, Luca, Hebach, Christina, Machauer, Rainer, Hollingworth, Gregory John, Holzer, Philipp, Vulpetti, Anna, Zoller, Thomas, Imbach-Weese, Patricia, Schmiedeberg, Niko

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INTERMEDIATES OF N-(3-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)PHENYL)BENZAMIDE DERIVATIVES von ZOLLER, Thomas, MACHAUER, Rainer, ARISTA, Luca, VULPETTI, Anna, LORBER, Julien, IMBACH-WEESE, Patricia, HOLZER, Philipp, SCHMIEDEBERG, Niko, HEBACH, Christina, HOLLINGWORTH, Gregory John

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Substituted pyrrolo[2,3-d]pyrimidines as Bruton's Tyrosine Kinase inhibitors von Arista, Luca, Hebach, Christina, Machauer, Rainer, Hollingworth, Gregory John, Holzer, Philipp, Vulpetti, Anna, Zoller, Thomas, Imbach-Weese, Patricia, Lorber, Julien, Schmiedeberg, Niko

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FATTY ACID-BIFUNCTIONAL DEGRADER CONJUGATES AND THEIR METHODS OF USE von Fazal, Tanzina, Hollingworth, Gregory John, Palermo, Mark Gabriel, Metcalf, III, Chester A, Zoller, Thomas, Duvadie, Rohit Kumar, Lorber, Julien, Plummer, Scott Vaughan, Li, Jialiang, Sendzik, Martin, Broennimann, Valerie, Vulpetti, Anna, Adcock, Claire, Grotzfeld, Robert Martin, Gao, Jinhai, Michael, Walter, Zhao, Liang, Usera, Aimee Richardson, Cheng, Jiashun, Guo, Fengfeng, Hebach, Christina, Zecri, Frederic, Karpov, Alexei, Jones, Darryl Brynley, Roache, James Harold, Thomas, Ranny Mathew

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3-hydroxy-N-(3-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)pyrrolidine-1-carboxamide Derivatives von Arista, Luca, Hebach, Christina, Machauer, Rainer, Hollingworth, Gregory John, Holzer, Philipp, Vulpetti, Anna, Zoller, Thomas, Imbach-Weese, Patricia, Schmiedeberg, Niko

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