Labelling of “Peripheral‐Type” Benzodiazepine Binding Sites in the Rat Brain By Using [3H]PK 11195, an Isoquinoline Carboxamide Derivative: Kinetic Studies and Autoradiographic Loc... von Benavides, J., Quarteronet, D., Imbault, F., Malgouris, C., Uzan, A., Renault, C., Dubroeucq, M. C., Gueremy, C., Fur, G. Le

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Riluzole Series. Synthesis and in Vivo “Antiglutamate” Activity of 6-Substituted-2-benzothiazolamines and 3-Substituted-2-imino-benzothiazolines von Jimonet, Patrick, Audiau, François, Barreau, Michel, Blanchard, Jean-Charles, Boireau, Alain, Bour, Yvette, Coléno, Marie-Annick, Doble, Adam, Doerflinger, Gilles, Do Huu, Claudine, Donat, Marie-Hélène, Duchesne, Jean Marie, Ganil, Pierre, Guérémy, Claude, Honoré, Eliane, Just, Bernard, Kerphirique, Roselyne, Gontier, Sylvie, Hubert, Philippe, Laduron, Pierre M, Le Blevec, Joseph, Meunier, Mireille, Miquet, Jean-Marie, Nemecek, Conception, Pasquet, Martine, Piot, Odile, Pratt, Jeremy, Rataud, Jean, Reibaud, Michel, Stutzmann, Jean-Marie, Mignani, Serge

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Pharmacological characterization of RP 62203, a novel 5‐hydroxytryptamine 5‐HT2 receptor antagonist von Doble, A., Girdlestone, D., Piot, O., Allam, D., Betschart, J., Boireau, A., Dupuy, A., Guérémy, C., Ménager, J., Zundel, J.L., Blanchard, J.C.

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Photoaffinity labeling of peripheral-type benzodiazepine-binding sites von DOBLE, A, FERRIS, O, BURGEVIN, M. C, MENAGER, J, UZAN, A, DUBRŒUCQ, M. C, RENAULT, C, GUEREMY, C, LE FUR, G

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A diastereoselective synthesis of girolline von COMMERCON, A, GUEREMY, C

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2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission—II: Biochemical properties von Benavides, J., Camelin, J.C., Mitrani, N., Flamand, F., Uzan, A., Legrand, J-J., Gueremy, C., Le Fur, G.

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2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission—I: Anticonvulsant properties von Mizoule, J., Meldrum, B., Mazadier, Martine, Croucher, M., Ollat, Catherine, Uzan, A., Legrand, J.-J., Gueremy, C., Le Fur, G.

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Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat von Mizoule, J., Gauthier, A., Uzan, A., Renault, C., Dubroeucq, M.C., Guéremy, C., Le Fur, G.

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Opposite effects of an agonist, RO5-4864, and an antagonist, PK 11195, of the peripheral type benzodiazepine binding sites on audiogenic seizures in DBA/2J mice von Bénavidès, J, Guilloux, F, Allam, D E, Uzan, A, Mizoule, J, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G

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PK 11195, an antagonist of peripheral benzodiazepine receptors, reduces ventricular arrhythmias during myocardial ischemia and reperfusion in the dog von Mestre, Michel, Bouetard, Giséle, Uzan, André, Gueremy, Claude, Renault, Christian, Dubroeucq, Marie-Christine, Le Fur, Gérard

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Characterization of solubilized “peripheral type” benzodiazepine binding sites from rat adrenals by using [ 3H]PK 11195, an isoquinoline carboxamide derivative von Benavides, J., Menager, J., Burgevin, M.C., Ferris, O., Uzan, A., Gueremy, C., Renault, C., Le Fur, G.

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Modulation of voltage-operated, but not receptor-operated, calcium channels in the rabbit aorta by PK 11195, an antagonist of peripheral-type benzodiazepine receptors von MESTRE, M, BELIN, C, UZAN, A, RENAULT, C, DUBRŒUCQ, M.-C, GUEREMY, C, LE FUR, G

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Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation von Mestre, M., Carriot, T., Belin, C., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C., Le Fur, G.

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Histidine modification with diethylpyrocarbonate induces a decrease in the binding of an antagonist, PK 11195, but not of an agonist, RO5-4864, of the peripheral benzodiazepine rec... von Bénavidès, J, Begassat, F, Phan, T, Tur, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G

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Stereoselective inhibition of the binding of [ 3H]PK 11195 to peripheral-type benzodiazepine binding sites by a quinolinepropanamide derivative von Dubroeucq, Marie-Christine, Bénavidès, Jesus, Doble, Adam, Guilloux, Françoise, Allam, Djamal, Vaucher, Nadine, Bertrand, Philippe, Guérémy, Claude, Renault, Christian, Uzan, Andre, Le Fur, Gérard

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Binding sites for a peripheral type benzodiazepine antagonist ([ 3H] PK 11195) in human iris von Valtier, D., Malgouris, C., Gilbert, J.-C., Guicheney, P., Uzan, A., Gueremy, C., Le Fur, G., Saraux, H., Meyer, P.

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Electrophysiological and pharmacological evidence that peripheral type benzodiazepine receptors are coupled to calcium channels in the heart von Mestre, M., Carriot, T., Belin, C., Uzan, A., Renault, C., Dubroeucq, M.C., Guérémy, C., Doble, A., Le Fur, G.

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Biochemical evidence that 2-phenyl-4[2-(4-piperidinyl) ethyl]quinoline, a quinoline derivative with pure anticonflict properties, is a partial agonist of benzodiazepine receptors von Benavides, J., Malgouris, C., Flamier, A., Tur, C., Quarteronet, D., Begassat, F., Camelin, J.-C., Uzan, A., Gueremy, C., Le Fur, G.

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Labelling of peripheral-type benzodiazepine binding sites in human brain with [ 3H]PK 11195: Anatomical and subcellular distribution von Doble, A., Malgouris, C., Daniel, M., Daniel, N., Imbault, F., Basbaum, A., Uzan, A., Guérémy, C., Le Fur, G.

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New indole derivatives as potent and selective serotonin uptake inhibitors von Malleron, Jean Luc, Gueremy, Claude, Mignani, Serge, Peyronel, Jean Francois, Truchon, Alain, Blanchard, Jean Charles, Doble, Adam, Laduron, Pierre, Piot, Odile

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