Application of BRET to monitor ligand binding to GPCRs von Stoddart, Leigh A, Johnstone, Elizabeth K M, Wheal, Amanda J, Goulding, Joëlle, Robers, Matthew B, Machleidt, Thomas, Wood, Keith V, Hill, Stephen J, Pfleger, Kevin D G

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Ligand-Directed Labeling of the Adenosine A1 Receptor in Living Cells von Comeo, Eleonora, Goulding, Joëlle, Lin, Chia-Yang, Groenen, Marleen, Woolard, Jeanette, Kindon, Nicholas D., Harwood, Clare R., Platt, Simon, Briddon, Stephen J., Kilpatrick, Laura E., Scammells, Peter J., Hill, Stephen J., Kellam, Barrie

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Small-Molecule Fluorescent Ligands for the CXCR4 Chemokine Receptor von Dekkers, Sebastian, Caspar, Birgit, Goulding, Joëlle, Kindon, Nicholas D., Kilpatrick, Laura E., Stoddart, Leigh A., Briddon, Stephen J., Kellam, Barrie, Hill, Stephen J., Stocks, Michael J.

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Advances in the application of fluorescence correlation spectroscopy to study detergent purified and encapsulated membrane proteins von Stoddart, Leigh A, Goulding, Joëlle, Briddon, Stephen J

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Subtype selective fluorescent ligands based on ICI 118,551 to study the human β2‐adrenoceptor in CRISPR/Cas9 genome‐edited HEK293T cells at low expression levels von Goulding, Joëlle, Mistry, Sarah J., Soave, Mark, Woolard, Jeanette, Briddon, Stephen J., White, Carl W., Kellam, Barrie, Hill, Stephen J.

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A high-affinity, cis-on photoswitchable beta blocker to optically control β2-adrenergic receptors in vitro and in vivo von Shi, Shuang, Zheng, Yang, Goulding, Joëlle, Marri, Silvia, Lucarini, Laura, Konecny, Benjamin, Sgambellone, Silvia, Villano, Serafina, Bosma, Reggie, Wijtmans, Maikel, Briddon, Stephen J., Zarzycka, Barbara A., Vischer, Henry F., Leurs, Rob

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Detection of genome‐edited and endogenously expressed G protein‐coupled receptors von Soave, Mark, Stoddart, Leigh A., White, Carl W., Kilpatrick, Laura E., Goulding, Joëlle, Briddon, Stephen J., Hill, Stephen J.

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Acylation of the Incretin Peptide Exendin-4 Directly Impacts Glucagon-Like Peptide-1 Receptor Signaling and Trafficking von Lucey, Maria, Ashik, Tanyel, Marzook, Amaara, Wang, Yifan, Goulding, Joëlle, Oishi, Atsuro, Broichhagen, Johannes, Hodson, David J., Minnion, James, Elani, Yuval, Jockers, Ralf, Briddon, Stephen J., Bloom, Stephen R., Tomas, Alejandra, Jones, Ben

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Application of Fluorescent Purinoceptor Antagonists for Bioluminescence Resonance Energy Transfer Assays and Fluorescent Microscopy von Soave, Mark, Goulding, Joëlle, Markus, Robert, Hill, Stephen J., Stoddart, Leigh A.

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Plasma membrane preassociation drives β-arrestin coupling to receptors and activation von Grimes, Jak, Koszegi, Zsombor, Lanoiselée, Yann, Miljus, Tamara, O’Brien, Shannon L., Stepniewski, Tomasz M., Medel-Lacruz, Brian, Baidya, Mithu, Makarova, Maria, Mistry, Ravi, Goulding, Joëlle, Drube, Julia, Hoffmann, Carsten, Owen, Dylan M., Shukla, Arun K., Selent, Jana, Hill, Stephen J., Calebiro, Davide

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CRISPR/Cas9-mediated generation and analysis of N terminus polymorphic models of β2AR in isogenic hPSC-derived cardiomyocytes von Kondrashov, Alexander, Mohd Yusof, Nurul A.N., Hasan, Alveera, Goulding, Joëlle, Kodagoda, Thusharika, Hoang, Duc M., Vo, Nguyen T.N., Melarangi, Tony, Dolatshad, Nazanin, Gorelik, Julia, Hill, Stephen J., Harding, Sian E., Denning, Chris

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Ligand-Directed Labeling of the Adenosine A 1 Receptor in Living Cells von Comeo, Eleonora, Goulding, Joëlle, Lin, Chia-Yang, Groenen, Marleen, Woolard, Jeanette, Kindon, Nicholas D, Harwood, Clare R, Platt, Simon, Briddon, Stephen J, Kilpatrick, Laura E, Scammells, Peter J, Hill, Stephen J, Kellam, Barrie

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A novel and selective fluorescent ligand for the study of adenosine A2B receptors von Patera, Foteini, Mistry, Sarah J., Kindon, Nicholas D., Comeo, Eleonora, Goulding, Joelle, Kellam, Barrie, Kilpatrick, Laura E., Franks, Hester, Hill, Stephen J.

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The use of fluorescence correlation spectroscopy to monitor cell surface β2‐adrenoceptors at low expression levels in human embryonic stem cell‐derived cardiomyocytes and fibroblas... von Goulding, Joëlle, Kondrashov, Alexander, Mistry, Sarah J., Melarangi, Tony, Vo, Nguyen T.N., Hoang, Duc M., White, Carl W., Denning, Chris, Briddon, Stephen J., Hill, Stephen J.

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Plasma membrane preassociation drives β-arrestin coupling to receptors and activation von Grimes, Jak, Koszegi, Zsombor, Lanoiselée, Yann, Miljus, Tamara, O'Brien, Shannon L, Stepniewski, Tomasz Maciej, 1988, Medel Lacruz, Brian, Baidya, Mithu, Makarova, Maria, Mistry, Ravi, Goulding, Joëlle, Drube, Julia, Hoffmann, Carsten, Owen, Dylan M, Shukla, Arun K, Selent, Jana, Hill, Stephen J, Calebiro, Davide

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Probing expression of E-selectin using CRISPR-Cas9-mediated tagging with HiBiT in human endothelial cells von Ogrodzinski, Lydia, Platt, Simon, Goulding, Joelle, Alexander, Cameron, Farr, Tracy D., Woolard, Jeanette, Hill, Stephen J., Kilpatrick, Laura E.

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A high-affinity, cis-on photoswitchable beta blocker to optically control β 2 -adrenergic receptors in vitro and in vivo von Shi, Shuang, Zheng, Yang, Goulding, Joëlle, Marri, Silvia, Lucarini, Laura, Konecny, Benjamin, Sgambellone, Silvia, Villano, Serafina, Bosma, Reggie, Wijtmans, Maikel, Briddon, Stephen J, Zarzycka, Barbara A, Vischer, Henry F, Leurs, Rob

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CRISPR/Cas9-mediated generation and analysis of N terminus polymorphic models of β 2 AR in isogenic hPSC-derived cardiomyocytes von Kondrashov, Alexander, Mohd Yusof, Nurul A N, Hasan, Alveera, Goulding, Joëlle, Kodagoda, Thusharika, Hoang, Duc M, Vo, Nguyen T N, Melarangi, Tony, Dolatshad, Nazanin, Gorelik, Julia, Hill, Stephen J, Harding, Sian E, Denning, Chris

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Characterisation of endogenous A2A and A2B receptor-mediated cyclic AMP responses in HEK 293 cells using the GloSensor™ biosensor: Evidence for an allosteric mechanism of action fo... von Goulding, Joelle, May, Lauren T., Hill, Stephen J.

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Single molecule binding of a ligand to a G-protein-coupled receptor in real time using fluorescence correlation spectroscopy, rendered possible by nano-encapsulation in styrene mal... von Grime, Rachael L, Goulding, Joelle, Uddin, Romez, Stoddart, Leigh A, Hill, Stephen J, Poyner, David R, Briddon, Stephen J, Wheatley, Mark

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