Subtype-selective sodium channel blockers promise a new era of pain research von Priest, Birgit T, Kaczorowski, Gregory J

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ProTx-II, a Selective Inhibitor of NaV1.7 Sodium Channels, Blocks Action Potential Propagation in Nociceptors von Schmalhofer, William A, Calhoun, Jeffrey, Burrows, Rachel, Bailey, Timothy, Kohler, Martin G, Weinglass, Adam B, Kaczorowski, Gregory J, Garcia, Maria L, Koltzenburg, Martin, Priest, Birgit T

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Contribution of the Tetrodotoxin-Resistant Voltage-Gated Sodium Channel NaV1.9 to Sensory Transmission and Nociceptive Behavior von Priest, Birgit T., Murphy, Beth A., Lindia, Jill A., Diaz, Carmen, Abbadie, Catherine, Ritter, Amy M., Liberator, Paul, Iyer, Leslie M., Kash, Shera F., Kohler, Martin G., Kaczorowski, Gregory J., MacIntyre, D. Euan, Martin, William J., Catterall, William A.

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The role of voltage-gated potassium channels Kv2.1 and Kv2.2 in the regulation of insulin and somatostatin release from pancreatic islets von Li, Xiaoyan Nina, Herrington, James, Petrov, Aleksandr, Ge, Lan, Eiermann, George, Xiong, Yusheng, Jensen, Mette V, Hohmeier, Hans E, Newgard, Christopher B, Garcia, Maria L, Wagner, Michael, Zhang, Bei B, Thornberry, Nancy A, Howard, Andrew D, Kaczorowski, Gregory J, Zhou, Yun-Ping

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Extracellular loop C of NPC1L1 is important for binding to ezetimibe von Weinglass, Adam B, Kohler, Martin, Schulte, Uwe, Liu, Jessica, Nketiah, Emmanuel O, Thomas, Anu, Schmalhofer, William, Williams, Brande, Bildl, Wolfgang, McMasters, Daniel R, Dai, Kevin, Beers, Lindsey, McCann, Margaret E, Kaczorowski, Gregory J, Garcia, Maria L

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Blockers of the Delayed-Rectifier Potassium Current in Pancreatic β-Cells Enhance Glucose-Dependent Insulin Secretion von Herrington, James, Zhou, Yun-Ping, Bugianesi, Randal M, Dulski, Paula M, Feng, Yue, Warren, Vivien A, Smith, McHardy M, Kohler, Martin G, Garsky, Victor M, Sanchez, Manuel, Wagner, Michael, Raphaelli, Kristin, Banerjee, Priya, Ahaghotu, Chinweze, Wunderler, Denise, Priest, Birgit T, Mehl, John T, Garcia, Maria L, McManus, Owen B, Kaczorowski, Gregory J, Slaughter, Robert S

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Characteristic time courses of cortical and medullary sodium signals measured by noninvasive 23Na-MRI in rat kidney induced by furosemide von Liu, Haiying, Zhou, Dan, Garcia, Maria L., Kohler, Martin G., Shen, Xiaolan, Williams, Donald S., Klimas, Michael T., Hargreaves, Richard J., Kaczorowski, Gregory J.

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Characterization of a New Class of Potent Inhibitors of the Voltage-Gated Sodium Channel Nav1.7 von Williams, Brande S, Felix, John P, Priest, Birgit T, Brochu, Richard M, Dai, Kefei, Hoyt, Scott B, London, Clare, Tang, Yui S, Duffy, Joseph L, Parsons, William H, Kaczorowski, Gregory J, Garcia, Maria L

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Ion channels as drug targets: the next GPCRs von Kaczorowski, Gregory J, McManus, Owen B, Priest, Birgit T, Garcia, Maria L

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Ion channels find a pathway for therapeutic success von Garcia, Maria L., Kaczorowski, Gregory J.

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Expression of Voltage-Gated Potassium Channels in Human and Rhesus Pancreatic Islets von Yan, Lizhen, Figueroa, David J, Austin, Christopher P, Liu, Yuan, Bugianesi, Randal M, Slaughter, Robert S, Kaczorowski, Gregory J, Kohler, Martin G

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Discovery of a novel class of benzazepinone Nav1.7 blockers: Potential treatments for neuropathic pain von Hoyt, Scott B., London, Clare, Gorin, David, Wyvratt, Matthew J., Fisher, Michael H., Abbadie, Catherine, Felix, John P., Garcia, Maria L., Li, Xiaohua, Lyons, Kathryn A., McGowan, Erin, MacIntyre, D. Euan, Martin, William J., Priest, Birgit T., Ritter, Amy, Smith, McHardy M., Warren, Vivien A., Williams, Brande S., Kaczorowski, Gregory J., Parsons, William H.

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Pharmacology of voltage-gated and calcium-activated potassium channels von Kaczorowski, Gregory J, Garcia, Maria L

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Discovery of Selective Small Molecule ROMK Inhibitors as Potential New Mechanism Diuretics von Tang, Haifeng, Walsh, Shawn P, Yan, Yan, de Jesus, Reynalda K, Shahripour, Aurash, Teumelsan, Nardos, Zhu, Yuping, Ha, Sookhee, Owens, Karen A, Thomas-Fowlkes, Brande S, Felix, John P, Liu, Jessica, Kohler, Martin, Priest, Birgit T, Bailey, Timothy, Brochu, Richard, Alonso-Galicia, Magdalena, Kaczorowski, Gregory J, Roy, Sophie, Yang, Lihu, Mills, Sander G, Garcia, Maria L, Pasternak, Alexander

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Targeting the inward-rectifier potassium channel ROMK in cardiovascular disease von Garcia, Maria L, Kaczorowski, Gregory J

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A pharmacologically validated, high-capacity, functional thallium flux assay for the human Ether-à-go-go related gene potassium channel von Schmalhofer, William A, Swensen, Andrew M, Thomas, Brande S, Felix, John P, Haedo, Rodolfo J, Solly, Kelli, Kiss, Laszlo, Kaczorowski, Gregory J, Garcia, Maria L

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The importance of being profiled: improving drug candidate safety and efficacy using ion channel profiling von Kaczorowski, Gregory J, Garcia, Maria L, Bode, Jacob, Hess, Stephen D, Patel, Umesh A

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Editorial overview: Cardiovascular and renal: Novel therapeutic strategies and approaches for targeting unmet cardiovascular needs von Kaczorowski, Gregory J, Pongs, Olaf

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Madin-Darby Canine Kidney II Cells: A Pharmacologically Validated System for NPC1L1-Mediated Cholesterol Uptake von Weinglass, Adam B, Köhler, Martin G, Nketiah, Emmanuel O, Liu, Jessica, Schmalhofer, William, Thomas, Anu, Williams, Brande, Beers, Lindsey, Smith, Lauren, Hafey, Mike, Bleasby, Kelly, Leone, Joseph, Tang, Yui Sing, Braun, Matthew, Ujjainwalla, Feroze, McCann, Margaret E, Kaczorowski, Gregory J, Garcia, Maria L

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Sodium Channel Blockade May Contribute to the Analgesic Efficacy of Antidepressants von Dick, Ivy E, Brochu, Richard M, Purohit, Yamini, Kaczorowski, Gregory J, Martin, William J, Priest, Birgit T

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