A novel dual glucagon‐like peptide and glucagon receptor agonist SAR425899: Results of randomized, placebo‐controlled first‐in‐human and first‐in‐patient trials von Tillner, Joachim, Posch, Maximilian G., Wagner, Frank, Teichert, Lenore, Hijazi, Youssef, Einig, Christine, Keil, Stefanie, Haack, Torsten, Wagner, Michael, Bossart, Martin, Larsen, Philip J.

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Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists von Evers, Andreas, Haack, Torsten, Lorenz, Martin, Bossart, Martin, Elvert, Ralf, Henkel, Bernd, Stengelin, Siegfried, Kurz, Michael, Glien, Maike, Dudda, Angela, Lorenz, Katrin, Kadereit, Dieter, Wagner, Michael

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Oral delivery of diabetes peptides — Comparing standard formulations incorporating functional excipients and nanotechnologies in the translational context von Lakkireddy, Harivardhan Reddy, Urmann, Matthias, Besenius, Melissa, Werner, Ulrich, Haack, Torsten, Brun, Priscilla, Alié, Jean, Illel, Brigitte, Hortala, Laurent, Vogel, Rachel, Bazile, Didier

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Running on mixed fuel‐dual agonistic approach of GLP‐1 and GCG receptors leads to beneficial impact on body weight and blood glucose control: A comparative study between mice and n... von Elvert, Ralf, Herling, Andreas W., Bossart, Martin, Weiss, Tilo, Zhang, Baohong, Wenski, Pierre, Wandschneider, Jörn, Kleutsch, Sabrina, Butty, Uwe, Kannt, Aimo, Wagner, Michael, Haack, Torsten, Evers, Andreas, Dudda, Angela, Lorenz, Martin, Keil, Stefanie, Larsen, Philip J.

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Conformational Control Inhibition of the BCR-ABL1 Tyrosine Kinase, Including the Gatekeeper T315I Mutant, by the Switch-Control Inhibitor DCC-2036 von Chan, Wayne W., Wise, Scott C., Kaufman, Michael D., Ahn, Yu Mi, Ensinger, Carol L., Haack, Torsten, Hood, Molly M., Jones, Jennifer, Lord, John W., Lu, Wei Ping, Miller, David, Patt, William C., Smith, Bryan D., Petillo, Peter A., Rutkoski, Thomas J., Telikepalli, Hanumaiah, Vogeti, Lakshminarayana, Yao, Tony, Chun, Lawrence, Clark, Robin, Evangelista, Peter, Gavrilescu, L. Cristina, Lazarides, Katherine, Zaleskas, Virginia M., Stewart, Lance J., Van Etten, Richard A., Flynn, Daniel L.

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Team Players or Opponents: Coadministration of Selective Glucagon and GLP-1 Receptor Agonists in Obese Diabetic Monkeys von Elvert, Ralf, Bossart, Martin, Herling, Andreas W, Weiss, Tilo, Zhang, Baohong, Kannt, Aimo, Wagner, Michael, Haack, Torsten, Evers, Andreas, Dudda, Angela, Keil, Stefanie, Lorenz, Martin, Lorenz, Katrin, Riz, Michela, Hennerici, Wolfgang, Larsen, Philip J

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Imaging of the Glucose-Dependent Insulinotropic Polypeptide Receptor Using a Novel Radiolabeled Peptide Rationally Designed Based on Endogenous GIP and Synthetic Exendin-4 Sequence... von Velikyan, Irina, Bossart, Martin, Haack, Torsten, Laitinen, Iina, Estrada, Sergio, Johansson, Lars, Pierrou, Stefan, Wagner, Michael, Eriksson, Olof

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Assessment of glucagon receptor occupancy by Positron Emission Tomography in non-human primates von Eriksson, Olof, Velikyan, Irina, Haack, Torsten, Bossart, Martin, Evers, Andreas, Laitinen, Iina, Larsen, Philip J., Plettenburg, Oliver, Takano, Akihiro, Halldin, Christer, Antoni, Gunnar, Johansson, Lars, Pierrou, Stefan, Wagner, Michael

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First-in-class positron emission tomography tracer for the glucagon receptor von Velikyan, Irina, Haack, Torsten, Bossart, Martin, Evers, Andreas, Laitinen, Iina, Larsen, Philip, Plettenburg, Oliver, Johansson, Lars, Pierrou, Stefan, Wagner, Michael, Eriksson, Olof

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1,1-Dioxo-5,6-dihydro-[4,1,2]oxathiazines, a novel class of 11ß-HSD1 inhibitors for the treatment of diabetes von Böhme, Thomas, Engel, Christian K., Farjot, Géraldine, Güssregen, Stefan, Haack, Torsten, Tschank, Georg, Ritter, Kurt

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Automated GMP-Compliant Production of [68Ga]Ga-DO3A-Tuna-2 for PET Microdosing Studies of the Glucagon Receptor in Humans von Wagner, Michael, Doverfjord, Johan G., Tillner, Joachim, Antoni, Gunnar, Haack, Torsten, Bossart, Martin, Laitinen, Iina, Johansson, Lars, Pierrou, Stefan, Eriksson, Olof, Velikyan, Irina

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Synthesis of Oximidine II by a Copper-Mediated Reductive Ene-Yne Macrocyclization von Schneider, Christopher M., Khownium, Kriangsak, Li, Wei, Spletstoser, Jared T., Haack, Torsten, Georg, Gunda I.

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Receptor occupancy of dual glucagon-like peptide 1/glucagon receptor agonist SAR425899 in individuals with type 2 diabetes von Eriksson, Olof, Haack, Torsten, Hijazi, Youssef, Teichert, Lenore, Tavernier, Veronique, Laitinen, Iina, Berglund, Jan Erik, Antoni, Gunnar, Velikyan, Irina, Johansson, Lars, Pierrou, Stefan, Wagner, Michael, Tillner, Joachim

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Formal Total Syntheses of the (−)-Salicylihalamides A and B From d-Glucose and l-Rhamnose von Haack, Torsten, Haack, KyoungLang, Diederich, Wibke E, Blackman, Burchelle, Roy, Subho, Pusuluri, Srinivas, Georg, Gunda I

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Drug Occupancy Assessment at the Glucose-Dependent Insulinotropic Polypeptide Receptor by Positron Emission Tomography von Eriksson, Olof, Velikyan, Irina, Haack, Torsten, Bossart, Martin, Evers, Andreas, Lorenz, Katrin, Laitinen, Iina, Larsen, Philip J, Plettenburg, Oliver, Johansson, Lars, Pierrou, Stefan, Wagner, Michael

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Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists Specifically Optimized for Multidose Formulations von Evers, Andreas, Bossart, Martin, Pfeiffer-Marek, Stefania, Elvert, Ralf, Schreuder, Herman, Kurz, Michael, Stengelin, Siegfried, Lorenz, Martin, Herling, Andreas, Konkar, Anish, Lukasczyk, Ulrike, Pfenninger, Anja, Lorenz, Katrin, Haack, Torsten, Kadereit, Dieter, Wagner, Michael

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Glucagonlike Peptide-1 Receptor Imaging in Individuals with Type 2 Diabetes von Eriksson, Olof, Velikyan, Irina, Haack, Torsten, Bossart, Martin, Laitinen, Iina, Larsen, Philip J, Berglund, Jan Erik, Antoni, Gunnar, Johansson, Lars, Pierrou, Stefan, Tillner, Joachim, Wagner, Michael

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Glucagon Like Peptide-1 receptor imaging in individuals with Type 2 Diabetes von Eriksson, Olof, Velikyan, Irina, Haack, Torsten, Bossart, Martin, Laitinen, Iina, Larsen, Philip Just, Berglund, Jan Erik, Antoni, Gunnar, Johansson, Lars, Pierrou, Stefan, Tillner, Joachim, Wagner, Michael

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Incretin combination therapy for the treatment of non‐alcoholic steatohepatitis von Kannt, Aimo, Madsen, Andreas Nygaard, Kammermeier, Claire, Elvert, Ralf, Klöckener, Tim, Bossart, Martin, Haack, Torsten, Evers, Andreas, Lorenz, Katrin, Hennerici, Wolfgang, Rocher, Corinne, Böcskei, Zsolt, Guillemot, Jean‐Claude, Mikol, Vincent, Pattou, Francois, Staels, Bart, Wagner, Michael

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Imaging of the Glucagon Receptor in Subjects with Type 2 Diabetes von Eriksson, Olof, Velikyan, Irina, Haack, Torsten, Bossart, Martin, Laitinen, Iina, Larsen, Philip J., Berglund, Jan Erik, Antoni, Gunnar, Johansson, Lars, Pierrou, Stefan, Tillner, Joachim, Wagner, Michael

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