Highly Efficient Asymmetric Synthesis of Sitagliptin von Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J, Armstrong, Joseph D

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Highly Regioselective Synthesis of 1-Aryl-3,4,5-Substituted Pyrazoles von Gosselin, Francis, O’Shea, Paul D., Webster, Robert A., Reamer, Robert A., Tillyer, Richard D., Grabowski, Edward J.

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Synthesis of Substituted Imidazoles via Organocatalysis von Frantz, Doug E, Morency, Louis, Soheili, Arash, Murry, Jerry A, Grabowski, Edward J. J, Tillyer, Richard D

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Highly Efficient Synthesis of β-Amino Acid Derivatives via Asymmetric Hydrogenation of Unprotected Enamines von Hsiao, Yi, Rivera, Nelo R, Rosner, Thorsten, Krska, Shane W, Njolito, Eugenia, Wang, Fang, Sun, Yongkui, Armstrong, Joseph D, Grabowski, Edward J. J, Tillyer, Richard D, Spindler, Felix, Malan, Christophe

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Correction to “Highly Efficient Asymmetric Synthesis of Sitagliptin” von Hansen, Karl B, Hsiao, Yi, Xu, Feng, Rivera, Nelo, Clausen, Andrew, Kubryk, Michele, Krska, Shane, Rosner, Thorsten, Simmons, Bryon, Balsells, Jaume, Ikemoto, Nori, Sun, Yongkui, Spindler, Felix, Malan, Christophe, Grabowski, Edward J. J

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Stereoselective Formation of Carbon−Carbon Bonds via SN2-Displacement:  Synthesis of Substituted Cycloalkyl[b]indoles von Hillier, Michael C, Marcoux, Jean-François, Zhao, Dalian, Grabowski, Edward J. J, McKeown, Arlene E, Tillyer, Richard D

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First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin von Hansen, Karl B, Balsells, Jaume, Dreher, Spencer, Hsiao, Yi, Kubryk, Michele, Palucki, Michael, Rivera, Nelo, Steinhuebel, Dietrich, Armstrong, Joseph D, Askin, David, Grabowski, Edward J. J

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A Novel, Highly Enantioselective Ketone Alkynylation Reaction Mediated by Chiral Zinc Aminoalkoxides von Tan, Lushi, Chen, Cheng-yi, Tillyer, Richard D., Grabowski, Edward J. J., Reider, Paul J.

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Mechanistic Evidence for an α-Oxoketene Pathway in the Formation of β-Ketoamides/Esters via Meldrum's Acid Adducts von Xu, Feng, Armstrong, Joseph D, Zhou, George X, Simmons, Bryon, Hughes, David, Ge, Zhihong, Grabowski, Edward J. J

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Stereoselective Carbon−Carbon Bond Formation via the Mitsunobu Displacement of Chiral Secondary Benzylic Alcohols von Hillier, Michael C, Desrosiers, Jean-Nicolas, Marcoux, Jean-François, Grabowski, Edward J. J

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Asymmetric Synthesis of a Prostaglandin D2 Receptor Antagonist von Campos, Kevin R, Journet, Michel, Lee, Sandra, Grabowski, Edward J. J, Tillyer, Richard D

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Synthesis of α-Amido Ketones via Organic Catalysis:  Thiazolium-Catalyzed Cross-Coupling of Aldehydes with Acylimines von Murry, Jerry A, Frantz, Doug E, Soheili, Arash, Tillyer, Richard, Grabowski, Edward J. J, Reider, Paul J

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Asymmetric Hydrogenation of N-Sulfonylated-α-dehydroamino Acids:  Toward the Synthesis of an Anthrax Lethal Factor Inhibitor von Shultz, C. Scott, Dreher, Spencer D, Ikemoto, Norihiro, Williams, J. Michael, Grabowski, Edward J. J, Krska, Shane W, Sun, Yongkui, Dormer, Peter G, DiMichele, Lisa

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Oxidation of Primary Alcohols to Carboxylic Acids with Sodium Chlorite Catalyzed by TEMPO and Bleach von Zhao, Mangzhu, Li, Jing, Mano, Eiichi, Song, Zhiguo, Tschaen, David M, Grabowski, Edward J. J, Reider, Paul J

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Practical Asymmetric Synthesis of a Potent PDE4 Inhibitor via Stereoselective Enolate Alkylation of a Chiral Aryl−Heteroaryl Secondary Tosylate von O'Shea, Paul D, Chen, Cheng-yi, Chen, Weirong, Dagneau, Philippe, Frey, Lisa F, Grabowski, Edward J. J, Marcantonio, Karen M, Reamer, Robert A, Tan, Lushi, Tillyer, Richard D, Roy, Amélie, Wang, Xin, Zhao, Dalian

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Lithium Ephedrate-Mediated Addition of a Lithium Acetylide to a Ketone:  Solution Structures and Relative Reactivities of Mixed Aggregates Underlying the High Enantioselectivities... von Thompson, Andrew, Corley, Edward G, Huntington, Martha F, Grabowski, Edward J. J, Remenar, Julius F, Collum, David B

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Practical Asymmetric Synthesis of a Potent Cathepsin K Inhibitor. Efficient Palladium Removal Following Suzuki Coupling von Chen, Cheng-yi, Dagneau, Philippe, Grabowski, Edward J. J, Oballa, Renata, O'Shea, Paul, Prasit, Peppi, Robichaud, Joël, Tillyer, Rich, Wang, Xin

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Highly Diastereoselective Heterogeneously Catalyzed Hydrogenation of Enamines for the Synthesis of Chiral β-Amino Acid Derivatives von Ikemoto, Norihiro, Tellers, David M, Dreher, Spencer D, Liu, Jinchu, Huang, Angie, Rivera, Nelo R, Njolito, Eugenia, Hsiao, Yi, McWilliams, J. Christopher, Williams, J. Michael, Armstrong, Joseph D, Sun, Yongkui, Mathre, David J, Grabowski, Edward J. J, Tillyer, Richard D

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Practical Synthesis of a Potent Hepatitis C Virus RNA Replication Inhibitor von Bio, Matthew M, Xu, Feng, Waters, Marjorie, Williams, J. Michael, Savary, Kimberly A, Cowden, Cameron J, Yang, Chunhua, Buck, Elizabeth, Song, Zhiguo J, Tschaen, David M, Volante, R. P, Reamer, Robert A, Grabowski, Edward J. J

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Practical Asymmetric Synthesis of Aprepitant, a Potent Human NK-1 Receptor Antagonist, via a Stereoselective Lewis Acid-Catalyzed Trans Acetalization Reaction von Zhao, Matthew M, McNamara, James M, Ho, Guo-Jie, Emerson, Khateeta M, Song, Zhiguo J, Tschaen, David M, Brands, Karel M. J, Dolling, Ulf-H, Grabowski, Edward J. J, Reider, Paul J, Cottrell, Ian F, Ashwood, Michael S, Bishop, Brian C

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