Absorption, distribution, metabolism, and excretion of ticagrelor in healthy subjects von Teng, Renli, Oliver, Stuart, Hayes, Martin A, Butler, Kathleen

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Phytochemicals in Drug Discovery-A Confluence of Tradition and Innovation von Chihomvu, Patience, Ganesan, A, Gibbons, Simon, Woollard, Kevin, Hayes, Martin A

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Late‐Stage Functionalization of Histidine in Unprotected Peptides von Noisier, Anaïs F. M., Johansson, Magnus J., Knerr, Laurent, Hayes, Martin A., Drury, William J., Valeur, Eric, Malins, Lara R., Gopalakrishnan, Ranganath

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Mass Spectrometry Imaging proves differential absorption profiles of well-characterised permeability markers along the crypt-villus axis von Nilsson, Anna, Peric, Alexandra, Strimfors, Marie, Goodwin, Richard J. A., Hayes, Martin A., Andrén, Per E., Hilgendorf, Constanze

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A P450 fusion library of heme domains from Rhodococcus jostii RHA1 and its evaluation for the biotransformation of drug molecules von Kulig, Justyna K., Spandolf, Claudia, Hyde, Ralph, Ruzzini, Antonio C., Eltis, Lindsay D., Grönberg, Gunnar, Hayes, Martin A., Grogan, Gideon

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Oxalate Oxidase for In Situ H2O2‐Generation in Unspecific Peroxygenase‐Catalysed Drug Oxyfunctionalisations von Romero, Elvira, Johansson, Magnus J., Cartwright, Jared, Grogan, Gideon, Hayes, Martin A.

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Enzymatic Late‐Stage Modifications: Better Late Than Never von Romero, Elvira, Jones, Bethan S., Hogg, Bethany N., Rué Casamajo, Arnau, Hayes, Martin A., Flitsch, Sabine L., Turner, Nicholas J., Schnepel, Christian

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Oxygenating Biocatalysts for Hydroxyl Functionalisation in Drug Discovery and Development von Charlton, Sacha N., Hayes, Martin A.

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Oxalate Oxidase for In Situ H 2 O 2 -Generation in Unspecific Peroxygenase-Catalysed Drug Oxyfunctionalisations von Romero, Elvira, Johansson, Magnus J, Cartwright, Jared, Grogan, Gideon, Hayes, Martin A

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The Impact of Metagenomics on Biocatalysis von Hogg, Bethany N., Schnepel, Christian, Finnigan, James D., Charnock, Simon J., Hayes, Martin A., Turner, Nicholas J.

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Hip To Be Square: Oxetanes as Design Elements To Alter Metabolic Pathways von Toselli, Francesca, Fredenwall, Marlene, Svensson, Peder, Li, Xue-Qing, Johansson, Anders, Weidolf, Lars, Hayes, Martin A

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Cytochrome P450 Is Present in Both Ferrous and Ferric Forms in the Resting State within Intact Escherichia coli and Hepatocytes von Johnston, Wayne A., Hunter, Dominic J.B., Noble, Christopher J., Hanson, Graeme R., Stok, Jeanette E., Hayes, Martin A., De Voss, James J., Gillam, Elizabeth M.J.

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Biocatalytic Monoacylation of Symmetrical Diamines and Its Application to the Synthesis of Pharmaceutically Relevant Amides von Lubberink, Max, Schnepel, Christian, Citoler, Joan, Derrington, Sasha R, Finnigan, William, Hayes, Martin A, Turner, Nicholas J, Flitsch, Sabine L

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Regiodivergent Radical Termination for Intermolecular Biocatalytic C–C Bond Formation von Petchey, Mark R., Ye, Yuxuan, Spelling, Victor, Finnigan, James D., Gittings, Samantha, Johansson, Magnus J., Hayes, Martin A., Hyster, Todd K.

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Toward safer and more sustainable by design biocatalytic amide-bond coupling von Söderberg, Elisabeth, von Borries, Kerstin, Norinder, Ulf, Petchey, Mark, Ranjani, Ganapathy, Chavan, Swapnil, Holmquist, Hanna, Johansson, Magnus, Cotgreave, Ian, Hayes, Martin A, Fantke, Peter, Syrén, Per-Olof

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A Universal, Continuous Assay for SAM‐dependent Methyltransferases von Menke, Marian J., Schneider, Pascal, Badenhorst, Christoffel P. S., Kunzendorf, Andreas, Heinz, Florian, Dörr, Mark, Hayes, Martin A., Bornscheuer, Uwe T.

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Engineering Biocatalysts for the C−H Activation of Fatty Acids by Ancestral Sequence Reconstruction von Jones, Bethan S., Ross, Connie M., Foley, Gabriel, Pozhydaieva, Nadiia, Sharratt, Joseph W., Kress, Nico, Seibt, Lisa S., Thomson, Raine E. S., Gumulya, Yosephine, Hayes, Martin A., Gillam, Elizabeth M. J., Flitsch, Sabine L.

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Biocatalysis in Drug Design: Engineered Reductive Aminases (RedAms) Are Used to Access Chiral Building Blocks with Multiple Stereocenters von Casamajo, Arnau Rué, Yu, Yuqi, Schnepel, Christian, Morrill, Charlotte, Barker, Rhys, Levy, Colin W., Finnigan, James, Spelling, Victor, Westerlund, Kristina, Petchey, Mark, Sheppard, Robert J., Lewis, Richard J., Falcioni, Francesco, Hayes, Martin A., Turner, Nicholas J.

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Discovery and Early Clinical Development of an Inhibitor of 5‑Lipoxygenase Activating Protein (AZD5718) for Treatment of Coronary Artery Disease von Pettersen, Daniel, Broddefalk, Johan, Emtenäs, Hans, Hayes, Martin A, Lemurell, Malin, Swanson, Marianne, Ulander, Johan, Whatling, Carl, Amilon, Carl, Ericsson, Hans, Westin Eriksson, Annika, Granberg, Kenneth, Plowright, Alleyn T, Shamovsky, Igor, Dellsèn, Anita, Sundqvist, Monica, Någård, Mats, Lindstedt, Eva-Lotte

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Metabolism of Strained Rings: Glutathione S -transferase-Catalyzed Formation of a Glutathione-Conjugated Spiro-azetidine without Prior Bioactivation von Li, Xue-Qing, Grönberg, Gunnar, Bangur, Eva-Henriette, Hayes, Martin A, Castagnoli, Jr, Neal, Weidolf, Lars

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