Electrolytic Macrocyclizations: Scalable Synthesis of a Diazonamide-Based Drug Development Candidate von Ding, Hui, DeRoy, Patrick L., Perreault, Christian, Larivée, Alexandre, Siddiqui, Arshad, Caldwell, Charles G., Harran, Susan, Harran, Patrick G.

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Exploring the Boundaries of “Practical”: De Novo Syntheses of Complex Natural Product-Based Drug Candidates von Allred, Tyler K, Manoni, Francesco, Harran, Patrick G

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Unconventional Fragment Usage Enables a Concise Total Synthesis of (−)-Callyspongiolide von Manoni, Francesco, Rumo, Corentin, Li, Liubo, Harran, Patrick G.

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Cascade Synthesis of Fluorinated Spiroheterocyclic Scaffolding for Peptidic Macrobicycles von Mendoza, Angel, Bernardino, Salvador J., Dweck, Morris J., Valencia, Isabel, Evans, Declan, Tian, Haowen, Lee, William, Li, Yu, Houk, Kendall N., Harran, Patrick G.

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Indolizinylalanine Regioisomers: Tryptophan Isosteres with Bathochromic Fluorescence Emission von Cooper, Gabriella I. D., Saha, Ishika, Newman, Jacob, Shin, Ruthy H., Harran, Patrick G.

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Origin of Octafluorocyclopentene Polyelectrophilicity von Tian, Haowen, Lee, William, Li, Yuli, Dweck, Morris J., Mendoza, Angel, Harran, Patrick G., Houk, K. N.

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Template-constrained macrocyclic peptides prepared from native, unprotected precursors von Lawson, Kenneth V., Rose, Tristan E., Harran, Patrick G.

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Anomalous Chromophore Disruption Enables an Eight-Step Synthesis and Stereochemical Reassignment of (+)-Marineosin A von Feng, Zhengao, Allred, Tyler K, Hurlow, Evan E, Harran, Patrick G

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Asymmetric Organocatalysis Enables Rapid Assembly of Portimine Precursor Chains von Li, Liubo, El Khoury, Anton, Clement, Brennan O’Neil, Wu, Carolyn, Harran, Patrick G

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Cascading Auto-oxidative Biproline Guanylations Form Optically Active Dispacamide Dimers and Permit an Eight-Step Synthesis of (−)-Ageliferin von Ding, Hui, Roberts, Andrew G, Chiang, Rocky, Harran, Patrick G

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Large ring-forming alkylations provide facile access to composite macrocycles von Rose, Tristan E, Lawson, Kenneth V, Harran, Patrick G

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Computational generation of an annotated gigalibrary of synthesizable, composite peptidic macrocycles von Saha, Ishika, Dang, Eric K., Svatunek, Dennis, Houk, Kendall N., Harran, Patrick G.

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Syntheses of Atypically Fluorinated Peptidyl Macrocycles through Sequential Vinylic Substitutions von Tsunemi, Tomoyuki, Bernardino, Salvador J., Mendoza, Angel, Jones, Christopher G., Harran, Patrick G.

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Modular Access to Complex Prodiginines: Total Synthesis of (+)-Roseophilin via its 2‑Azafulvene Prototropisomer von Frederich, James H, Harran, Patrick G

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In Search of Small Molecules That Selectively Inhibit MBOAT4 von Murzinski, Emily S, Saha, Ishika, Ding, Hui, Strugatsky, David, Hollibaugh, Ryan A, Liu, Haixia, Tontonoz, Peter, Harran, Patrick G

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Template-induced macrocycle diversity through large ring-forming alkylations of tryptophan von Lawson, Kenneth V., Rose, Tristan E., Harran, Patrick G.

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A Small Molecule Smac Mimic Potentiates TRAIL- and TNFα-Mediated Cell Death von Li, Lin, Thomas, Ranny Mathew, Suzuki, Hidetaka, De Brabander, Jef K., Wang, Xiaodong, Harran, Patrick G.

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Synthetic (±)-Axinellamines Deficient in Halogen von Ding, Hui, Roberts, Andrew G., Harran, Patrick G.

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Photorearrangement of [8]-2,6-Pyridinophane N‑Oxide von Hurlow, Evan E, Lin, Janice B, Dweck, Morris J, Nuryyeva, Selbi, Feng, Zhengao, Allred, Tyler K, Houk, K. N, Harran, Patrick G

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Callyspongiolide Is a Potent Inhibitor of the Vacuolar ATPase von Fogarty, Sarah, Ouyang, Yeyun, Li, Liubo, Chen, Yu-chan, Rane, Hallie, Manoni, Francesco, Parra, Karlett J, Rutter, Jared, Harran, Patrick G

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