Selection of Fragments for Kinase Inhibitor Design: Decoration Is Key von Czodrowski, Paul, Hölzemann, Günter, Barnickel, Gerhard, Greiner, Hartmut, Musil, Djordje

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Structural and Biophysical Characterization of the Syk Activation Switch von Grädler, Ulrich, Schwarz, Daniel, Dresing, Verena, Musil, Djordje, Bomke, Jörg, Frech, Matthias, Greiner, Hartmut, Jäkel, Stefan, Rysiok, Thomas, Müller-Pompalla, Dirk, Wegener, Ansgar

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Fragment-Based Discovery of New Highly Substituted 1H‑Pyrrolo[2,3‑b]- and 3H‑Imidazolo[4,5‑b]‑Pyridines as Focal Adhesion Kinase Inhibitors von Heinrich, Timo, Seenisamy, Jeyaprakashnarayanan, Emmanuvel, Lourdusamy, Kulkarni, Santosh S, Bomke, Jörg, Rohdich, Felix, Greiner, Hartmut, Esdar, Christina, Krier, Mireille, Grädler, Ulrich, Musil, Djordje

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Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling-TMS-deprotection-CuAAC sequence von Merkul, Eugen, Klukas, Fabian, Dorsch, Dieter, Grädler, Ulrich, Greiner, Hartmut E, Müller, Thomas J J

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Synthesis and Structure−Activity Relationship in a Class of Indolebutylpiperazines as Dual 5-HT1A Receptor Agonists and Serotonin Reuptake Inhibitors von Heinrich, Timo, Böttcher, Henning, Gericke, Rolf, Bartoszyk, Gerd D, Anzali, Soheila, Seyfried, Christoph A, Greiner, Hartmut E, van Amsterdam, Christoph

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Dual 5-HT1A agonists and 5-HT re-uptake inhibitors by combination of indole-butyl-amine and chromenonyl-piperazine structural elements in a single molecular entity von Heinrich, Timo, Böttcher, Henning, Schiemann, Kai, Hölzemann, Günter, Schwarz, Michael, Bartoszyk, Gerd D., van Amsterdam, Christoph, Greiner, Hartmut E., Seyfried, Christoph A.

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Indolebutylamines as Selective 5-HT1A Agonists von Heinrich, Timo, Böttcher, Henning, Bartoszyk, Gerd D, Greiner, Hartmut E, Seyfried, Christoph A, van Amsterdam, Christoph

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5-HT Reuptake Inhibitors with 5-HT1B/1D Antagonistic Activity:  A New Approach toward Efficient Antidepressants von Matzen, Lisa, van Amsterdam, Christoph, Rautenberg, Wilfried, Greiner, Hartmut E, Harting, Jürgen, Seyfried, Christoph A, Böttcher, Henning

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Discovery of novel 7-azaindoles as PDK1 inhibitors von Wucherer-Plietker, Margarita, Merkul, Eugen, Müller, Thomas J.J., Esdar, Christina, Knöchel, Thorsten, Heinrich, Timo, Buchstaller, Hans-Peter, Greiner, Hartmut, Dorsch, Dieter, Finsinger, Dirk, Calderini, Michel, Bruge, David, Grädler, Ulrich

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Fragment-based discovery of focal adhesion kinase inhibitors von Grädler, Ulrich, Bomke, Jörg, Musil, Djordje, Dresing, Verena, Lehmann, Martin, Hölzemann, Günter, Greiner, Hartmut, Esdar, Christina, Krier, Mireille, Heinrich, Timo

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Fragment-Based Discovery of New Highly Substituted 1 H -Pyrrolo[2,3- b ]- and 3 H -Imidazolo[4,5- b ]-Pyridines as Focal Adhesion Kinase Inhibitors von Heinrich, Timo, Seenisamy, Jeyaprakashnarayanan, Emmanuvel, Lourdusamy, Kulkarni, Santosh S., Bomke, Jörg, Rohdich, Felix, Greiner, Hartmut, Esdar, Christina, Krier, Mireille, Grädler, Ulrich, Musil, Djordje

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Sar of novel biarylmethylamine dopamine D4 receptor ligands von ARLT, M, BÖTTCHER, H, RIETHMÜLLER, A, SCHNEIDER, G, BARTOSZYK, G. D, GREINER, H, SEYFRIED, C. A

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2-Alkyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indoles as novel 5-HT6 receptor agonists von Mattsson, Cecilia, Sonesson, Clas, Sandahl, Anna, Greiner, Hartmut E, Gassen, Michael, Plaschke, Jörg, Leibrock, Joachim, Böttcher, Henning

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Bioisosterism of Fluorine and Cyano as Indole Substituents. Theoretical, in vitro and in vivo Examination von Heinrich, Timo, Böttcher, Henning, Bartoszyk, Gerd D., Schwartz, Harry, Anzali, Soheila, März, Joachim, Greiner, Hartmut E., Seyfried, Christoph A.

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2-Alkyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indoles as novel 5-HT6 receptor agonists von Mattsson, Cecilia, Sonesson, Clas, Sandahl, Anna, Greiner, Hartmut E., Gassen, Michael, Plaschke, Jörg, Leibrock, Joachim, Böttcher, Henning

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5-HT reuptake inhibitors with 5-HT(1B/1D) antagonistic activity: a new approach toward efficient antidepressants von Matzen, L, van Amsterdam, C, Rautenberg, W, Greiner, H E, Harting, J, Seyfried, C A, Böttcher, H

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Indolebutylamines as selective 5-HT(1A) agonists von Heinrich, Timo, Böttcher, Henning, Bartoszyk, Gerd D, Greiner, Hartmut E, Seyfried, Christoph A, Van Amsterdam, Christoph

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Indolebutylamines as Selective 5-HT 1A Agonists von Heinrich, Timo, Böttcher, Henning, Bartoszyk, Gerd D., Greiner, Hartmut E., Seyfried, Christoph A., van Amsterdam, Christoph

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Synthesis and structure--activity relationship in a class of indolebutylpiperazines as dual 5-HT(1A) receptor agonists and serotonin reuptake inhibitors von Heinrich, Timo, Böttcher, Henning, Gericke, Rolf, Bartoszyk, Gerd D, Anzali, Soheila, Seyfried, Christoph A, Greiner, Hartmut E, Van Amsterdam, Christoph

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Synthesis and Structure−Activity Relationship in a Class of Indolebutylpiperazines as Dual 5-HT 1A Receptor Agonists and Serotonin Reuptake Inhibitors von Heinrich, Timo, Böttcher, Henning, Gericke, Rolf, Bartoszyk, Gerd D., Anzali, Soheila, Seyfried, Christoph A., Greiner, Hartmut E., van Amsterdam, Christoph

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