Development of an Enantioselective [3 + 2] Cycloaddition To Synthesize the Pyrrolidine Core of ABBV-3221 on Multikilogram Scale von Hartung, John, Greszler, Stephen N, Klix, Russell C, Kallemeyn, Jeffrey M

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Diastereoselective Synthesis of Pentasubstituted γ-Butyrolactones from Silyl Glyoxylates and Ketones through a Double Reformatsky Reaction von Greszler, Stephen N, Johnson, Jeffrey S

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Asymmetric Synthesis of Dihydroindanes by Convergent Alkoxide-Directed Metallacycle-Mediated Bond Formation von Greszler, Stephen N, Reichard, Holly A, Micalizio, Glenn C

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Formal Synthesis of Leustroducsin B via Reformatsky/Claisen Condensation of Silyl Glyoxylates von Greszler, Stephen N, Malinowski, Justin T, Johnson, Jeffrey S

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Enabling Asymmetric Synthesis of ABBV-3748, a Corrector Compound for the Treatment of Cystic Fibrosis von Greszler, Stephen N., Zhao, Gang, Shelat, Bhadra, Voight, Eric A.

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Enabling Synthesis of ABBV-2222, A CFTR Corrector for the Treatment of Cystic Fibrosis von Greszler, Stephen N, Shelat, Bhadra, Voight, Eric A

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Catalytic Redox-Initiated Glycolate Aldol Additions of Silyl Glyoxylates von Greszler, Stephen N, Johnson, Jeffrey S

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General Asymmetric Synthesis of Densely Functionalized Pyrrolidines via Endo -Selective [3+2] Cycloaddition of β-Quaternary-Substituted Nitroalkenes and Azomethine Ylides von Greszler, Stephen N, Zhao, Gang, Buchman, Marek, Searle, Xenia B, Liu, Bo, Voight, Eric A

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Synthesis of Substituted Cyclopropanecarboxylates via Room Temperature Palladium-Catalyzed α‑Arylation of Reformatsky Reagents von Greszler, Stephen N, Halvorsen, Geoff T, Voight, Eric A

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Fueling the Pipeline via Innovations in Organic Synthesis von Voight, Eric A, Greszler, Stephen N, Kym, Philip R

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Synthesis of the Cortistatin Pentacyclic Core by Alkoxide-Directed Metallacycle-Mediated Annulative Cross-Coupling von Aquino, Claudio, Greszler, Stephen N, Micalizio, Glenn C

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Lithioarene Cycliacylation and Pd-Catalyzed Aminoethylation/Cyclization to Access Electronically Diverse Saturated Isoquinoline Derivatives von Buchman, Marek, Farney, Elliot P, Greszler, Stephen N, Altenbach, Robert J, Gfesser, Gregory A, Voight, Eric A

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Prodrug Strategies to Improve the Solubility of the HCV NS5A Inhibitor Pibrentasvir (ABT-530) von Randolph, John T, Voight, Eric A, Greszler, Stephen N, Uno, Brice E, Newton, James N, Gleason, Kenneth M, Stolarik, DeAnne, Van Handel, Cecilia, Bow, Daniel A. J, DeGoey, David A

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Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds von Ramos, Ashley L., Goedken, Eric R., Frank, Kristine E., Argiriadi, Maria A., Bazzaz, Sana, Bian, Zhiguo, Brown, Jesse T. C., Centrella, Paolo A., Chen, Hui-Ju, Disch, Jeremy S., Donner, Pamela L., Duignan, David B., Gikunju, Diana, Greszler, Stephen N., Guié, Marie-Aude, Habeshian, Sevan, Hartl, Hajnalka E., Hein, Christopher D., Hutchins, Charles W., Jetson, Rachael, Keefe, Anthony D., Khan, Hasan, Li, Huan-Qiu, Olszewski, Allison, Ortiz Cardona, Benjamin J., Osuma, Augustine, Panchal, Sanjay C., Phelan, Ryan, Qiu, Wei, Shotwell, J. Brad, Shrestha, Anurupa, Srikumaran, Myron, Su, Zhi, Sun, Chaohong, Upadhyay, Anup K., Wood, Michael D., Wu, Haihong, Zhang, Ruijie, Zhang, Ying, Zhao, Gang, Zhu, Haizhong, Webster, Matthew P.

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Remote Stereoinduction in the Acylation of Fully Substituted Enolates: Tandem Reformatsky/Quaternary Claisen Condensations of Silyl Glyoxylates and β-Lactones von Greszler, Stephen N, Malinowski, Justin T, Johnson, Jeffrey S

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Desymmetrization of pibrentasvir for efficient prodrug synthesis von Voight, Eric A, Greszler, Stephen N, Hartung, John, Ji, Jianguo, Klix, Russell C, Randolph, John T, Shelat, Bhadra H, Waters, Jan E, DeGoey, David A

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Synthesis of ABBV-168, a 2′-Bromouridine for the Treatment of Hepatitis C von Voight, Eric A, Brown, Brian S, Greszler, Stephen N, Halvorsen, Geoff T, Zhao, Gang, Kruger, Albert W, Hartung, John, Lukin, Kirill A, Martinez, Steven R, Moschetta, Eric G, Tudesco, Michael T, Ide, Nathan D

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Synthesis of A‑9758, an Inverse Agonist of Retinoic Acid-Related Orphan Receptor γt von Marvin, Christopher C., Greszler, Stephen N., Shelat, Bhadra H., Voight, Eric A.

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Silyl Glyoxylates. Conception and Realization of Flexible Conjunctive Reagents for Multicomponent Coupling von Boyce, Gregory R, Greszler, Stephen N, Johnson, Jeffrey S, Linghu, Xin, Malinowski, Justin T, Nicewicz, David A, Satterfield, Andrew D, Schmitt, Daniel C, Steward, Kimberly M

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Stereoselective Synthesis of ABBV-992 Enabled by a Flow Diazotization and a Partial Reduction of a Pyridone von Brady, Patrick B., Harper, Kaid C., Sorensen, Bryan K., Greszler, Stephen N., Lai, Chunqiu, Florjancic, Alan S., Zhao, Gang, Shelat, Bhadra H., Storer, Gregory E., Henry, Rodger F., Hansen, T. Matthew

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